Target Details
| UniProt AC | P22894 |
|---|---|
| Gene Symbol | MMP8 |
| Protein Name | Neutrophil collagenase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 934
- Clinical molecules 624
- Avg pChEMBL 7.65
Active Molecules (934)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CSLRMNGVKPXZNV
|
7.1 | IC50 | 2 | Yes | |
CSLRMNGVKPXZNV
|
7.1 | IC50 | 2 | — | |
MTRATHZFTCSGDT
|
7.1 | Ki | 6 | Yes | |
PBUKUIIGUHJHQN
|
7.1 | IC50 | 3 | Yes | |
QESMDPOTHYLJHG
|
7.1 | IC50 | 3 | Yes | |
SMWGTYPHHCYQHB
|
7.1 | IC50 | 5 | Yes | |
QASGJNZOZYCBGQ
|
7.1 | IC50 | 4 | — | |
RTBMLCLTYAPKIF
|
7.1 | IC50 | 5 | Yes | |
SQWPYMHLYZKCEN
|
7.1 | IC50 | 3 | — | |
UHXPHVQOXYZQPP
|
7.1 | IC50 | 4 | — | |
YXQWYGVDVQBPGA
|
7.1 | IC50 | 4 | — | |
XATUMTIXUAJCSA
|
7.1 | IC50 | 4 | — | |
OREDIHYKGISTDR
|
7.1 | IC50 | 6 | Yes | |
WDDBBBHPBMFFCX
|
7.1 | IC50 | 4 | — | |
LKFQHLGPHTXZAW
|
7.0 | IC50 | 3 | Yes | |
MOQWSIABFGAXAW
|
7.0 | IC50 | 5 | — | |
PTYZKNZXNKWTEF
|
7.0 | IC50 | 6 | Yes | |
QPLQAMVXCDXOBY
|
7.0 | IC50 | 5 | — | |
YXXPZIJDDIJKDH
|
7.0 | IC50 | 2 | Yes | |
XLNFBXKUCFOQRQ
|
7.0 | IC50 | 4 | — | |
BZKOBLHHRSTMHO
|
7.0 | Ki | 4 | — | |
PXQPONLRTWLOTH
|
7.0 | Ki | 3 | — | |
USIMDPVZFWUXPH
|
7.0 | IC50 | 6 | Yes | |
UBHBDSABSVVUTP
|
7.0 | IC50 | 4 | — | |
PLJKONSYASWBHO
|
7.0 | Ki | 3 | — | |
WPGRSZLFNFYSPR
|
7.0 | IC50 | 4 | — | |
BBPLRBWLQWBZIO
|
7.0 | IC50 | 5 | — | |
CAXAOIUOYPZXNV
|
7.0 | IC50 | 3 | Yes | |
FIPYOKGRSDJCAR
|
7.0 | IC50 | 9 | Yes | |
HHJKMUMZRIIHIU
|
7.0 | Ki | 10 | Yes | |
IKFXTEOZLBAELL
|
7.0 | Ki | 3 | — | |
IKFXTEOZLBAELL
|
7.0 | Ki | 3 | Yes | |
LRMGKWDRORXPRE
|
7.0 | IC50 | 5 | Yes | |
MSWCSYXARJOPRA
|
7.0 | IC50 | 3 | Yes | |
OUZMHHWAGJCAFA
|
7.0 | Ki | 8 | — | |
OVICMAJBKGLSNC
|
7.0 | IC50 | 5 | Yes | |
QROXNPLBULDOSL
|
7.0 | IC50 | 4 | Yes | |
VVEIZVKRPYJCPP
|
7.0 | IC50 | 6 | Yes | |
VWOQXPBXOWHZCH
|
7.0 | IC50 | 6 | Yes | |
ZNTBEHZFMMNDRG
|
7.0 | IC50 | 5 | Yes | |
ZUZHAPXKYPLQLC
|
7.0 | Ki | 5 | Yes | |
SUFSQYXUPYDFHG
|
7.0 | IC50 | 7 | Yes | |
WATNMHGSJFUVDX
|
7.0 | Ki | 5 | Yes | |
VSJBIWYXNLUPIE
|
7.0 | Ki | 10 | Yes | |
WGTWQHQAJDQPEW
|
7.0 | IC50 | 5 | Yes | |
WLZQVNRDQZYTID
|
7.0 | Ki | 6 | — | |
ZWFVIZGPXNSREN
|
7.0 | IC50 | 3 | — | |
LWNWGJXWKYGLPU
|
7.0 | IC50 | 5 | Yes | |
STWCTQDLUUVJMC
|
7.0 | Ki | 10 | Yes | |
AGSXHHFUSDGSSO
|
7.0 | IC50 | 5 | Yes |