Target Details
| UniProt AC | P22102 |
|---|---|
| Gene Symbol | GART |
| Protein Name | Trifunctional purine biosynthetic protein adenosine-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00586 (AIRS) PF02769 (AIRS_C) PF00551 (Formyl_trans_N) PF01071 (GARS_A) PF02843 (GARS_C) PF02844 (GARS_N) |
Summary
- Multi-target molecules 46
- Clinical molecules 2
- Avg pChEMBL 7.98
KEGG Pathways (4)
Active Molecules (46)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PFJDDXFAFBODCL
|
10.1 | IC50 | 3 | — | |
WKIIITBMPWEWKZ
|
9.8 | IC50 | 3 | — | |
JWZBILLJZHUAOY
|
9.2 | IC50 | 5 | — | |
VEKHZPVGFDPVJG
|
9.0 | IC50 | 5 | — | |
VMGGIKVXYOZFJO
|
9.0 | IC50 | 4 | — | |
WMTFSFGBNBUALY
|
8.9 | IC50 | 5 | — | |
FSOJIOKMUXQEMI
|
8.8 | IC50 | 5 | — | |
QLSVPQAGJDLITE
|
8.7 | IC50 | 5 | — | |
JXLUUFBZGXCZRH
|
8.7 | Ki | 2 | — | |
STQPVYHCDNSBIJ
|
8.7 | IC50 | 5 | — | |
JBVKQLSCSCXKDY
|
8.7 | IC50 | 2 | — | |
UNSSSMUKJOLMJV
|
8.6 | IC50 | 5 | — | |
HHKAOUMVRGSKLS
|
8.5 | Ki | 2 | — | |
ADFLVKAWSSGDBU
|
8.5 | IC50 | 3 | — | |
WMBYSCVMFMNUQV
|
8.5 | IC50 | 5 | — | |
OUMBMSSXXWAJDS
|
8.3 | IC50 | 3 | — | |
RMEHPWHLFJJYTB
|
8.3 | IC50 | 5 | — | |
CEPQCJFDTGQKDN
|
8.2 | IC50 | 4 | — | |
CETGJKHDVDGZDA
|
8.1 | IC50 | 3 | — | |
QSMJJFQXDNSFGZ
|
8.1 | Ki | 2 | — | |
FBOZXECLQNJBKD
|
8.0 | IC50 | 16 | — | |
NDBHIBYSTUVPRS
|
7.9 | IC50 | 3 | — | |
UFNWIIALSMNORN
|
7.9 | IC50 | 5 | — | |
KVBZUTNKUVNMNN
|
7.9 | IC50 | 3 | — | |
CYOOKDIMCAPJGV
|
7.8 | IC50 | 5 | — | |
JXLUUFBZGXCZRH
|
7.8 | Ki | 2 | — | |
UPENPAQNDNZZTP
|
7.7 | IC50 | 5 | — | |
VFYUKZOGWIMWFW
|
7.7 | IC50 | 5 | — | |
FTSMBZFBGMYYIT
|
7.6 | IC50 | 5 | — | |
HHKAOUMVRGSKLS
|
7.5 | Ki | 2 | — | |
ZGMCQEIDLHETAQ
|
7.5 | Ki | 2 | — | |
RPXDQPDLDPKBHG
|
7.5 | Ki | 3 | Yes | |
HPAURQDCTYKMTE
|
7.5 | IC50 | 4 | — | |
KXVFDIDJQOTBSL
|
7.5 | Ki | 2 | — | |
NQIQMFMYULMMGE
|
7.5 | Ki | 2 | — | |
KYKDIKFUXRYZEH
|
7.4 | IC50 | 3 | — | |
WBXPDJSOTKVWSJ
|
7.4 | IC50 | 10 | Yes | |
ZUQBAQVRAURMCL
|
7.2 | Ki | 2 | — | |
JLRJTWXBYRMGEB
|
7.2 | IC50 | 4 | — | |
TUFOXZXSKHTTLC
|
7.1 | IC50 | 4 | — | |
IPVCAFLQSKTPOY
|
7.0 | IC50 | 3 | — | |
YSCGOYFEYRSGDL
|
7.0 | IC50 | 3 | — | |
ZUPOLQOQXJAAHS
|
7.0 | IC50 | 3 | — | |
MWKSRKSEWLRPBL
|
6.9 | Kd | 1075 | — | |
RQAHNHUMMCUWMX
|
6.5 | Ki | 3 | — | |
CCSMRAGPBNANSC
|
6.4 | Ki | 3 | — |