Target Details
| UniProt AC | P22460 |
|---|---|
| Gene Symbol | KCNA5 |
| Protein Name | Potassium voltage-gated channel subfamily A member 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02214 (BTB_2) PF00520 (Ion_trans) |
Summary
- Multi-target molecules 61
- Clinical molecules 0
- Avg pChEMBL 6.6
Associated Diseases (1)
Active Molecules (61)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XWQQRPSPOBDJLI
|
9.8 | IC50 | 40 | — | |
JJAWGNIQEOFURP
|
8.1 | IC50 | 2 | — | |
QPWKXYZJANVPLF
|
8.0 | IC50 | 3 | — | |
JSYVMXAHYRRFOQ
|
7.2 | IC50 | 2 | — | |
KINMYBBFQRSVLL
|
7.1 | IC50 | 6 | — | |
QWDDTOMERKJRQK
|
7.0 | IC50 | 2 | — | |
KITYXUGKWPDMSJ
|
7.0 | IC50 | 2 | — | |
MGRLWDRGBXQTMU
|
6.8 | IC50 | 3 | — | |
OXMXIXOKIIPOHL
|
6.8 | IC50 | 3 | — | |
UVMFWOKHXJEFRH
|
6.8 | IC50 | 3 | — | |
HUIYSGLQEYEPFI
|
6.8 | IC50 | 3 | — | |
INIUOCWMNJACSH
|
6.8 | IC50 | 2 | — | |
NOHWRIQJLRSUIM
|
6.8 | IC50 | 3 | — | |
QEBMMPNMOSIUKC
|
6.8 | IC50 | 3 | — | |
POZWXIVIAWFJOK
|
6.7 | IC50 | 2 | — | |
ALRMPHHZEVRXDO
|
6.7 | IC50 | 3 | — | |
KYZSDKSHODHMRD
|
6.7 | IC50 | 3 | — | |
MTYFDEYZRYWPAI
|
6.7 | IC50 | 2 | — | |
PZCYDKAVVVBKMA
|
6.7 | IC50 | 3 | — | |
MZIJPPLPZPKXEU
|
6.6 | IC50 | 2 | — | |
WOOQITHNVSFGKK
|
6.6 | IC50 | 3 | — | |
UWRHVPLUUPPQMY
|
6.6 | IC50 | 3 | — | |
BORCZNYMAGQEGS
|
6.6 | IC50 | 3 | — | |
MMCFFZBMJHBWGM
|
6.6 | IC50 | 2 | — | |
CFHAMFAFVWBLDT
|
6.5 | IC50 | 3 | — | |
DBNPCPDXYFIRGT
|
6.5 | IC50 | 2 | — | |
MTYFDEYZRYWPAI
|
6.5 | IC50 | 2 | — | |
NYSHIPDVLVFILL
|
6.5 | IC50 | 3 | — | |
XAMJZICIEQIVJK
|
6.5 | IC50 | 2 | — | |
HWHJLTXOSDACJN
|
6.5 | IC50 | 3 | — | |
BJRMDIIIWVVQSZ
|
6.5 | IC50 | 2 | — | |
QYICUUHLNRBIMS
|
6.5 | IC50 | 2 | — | |
KSZRMQOUHDNLBY
|
6.5 | IC50 | 2 | — | |
DUVMSDROOBQDDF
|
6.5 | IC50 | 2 | — | |
CMPJAGCXBOHFAF
|
6.4 | IC50 | 3 | — | |
YSNROTHUHBZNDE
|
6.4 | IC50 | 2 | — | |
HVZWHAHDNKMEHJ
|
6.4 | IC50 | 2 | — | |
OTSKYWVPYJRLJF
|
6.4 | IC50 | 2 | — | |
QEXPFDNRGMLZPW
|
6.4 | IC50 | 3 | — | |
GVOVTRIALVWKIK
|
6.4 | IC50 | 2 | — | |
CHQGILRQWLEPAK
|
6.4 | IC50 | 3 | — | |
HKOFDZHMCAXCDS
|
6.4 | IC50 | 3 | — | |
IWAGYADOEPALTO
|
6.4 | IC50 | 2 | — | |
GIZJXCZQTLNBNJ
|
6.3 | IC50 | 2 | — | |
NUGSUIAMNWUMFA
|
6.3 | IC50 | 2 | — | |
GAKQXDXJHZRVJC
|
6.3 | IC50 | 2 | — | |
USFGZWPSRSTMGP
|
6.3 | IC50 | 2 | — | |
CBJBDCXJQSNMSZ
|
6.3 | IC50 | 3 | — | |
MRFUMRJHDPXIAR
|
6.3 | IC50 | 2 | — | |
XSVYDPIWGWYQKU
|
6.3 | IC50 | 2 | — |