Target Details
| UniProt AC | P22607 |
|---|---|
| Gene Symbol | FGFR3 |
| Protein Name | Fibroblast growth factor receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21165 (FGFR3_TM) PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,742
- Clinical molecules 64
- Avg pChEMBL 7.75
KEGG Pathways (13)
- Bladder cancer
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- MAPK signaling pathway
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (15)
- Achondroplasia
- Bladder cancer
- CATSHL syndrome
- Colorectal cancer
- Crouzon syndrome
- Epidermal nevus
- FGFR3-related short limb skeletal dysplasia
- Hypochondroplasia
- Lacrimo-auriculo-dento-digital syndrome
- Muenke syndrome
- Multiple myeloma
- SADDAN
- Syndromic craniosynostoses
- Testicular cancer
- Thanatophoric dysplasia
Active Molecules (2,742)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RVPLSKAFRYMLOL
|
8.6 | IC50 | 2 | — | |
VCNJSFBAEBDCKK
|
8.6 | IC50 | 5 | — | |
XZJZLDYVCVKCSJ
|
8.6 | IC50 | 2 | — | |
MDPWQSCOLLDWIY
|
8.6 | IC50 | 5 | — | |
ODRNQGSZGLHVGG
|
8.6 | IC50 | 5 | — | |
BTGLYCHFNHKNDV
|
8.6 | IC50 | 3 | — | |
DCPPHIRTTFNMRQ
|
8.6 | IC50 | 2 | — | |
FDEHCJCKFIQBIS
|
8.6 | IC50 | 5 | — | |
ZZWQREKFRLSPQU
|
8.6 | IC50 | 2 | — | |
BBPYINKOTXNMRZ
|
8.6 | IC50 | 3 | — | |
FOJJNIMHMLFIAZ
|
8.6 | IC50 | 3 | — | |
IATQVFKHNZFWTF
|
8.6 | IC50 | 3 | — | |
IGXJTXDPMDXZJZ
|
8.6 | IC50 | 3 | — | |
JMKKBCYATYJNOD
|
8.6 | IC50 | 2 | — | |
KPDFFUWYNAEXCW
|
8.6 | IC50 | 3 | — | |
NKNHEZFIUHHBJX
|
8.6 | IC50 | 3 | — | |
NTPSXOIFCGNPHC
|
8.6 | IC50 | 3 | — | |
OTMSABHPICNCIU
|
8.6 | IC50 | 3 | — | |
QYDBJBJRCCHDBO
|
8.6 | IC50 | 3 | — | |
QYOSWBKWDQWBJG
|
8.6 | IC50 | 3 | — | |
SRFTVRWDQRUZRY
|
8.6 | IC50 | 3 | — | |
YZRSMWKLOJZVAD
|
8.6 | IC50 | 4 | — | |
ZHVCDQSIPKIGFZ
|
8.6 | IC50 | 2 | — | |
ACCSYFAQPQXJJO
|
8.6 | Ki | 6 | — | |
BNBYLDDIZKKPGC
|
8.6 | IC50 | 2 | — | |
GDNZRDDMJFKRAA
|
8.6 | IC50 | 2 | — | |
GWCJUEKQORIUTJ
|
8.6 | IC50 | 5 | — | |
HVIMAXORBAESDU
|
8.6 | IC50 | 2 | — | |
KNACLJBHKVSTDL
|
8.6 | Ki | 40 | — | |
PSRCAUFYXJRQBZ
|
8.6 | IC50 | 2 | — | |
QSZLOMZJWAOHPQ
|
8.6 | IC50 | 5 | — | |
QXCPWDLEEJRGER
|
8.6 | IC50 | 2 | — | |
WITKAEIQNFPTFS
|
8.6 | IC50 | 5 | — | |
WNUXYTTWUXBQMA
|
8.6 | IC50 | 2 | — | |
WZOJLYYGKNGLLO
|
8.6 | IC50 | 3 | — | |
YIQKRGSTCNRKES
|
8.6 | Ki | 6 | — | |
ZXCGLXZIDVIUJE
|
8.6 | IC50 | 5 | — | |
BQCQOBOXMZWHQL
|
8.6 | IC50 | 5 | — | |
BSKSTNRPIFLDMV
|
8.6 | IC50 | 2 | — | |
CCVQDAVSKDENJO
|
8.6 | IC50 | 2 | — | |
JNYVQUCEMBFJBC
|
8.6 | IC50 | 2 | — | |
MIWWARHIDNFXAZ
|
8.6 | IC50 | 6 | — | |
WNJVGIPJSLLBIX
|
8.6 | IC50 | 2 | — | |
WOGGKLMGFJJKGY
|
8.6 | IC50 | 5 | — | |
YMXQQOATOHFDLF
|
8.6 | IC50 | 5 | — | |
AHQPYHJCFNYNTJ
|
8.6 | IC50 | 3 | — | |
ODMSZDHTOWFRQP
|
8.6 | IC50 | 2 | — | |
QIXCNXNXARCJIU
|
8.6 | IC50 | 3 | — | |
RAMCMRRBGWIDLK
|
8.6 | IC50 | 8 | Yes | |
SBXJWOVGQTVLAE
|
8.6 | IC50 | 3 | — |