Target Details
| UniProt AC | P22607 |
|---|---|
| Gene Symbol | FGFR3 |
| Protein Name | Fibroblast growth factor receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21165 (FGFR3_TM) PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,742
- Clinical molecules 64
- Avg pChEMBL 7.75
KEGG Pathways (13)
- Bladder cancer
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- MAPK signaling pathway
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (15)
- Achondroplasia
- Bladder cancer
- CATSHL syndrome
- Colorectal cancer
- Crouzon syndrome
- Epidermal nevus
- FGFR3-related short limb skeletal dysplasia
- Hypochondroplasia
- Lacrimo-auriculo-dento-digital syndrome
- Muenke syndrome
- Multiple myeloma
- SADDAN
- Syndromic craniosynostoses
- Testicular cancer
- Thanatophoric dysplasia
Active Molecules (2,742)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ADIFMZOOUGSSJC
|
8.4 | IC50 | 2 | — | |
AHEDUFSEDRFCTH
|
8.4 | IC50 | 4 | — | |
AQMXONPVPCMPJM
|
8.4 | IC50 | 3 | — | |
DKRZSFVZVVDUSO
|
8.4 | IC50 | 3 | — | |
DMLTXHUJLWPBCX
|
8.4 | IC50 | 2 | — | |
JXYINBAIXJFWAT
|
8.4 | IC50 | 2 | — | |
MKWMZFFPSBNEIH
|
8.4 | IC50 | 2 | — | |
SQEZUHWWJYSRDG
|
8.4 | IC50 | 5 | — | |
UBGBIWLWSXCNJS
|
8.4 | IC50 | 3 | — | |
ULZYEHHPVPISAH
|
8.4 | IC50 | 3 | — | |
ZAGOLYGHOPAHBL
|
8.4 | IC50 | 5 | — | |
CVOXIJBPYJDKHX
|
8.4 | IC50 | 3 | — | |
GXQZPCUWRYWOJV
|
8.4 | IC50 | 5 | — | |
HOVGKFRLRAHOTJ
|
8.4 | IC50 | 2 | — | |
HOVGKFRLRAHOTJ
|
8.4 | IC50 | 2 | — | |
IWBVZILESKBVJL
|
8.4 | IC50 | 6 | — | |
JTSGAAOXUAIUDH
|
8.4 | IC50 | 3 | — | |
JXBOABQESNSJLD
|
8.4 | IC50 | 2 | — | |
LVRQYRWZIOHHHF
|
8.4 | IC50 | 3 | — | |
MSLILZFULYZLIC
|
8.4 | IC50 | 3 | — | |
NEFZUKWATFHFMM
|
8.4 | IC50 | 2 | — | |
ONAZMIGCNRUYHT
|
8.4 | IC50 | 5 | — | |
PYUIBNGQBBAKFO
|
8.4 | IC50 | 7 | Yes | |
STINDBVFOPRZHE
|
8.4 | IC50 | 8 | Yes | |
ULHGAQSVFPOUDY
|
8.4 | Ki | 43 | — | |
VSNIYTDVOFCOEC
|
8.4 | IC50 | 3 | — | |
AVEPOXATJSYYGP
|
8.4 | IC50 | 5 | — | |
JLQHGFULSVHTBJ
|
8.4 | IC50 | 5 | — | |
VSYUQTBCUZLAOX
|
8.4 | IC50 | 2 | — | |
ZEONLOUAYWYGAS
|
8.4 | IC50 | 5 | — | |
AOWDVVUJNHATEM
|
8.4 | IC50 | 2 | — | |
DIYIEVQNIORQDL
|
8.4 | IC50 | 5 | — | |
HLRBIOMHENPNQT
|
8.4 | IC50 | 3 | — | |
IVLJANLBHIHWHO
|
8.4 | IC50 | 3 | — | |
JVHRYVZNKJPNLU
|
8.4 | IC50 | 5 | — | |
KONCHEYJKNSRJF
|
8.4 | IC50 | 5 | — | |
KTQNUSVVKAQAIV
|
8.4 | IC50 | 5 | — | |
KUZHPFCXWLMAPX
|
8.4 | IC50 | 2 | — | |
LBHGMHQDOQYTKT
|
8.4 | IC50 | 5 | — | |
MXMLJQCILGAGCP
|
8.4 | IC50 | 5 | — | |
SAHTUCUOJHIHGN
|
8.4 | IC50 | 5 | — | |
TUSASGMHAWDHSE
|
8.4 | IC50 | 2 | — | |
UVZKMOOZAKKRIJ
|
8.4 | IC50 | 3 | — | |
YEZYAHOOMMGLLK
|
8.4 | IC50 | 2 | — | |
YHZPMSJNFKZYKK
|
8.4 | IC50 | 2 | — | |
ZZDKMIARNROCNG
|
8.4 | IC50 | 2 | — | |
AVHLETMOCLYGNK
|
8.4 | IC50 | 5 | — | |
HXVGNVTWSKNDRL
|
8.4 | Kd | 4 | — | |
JGAIVBOWNPLAHY
|
8.4 | IC50 | 3 | — | |
MLGJITMGHIKNFO
|
8.4 | IC50 | 3 | — |