Target Details
| UniProt AC | P22894 |
|---|---|
| Gene Symbol | MMP8 |
| Protein Name | Neutrophil collagenase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 934
- Clinical molecules 624
- Avg pChEMBL 7.65
Active Molecules (934)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MUMVNZHARHFSLP
|
6.8 | IC50 | 4 | Yes | |
AHDPJKYOQXMDIX
|
6.8 | Ki | 4 | — | |
MWKXYRJSVHPPLM
|
6.8 | IC50 | 4 | — | |
RWKJBOMUESGCBO
|
6.8 | Ki | 4 | Yes | |
BQOKFWQTKSZIMZ
|
6.8 | Ki | 4 | Yes | |
FHCIUVTYGHWJQR
|
6.8 | IC50 | 4 | — | |
ZJVORNZEDYXDGJ
|
6.8 | IC50 | 4 | — | |
BNPWNBBKUMLEJM
|
6.8 | Ki | 5 | Yes | |
CADOQGNFDXDEHI
|
6.8 | IC50 | 5 | Yes | |
MCDVAZDSWVFMGC
|
6.8 | Ki | 2 | Yes | |
UACUZULRKJKTHE
|
6.8 | Ki | 5 | Yes | |
UVGAWIJNBYCHSP
|
6.8 | Ki | 9 | Yes | |
UVGAWIJNBYCHSP
|
6.8 | Ki | 7 | — | |
KHCZZISCPQRODX
|
6.8 | Ki | 6 | Yes | |
RLDMWDXYWMJUAA
|
6.8 | IC50 | 3 | — | |
AGAWLHFJRLMKEA
|
6.7 | IC50 | 3 | — | |
KOVQMCGGWATESY
|
6.7 | Ki | 7 | — | |
KOVQMCGGWATESY
|
6.7 | Ki | 7 | — | |
MBHDDZHFZICCLX
|
6.7 | IC50 | 4 | — | |
NKVKCTYTQNQNIH
|
6.7 | Ki | 3 | — | |
VCIBNYPUVKINDS
|
6.7 | Ki | 5 | Yes | |
VTRJTXRAOIMSTL
|
6.7 | Ki | 8 | Yes | |
WJWOJAKOSRCFKB
|
6.7 | Ki | 9 | Yes | |
GISWZMJMNJMSEO
|
6.7 | IC50 | 4 | — | |
LEDMBBYIVRLZAS
|
6.7 | Ki | 9 | Yes | |
OURSUJYXZLSVCS
|
6.7 | IC50 | 5 | — | |
UIGGXLFLAQCMAY
|
6.7 | IC50 | 6 | Yes | |
XJLATMLVMSFZBN
|
6.7 | Ki | 5 | Yes | |
XJLATMLVMSFZBN
|
6.7 | Ki | 9 | Yes | |
ARFFCGXUOISSHZ
|
6.7 | IC50 | 6 | Yes | |
BLIQFUCBRCDFAI
|
6.7 | Ki | 5 | Yes | |
GINBTQGVSPUJLE
|
6.7 | Ki | 9 | Yes | |
HPPQTJSDCSGPAX
|
6.7 | IC50 | 4 | — | |
IEFFRLNSCQIVBY
|
6.7 | Ki | 5 | Yes | |
IGJDRNDPWLIBBQ
|
6.7 | IC50 | 2 | Yes | |
JROHDXNIWULULC
|
6.7 | IC50 | 2 | Yes | |
MVRHXCGLUWVMKH
|
6.7 | IC50 | 7 | Yes | |
OIZMOMFOLNBXHF
|
6.7 | IC50 | 9 | — | |
QULPHXDROMVDLR
|
6.7 | Ki | 3 | — | |
QULPHXDROMVDLR
|
6.7 | Ki | 4 | Yes | |
RNMKXQYTQJNJRJ
|
6.7 | IC50 | 3 | Yes | |
VOORVZQGMACJHE
|
6.7 | IC50 | 2 | Yes | |
XNEFJXZBPPJDHR
|
6.7 | IC50 | 2 | Yes | |
YZKJTNXYLZWHHJ
|
6.7 | IC50 | 7 | Yes | |
KDDWLGBIYXTPJG
|
6.7 | Ki | 5 | — | |
KNOYHJOPRUTPSQ
|
6.7 | Ki | 7 | — | |
LHURUBKIFBZDNZ
|
6.7 | Ki | 3 | — | |
FHMXFHQIBLHDDW
|
6.7 | IC50 | 3 | — | |
WOIMZSMDPIJLFO
|
6.7 | Ki | 9 | Yes | |
BODLESUVCQEUII
|
6.7 | Ki | 7 | Yes |