Target Details
| UniProt AC | P22894 |
|---|---|
| Gene Symbol | MMP8 |
| Protein Name | Neutrophil collagenase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 934
- Clinical molecules 624
- Avg pChEMBL 7.65
Active Molecules (934)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CLXRDURJLYSMHZ
|
7.3 | IC50 | 5 | Yes | |
LEIFVUOVYOUZFH
|
7.3 | IC50 | 5 | Yes | |
VCJGVCZITQVJET
|
7.3 | Ki | 4 | — | |
HYNBRLICGGQMNU
|
7.3 | IC50 | 3 | Yes | |
QRQKVQCDKFEWSW
|
7.3 | IC50 | 4 | — | |
RMAHZBKEPFXNHG
|
7.3 | IC50 | 3 | Yes | |
XUDODBAIOYVRJQ
|
7.3 | IC50 | 3 | Yes | |
AEOWLQGPNGMHBP
|
7.3 | Ki | 8 | — | |
PYNQNWZHEDOQHX
|
7.3 | IC50 | 6 | Yes | |
FJEJHTFPLBTMLO
|
7.3 | IC50 | 4 | — | |
NITYDPDXAAFEIT
|
7.3 | Ki | 3 | Yes | |
ZCRWOWSOWBMWGI
|
7.3 | IC50 | 8 | Yes | |
WNEMBEALMHVXIK
|
7.3 | IC50 | 7 | — | |
BITKIWWLFIJBSD
|
7.2 | IC50 | 3 | — | |
UGWWPGUNBPZMDD
|
7.2 | IC50 | 5 | — | |
HBDUXNUNXGZOCK
|
7.2 | IC50 | 4 | — | |
HSWKOBISGMUSTR
|
7.2 | IC50 | 5 | Yes | |
QHDIXGPUTSAIJX
|
7.2 | IC50 | 2 | Yes | |
UALGGXUAYUNRBS
|
7.2 | Ki | 7 | Yes | |
QSOYTCHABFMDFV
|
7.2 | IC50 | 10 | Yes | |
YDZNXFWUNLRONX
|
7.2 | IC50 | 4 | — | |
BTMGFNYLYGWAKT
|
7.2 | Ki | 7 | Yes | |
DOLJQSYCTYZCTL
|
7.2 | IC50 | 3 | Yes | |
HTUSESRFPXTJLY
|
7.2 | IC50 | 4 | — | |
OVSRFDPZSPSZOR
|
7.2 | IC50 | 4 | — | |
UWVBDELWTIGPFO
|
7.2 | Ki | 4 | — | |
SJWYFGLDVUQIEF
|
7.2 | Ki | 4 | — | |
UTCUOTDVVXFCLJ
|
7.2 | IC50 | 6 | Yes | |
ZMGHGYMGQVMACZ
|
7.2 | Ki | 3 | — | |
DJDWNBGULWSWLG
|
7.2 | IC50 | 4 | — | |
LBKCSOUMADYGHM
|
7.2 | IC50 | 6 | Yes | |
DUYNKLSOEWBOEC
|
7.2 | IC50 | 3 | — | |
WVAIZSKMOMDPIT
|
7.2 | IC50 | 6 | Yes | |
DLMROZSTEBHAOO
|
7.2 | IC50 | 4 | Yes | |
JVBFGGAYMSJQBZ
|
7.2 | IC50 | 7 | Yes | |
MQOPTJYOSJSPJX
|
7.2 | IC50 | 3 | Yes | |
QDCHOZJXLIIHRT
|
7.2 | Ki | 5 | Yes | |
RDHFQPOQGDBVBN
|
7.2 | IC50 | 3 | Yes | |
BGJNPKHDPBUJSP
|
7.1 | IC50 | 4 | — | |
CPYISUHNJGFCRY
|
7.1 | Ki | 3 | — | |
CTCTZAXBKWKMKL
|
7.1 | Ki | 3 | — | |
HHHAELOQIYTSIY
|
7.1 | IC50 | 6 | Yes | |
UAFRGDNTZQMZFA
|
7.1 | Ki | 5 | Yes | |
UKNOMEZXDWRZAF
|
7.1 | Ki | 4 | Yes | |
JRPLACGAMSWTCU
|
7.1 | Ki | 5 | Yes | |
CWDYQHCEZVYJNX
|
7.1 | Ki | 3 | — | |
DFWYBNIMFAUWSX
|
7.1 | IC50 | 5 | Yes | |
FOVJQTLLPOZKTJ
|
7.1 | IC50 | 4 | — | |
ZRSUANFPMBWMDZ
|
7.1 | Ki | 4 | Yes | |
CLKXWRSURRSEKP
|
7.1 | IC50 | 3 | Yes |