Target Details
| UniProt AC | P22894 |
|---|---|
| Gene Symbol | MMP8 |
| Protein Name | Neutrophil collagenase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 934
- Clinical molecules 624
- Avg pChEMBL 7.65
Active Molecules (934)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZTJUBPXNBSLSGL
|
7.5 | IC50 | 6 | Yes | |
BBMXXNQSDJPWKT
|
7.5 | IC50 | 4 | — | |
JXZUMXBHWMKALL
|
7.5 | Ki | 3 | — | |
WSGLDBYEABEDRD
|
7.5 | Ki | 4 | Yes | |
RGDPJPMKLABBRX
|
7.5 | Ki | 7 | Yes | |
BVNHOVTUHKATJL
|
7.5 | Ki | 4 | Yes | |
YDCLZJDJJGSFJZ
|
7.5 | Ki | 7 | Yes | |
LQNSDZTXHZUYKJ
|
7.5 | IC50 | 10 | Yes | |
MIKGRMSWGTVOSA
|
7.5 | IC50 | 4 | — | |
OPYOHFRGHGDNSJ
|
7.5 | Ki | 7 | Yes | |
RTYBJAJUHLHGKX
|
7.5 | IC50 | 3 | — | |
VMOSDDURWLNMNG
|
7.5 | IC50 | 8 | Yes | |
UGLOKYALFGIDPP
|
7.4 | IC50 | 4 | Yes | |
DOZFSSIRRROWRF
|
7.4 | Ki | 3 | — | |
FWPVXLYOKAOERT
|
7.4 | IC50 | 8 | Yes | |
FWPVXLYOKAOERT
|
7.4 | IC50 | 4 | — | |
RPWGPXSVYLHGRZ
|
7.4 | IC50 | 7 | Yes | |
ZYIMYAJZHPOFQU
|
7.4 | Ki | 4 | — | |
SQWPYMHLYZKCEN
|
7.4 | IC50 | 3 | — | |
HHSADBHNZPOTTJ
|
7.4 | Ki | 7 | Yes | |
RSGNLFDKUXBMRT
|
7.4 | IC50 | 4 | — | |
YDDMVPLLJTZTQL
|
7.4 | Ki | 7 | Yes | |
CXPHOOFGGKZGTC
|
7.4 | Ki | 5 | — | |
DNFKKMGBEKWECE
|
7.4 | IC50 | 3 | Yes | |
HXTKAAOSFRMCEF
|
7.4 | IC50 | 3 | Yes | |
QFZXMLHPDXMOKQ
|
7.4 | IC50 | 3 | Yes | |
QHRUJPVXLYJUEM
|
7.4 | IC50 | 6 | Yes | |
ZGTPJERIIBYCFG
|
7.4 | Ki | 5 | Yes | |
ZKKQCCSHBYRQHR
|
7.4 | IC50 | 3 | Yes | |
QQGKYSPTORHWNZ
|
7.4 | Ki | 6 | — | |
CZWJAEJHLBICAX
|
7.4 | IC50 | 3 | — | |
KQIFSUSWYMDFOC
|
7.4 | IC50 | 5 | Yes | |
DQDPBMDGDOPPLK
|
7.4 | Ki | 7 | Yes | |
FTQOZDRDOVWSBK
|
7.4 | Ki | 3 | — | |
IHPUTEIJIZVYPC
|
7.4 | Ki | 7 | Yes | |
PHKLGXHLOXCURO
|
7.4 | IC50 | 4 | — | |
IMQVPVWXNJYVAS
|
7.3 | IC50 | 7 | Yes | |
LHVGXRIIQBVWQU
|
7.3 | Ki | 4 | Yes | |
UJKQHAYQMMMAEL
|
7.3 | Ki | 7 | Yes | |
YXSJVSGLVWXWOT
|
7.3 | IC50 | 4 | — | |
NGVKQXNJLILPFW
|
7.3 | IC50 | 3 | — | |
UKASSNVNXOWYDK
|
7.3 | IC50 | 4 | — | |
DRWHINQPSIPRHF
|
7.3 | IC50 | 6 | Yes | |
GWHSSPUFNDIEEQ
|
7.3 | Ki | 4 | — | |
HBXKDLPCZIPLFA
|
7.3 | IC50 | 3 | — | |
APJIPTNFOKEMIQ
|
7.3 | IC50 | 5 | Yes | |
GIEQMQWMJSYCKB
|
7.3 | Ki | 5 | — | |
MOPRTFSMCQNUCT
|
7.3 | IC50 | 5 | Yes | |
OEHVKBKRRIUTOR
|
7.3 | Ki | 6 | Yes | |
PZJJOMPTIHBGHO
|
7.3 | IC50 | 8 | Yes |