Target Details
| UniProt AC | P22314 |
|---|---|
| Gene Symbol | UBA1 |
| Protein Name | Ubiquitin-like modifier-activating enzyme 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF16191 (E1_4HB) PF16190 (E1_FCCH) PF09358 (E1_UFD) PF00899 (ThiF) PF10585 (UBA_E1_SCCH) |
Summary
- Multi-target molecules 30
- Clinical molecules 0
- Avg pChEMBL 6.92
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (30)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
APJANDAVERUGOK
|
7.3 | IC50 | 3 | — | |
BOWWVKGCWVBOPJ
|
7.3 | IC50 | 3 | — | |
CZHBRQKRUJRKSV
|
7.3 | IC50 | 3 | — | |
GOIILOFEIUREBR
|
7.3 | IC50 | 3 | — | |
GYMPFXKRZWRPJD
|
7.3 | IC50 | 3 | — | |
HRSBOFUEDXCMBN
|
7.3 | IC50 | 3 | — | |
HSQSIEIPMZGXCI
|
7.3 | IC50 | 3 | — | |
KXDNYXMFALGPJQ
|
7.3 | IC50 | 3 | — | |
MEJVUUFUGXLCAU
|
7.3 | IC50 | 3 | — | |
NUWGQHGWOIICDS
|
7.3 | IC50 | 3 | — | |
ODKUMVDDQKSXSW
|
7.3 | IC50 | 3 | — | |
OLUBTRMMTMIAJS
|
7.3 | IC50 | 3 | — | |
PFIDQKRZRSMQRC
|
7.3 | IC50 | 3 | — | |
PRMHMOBKWNLIGR
|
7.3 | IC50 | 3 | — | |
RIJVXPSEZBXRBU
|
7.3 | IC50 | 3 | — | |
XBFRVNJVAJTVDV
|
7.3 | IC50 | 3 | — | |
XDXPCTFDYJMPLE
|
7.3 | IC50 | 3 | — | |
YKXAYIRICCLAQW
|
7.3 | IC50 | 3 | — | |
FRCOPIZAOPFHPW
|
7.2 | IC50 | 3 | — | |
MWKSRKSEWLRPBL
|
7.0 | Kd | 1075 | — | |
TZTRUHFXPVXWRD
|
6.3 | IC50 | 4 | — | |
LFVBSFKFKWBKIB
|
6.3 | IC50 | 3 | — | |
MZWFHZDGVLGVPB
|
6.3 | IC50 | 3 | — | |
PUMBIYVFJUTEPW
|
6.3 | IC50 | 3 | — | |
PZOHRIXWJNTDKJ
|
6.3 | IC50 | 3 | — | |
RKNTWRDJZIZVTB
|
6.3 | IC50 | 3 | — | |
SYJSIKOBBZVNJB
|
6.3 | IC50 | 3 | — | |
UPUSYLJKPLQMMM
|
6.3 | IC50 | 3 | — | |
XWEFXSGIPCOLJG
|
6.3 | IC50 | 3 | — | |
YYXBNLJWLAQNCX
|
6.3 | IC50 | 3 | — |