Target Details
| UniProt AC | P22894 |
|---|---|
| Gene Symbol | MMP8 |
| Protein Name | Neutrophil collagenase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 934
- Clinical molecules 624
- Avg pChEMBL 7.65
Active Molecules (934)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FITYZYBFZVGBBP
|
7.0 | IC50 | 4 | — | |
FXZROVPZUUATHR
|
7.0 | IC50 | 4 | Yes | |
HIPJPXVTDXVQMU
|
7.0 | IC50 | 3 | — | |
JCUTWTFOYUXMPS
|
7.0 | Ki | 10 | Yes | |
JSQUVSOHRBZSNW
|
7.0 | IC50 | 5 | Yes | |
RDMHVXDIUPIFCJ
|
7.0 | IC50 | 4 | — | |
SQWPYMHLYZKCEN
|
7.0 | IC50 | 3 | — | |
WOIMZSMDPIJLFO
|
7.0 | Ki | 7 | Yes | |
YXPTXTBBPCLWPQ
|
7.0 | IC50 | 4 | — | |
LIIRZRQVACDFBI
|
7.0 | Ki | 3 | — | |
SOPBVJMMDDZVHQ
|
7.0 | IC50 | 3 | — | |
AUIKJLRMPLDORG
|
6.9 | Ki | 10 | Yes | |
HCTHWCGSCVVHLJ
|
6.9 | Ki | 3 | — | |
PTJXSKQZLWNDNB
|
6.9 | IC50 | 5 | Yes | |
CSAFQHHGNGUQOL
|
6.9 | Ki | 10 | Yes | |
LYRSIRCJLISGFP
|
6.9 | IC50 | 4 | — | |
SQWPYMHLYZKCEN
|
6.9 | IC50 | 3 | — | |
DJZNIZCARKSSDE
|
6.9 | IC50 | 9 | Yes | |
FBDOWURNGYMLPJ
|
6.9 | Ki | 7 | — | |
SJTWWQWUAQAYAB
|
6.9 | IC50 | 4 | Yes | |
USQRZPGPLTUIHD
|
6.9 | Ki | 7 | Yes | |
CPWMZTRXCCYTDM
|
6.9 | Ki | 10 | Yes | |
DRCOOMXUPYOBBW
|
6.9 | IC50 | 4 | — | |
FYYNAVTYOZPHTC
|
6.9 | IC50 | 4 | Yes | |
SUEBJDNLBVTIQP
|
6.9 | Ki | 10 | Yes | |
VOESHNWTIDIZCL
|
6.9 | Ki | 10 | Yes | |
WQCYWYOJQMZTMB
|
6.9 | IC50 | 4 | — | |
WWQRPJINVFSPDF
|
6.9 | Ki | 10 | Yes | |
CQGUKDZSAPDCJL
|
6.9 | IC50 | 5 | Yes | |
FGDQQAHGMHOQDV
|
6.9 | Ki | 5 | Yes | |
HJAQLIVSMXUHPV
|
6.9 | Ki | 10 | Yes | |
HSQOMGXZKXTHEM
|
6.9 | IC50 | 5 | Yes | |
QNKSDDQPRLWOEC
|
6.9 | Ki | 5 | Yes | |
WGPPHZNYJYFKJE
|
6.9 | IC50 | 3 | — | |
MXFJZXDWWXHXMV
|
6.9 | Ki | 7 | — | |
BRXGWWVUCIZYMM
|
6.9 | IC50 | 4 | — | |
BRXGWWVUCIZYMM
|
6.9 | IC50 | 5 | Yes | |
WLZISXXOYYGJNT
|
6.9 | Ki | 12 | Yes | |
BKFQDASOGHAZSH
|
6.8 | IC50 | 3 | — | |
FVPQYGSYGOKFLW
|
6.8 | Ki | 5 | Yes | |
JNMYIRAUFFFDQS
|
6.8 | IC50 | 4 | Yes | |
KJDPTHLLJDQIMT
|
6.8 | IC50 | 5 | Yes | |
OXTBPBSHWBJLJN
|
6.8 | IC50 | 4 | — | |
WBIKMXRYXWFRCE
|
6.8 | IC50 | 4 | Yes | |
XLKQIIIKETWLMI
|
6.8 | Ki | 8 | — | |
ZVQKPPCVSXIXMD
|
6.8 | IC50 | 5 | — | |
GGMOCOYDYRCVAH
|
6.8 | IC50 | 5 | Yes | |
GRRDUDJQILRRES
|
6.8 | Ki | 4 | — | |
JXHAGXRDZALSLG
|
6.8 | Ki | 9 | Yes | |
VGXSIAPPDJZRCX
|
6.8 | IC50 | 3 | — |