Target Details
| UniProt AC | P22735 |
|---|---|
| Gene Symbol | TGM1 |
| Protein Name | Protein-glutamine gamma-glutamyltransferase K |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00927 (Transglut_C) PF01841 (Transglut_core) PF00868 (Transglut_N) |
Summary
- Multi-target molecules 6
- Clinical molecules 0
- Avg pChEMBL 6.6
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (6)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OYEOXFZRVNDRKZ
|
7.7 | IC50 | 5 | — | |
CSSMDVCMCOVRQK
|
6.6 | IC50 | 2 | — | |
IJUIDQWNEGTWHT
|
6.6 | IC50 | 2 | — | |
IJUIDQWNEGTWHT
|
6.6 | IC50 | 2 | — | |
WZTJFZPMDNYCQU
|
6.0 | IC50 | 2 | — | |
AUAPVOQGBUKHMB
|
6.0 | IC50 | 3 | — |