Target Details
| UniProt AC | P22607 |
|---|---|
| Gene Symbol | FGFR3 |
| Protein Name | Fibroblast growth factor receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21165 (FGFR3_TM) PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,742
- Clinical molecules 64
- Avg pChEMBL 7.75
KEGG Pathways (13)
- Bladder cancer
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- MAPK signaling pathway
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (15)
- Achondroplasia
- Bladder cancer
- CATSHL syndrome
- Colorectal cancer
- Crouzon syndrome
- Epidermal nevus
- FGFR3-related short limb skeletal dysplasia
- Hypochondroplasia
- Lacrimo-auriculo-dento-digital syndrome
- Muenke syndrome
- Multiple myeloma
- SADDAN
- Syndromic craniosynostoses
- Testicular cancer
- Thanatophoric dysplasia
Active Molecules (2,742)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YXTHFMOUCQZVJH
|
8.5 | IC50 | 3 | — | |
ZMOFBPPQIDCDSS
|
8.5 | IC50 | 2 | — | |
KBUPLPBZRGPNCS
|
8.5 | IC50 | 2 | — | |
CMMUVKONDKDCCZ
|
8.5 | IC50 | 5 | — | |
HRADXFDASOBMPX
|
8.5 | IC50 | 5 | — | |
IYEGFWFCWTYSJJ
|
8.5 | IC50 | 2 | — | |
MOCIDOAKXWFCQL
|
8.5 | IC50 | 3 | — | |
YICOQNPWMAVVBP
|
8.5 | IC50 | 2 | — | |
YXAFWGPKAAKJHB
|
8.5 | IC50 | 5 | — | |
CJCVUUCNWAXQGA
|
8.5 | IC50 | 2 | — | |
GIGLTKPRJFVONN
|
8.5 | IC50 | 3 | — | |
GUEZCEZQFMVREH
|
8.5 | IC50 | 3 | — | |
GXMSDNOAHZYMEL
|
8.5 | IC50 | 3 | — | |
HUVVCRLMPWOMJX
|
8.5 | IC50 | 4 | — | |
IOKLYXDNQOPONA
|
8.5 | IC50 | 3 | — | |
JWOIPGHVEJHTRG
|
8.5 | IC50 | 3 | — | |
MJHFGTHWKHPARC
|
8.5 | IC50 | 5 | — | |
NDGPXJXKLJJMFA
|
8.5 | IC50 | 3 | — | |
OIYSNFGRVNTTAT
|
8.5 | IC50 | 3 | — | |
RAJGOCXFXWSCOM
|
8.5 | IC50 | 2 | — | |
SUIFLKARRVDMQC
|
8.5 | IC50 | 3 | — | |
TVWOUPGUUIDZET
|
8.5 | IC50 | 6 | — | |
XORAFTFBTLPFEB
|
8.5 | IC50 | 3 | — | |
XSDFUOBWKCWNGD
|
8.5 | IC50 | 3 | — | |
XSDFUOBWKCWNGD
|
8.5 | IC50 | 3 | — | |
CCWQRQKDZAKBBS
|
8.4 | IC50 | 6 | — | |
CUMCBEDCPQGOTJ
|
8.4 | IC50 | 5 | — | |
OVZKBAUSZIANJA
|
8.4 | IC50 | 5 | — | |
PMMLVRGAMVZREV
|
8.4 | IC50 | 2 | — | |
PVFMVTVHNHARHS
|
8.4 | IC50 | 2 | — | |
QNXOYMFBIACDSL
|
8.4 | IC50 | 5 | — | |
BDOBQLMVWBQCBI
|
8.4 | IC50 | 2 | — | |
BROOSVBOLOJDTF
|
8.4 | IC50 | 2 | — | |
GUKLJPKDSMJFLV
|
8.4 | IC50 | 2 | — | |
IVQXFJNVCKJIHX
|
8.4 | IC50 | 5 | — | |
KTMMZCLUGNPLAT
|
8.4 | IC50 | 3 | — | |
MCMNKYIBBPTWOO
|
8.4 | IC50 | 2 | — | |
RKRDVEBFGMJINX
|
8.4 | IC50 | 2 | — | |
SBMUXRCSESCJIO
|
8.4 | IC50 | 3 | — | |
XWQJWMKIXLWIOD
|
8.4 | IC50 | 2 | — | |
ZAPUSNWRFJVSGX
|
8.4 | IC50 | 5 | — | |
ZDKQWJFWRHHHFH
|
8.4 | IC50 | 2 | — | |
ZHYANUGGYRLICR
|
8.4 | IC50 | 2 | — | |
CMQBIUKGSMOTTQ
|
8.4 | IC50 | 5 | — | |
HGUINYREMXETNK
|
8.4 | IC50 | 2 | — | |
JJGLWOVGLSSBEB
|
8.4 | IC50 | 2 | — | |
MJZLZOOCTKZOHS
|
8.4 | IC50 | 5 | — | |
PFTPAJNMFJOUIG
|
8.4 | IC50 | 5 | — | |
SNPGOAWRSCUFOV
|
8.4 | IC50 | 3 | — | |
YYJUTCUEPVSXDM
|
8.4 | IC50 | 3 | — |