Target Details
| UniProt AC | P22001 |
|---|---|
| Gene Symbol | KCNA3 |
| Protein Name | Potassium voltage-gated channel subfamily A member 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02214 (BTB_2) PF00520 (Ion_trans) |
Summary
- Multi-target molecules 156
- Clinical molecules 0
- Avg pChEMBL 9.01
Active Molecules (156)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XZWJCUBBBUYBFD
|
9.1 | IC50 | 2 | — | |
HXWRRTCVHCEFEO
|
9.1 | IC50 | 2 | — | |
YTMOJRFDMQVJGK
|
9.1 | IC50 | 2 | — | |
YMGSFPHRPRBAFF
|
9.1 | IC50 | 2 | — | |
OLZRHVFWMXZNMK
|
9.1 | IC50 | 2 | — | |
YRMNNNMNSFWNIR
|
9.0 | IC50 | 2 | — | |
IEGDVJDHRFSJAC
|
9.0 | IC50 | 2 | — | |
OOUWDISFEFEHIW
|
8.9 | IC50 | 2 | — | |
LNILZCFUNKQKGB
|
8.9 | IC50 | 2 | — | |
PDVMTOIBVXVEMS
|
8.8 | IC50 | 2 | — | |
VSMRVDFLWXBTCO
|
8.8 | IC50 | 2 | — | |
FCNHGNSESJZBMO
|
8.7 | IC50 | 2 | — | |
KWIHOEXEWRNRMW
|
8.5 | IC50 | 2 | — | |
PFWOJTLVNOZSGQ
|
8.5 | IC50 | 2 | — | |
HWOSZLZJQKYXHL
|
8.5 | IC50 | 2 | — | |
XSSVGYVSNAGLBL
|
8.4 | IC50 | 2 | — | |
MNHNQVHNKNMYAI
|
8.4 | IC50 | 2 | — | |
KINMYBBFQRSVLL
|
8.3 | IC50 | 6 | — | |
WBCRUAYGKPHAFU
|
8.3 | IC50 | 2 | — | |
QOGZMGDNFLQOLD
|
8.2 | IC50 | 2 | — | |
LJTSSXVJDHQUSV
|
8.2 | IC50 | 2 | — | |
NSQPUHWCJPLGPR
|
8.2 | IC50 | 2 | — | |
JMGJFYAGKIZLOT
|
7.8 | IC50 | 2 | — | |
AAVNWPCABSDFAJ
|
7.8 | IC50 | 2 | — | |
OKHJMRQSVKWXRA
|
7.8 | IC50 | 2 | — | |
MJVNYZRDRDGSII
|
7.7 | IC50 | 2 | — | |
PTSSFSTYSLYKSC
|
7.6 | IC50 | 2 | — | |
JJAWGNIQEOFURP
|
7.3 | IC50 | 2 | — | |
NUCQMWUHUMQXKP
|
7.2 | IC50 | 2 | — | |
MZIJPPLPZPKXEU
|
7.1 | IC50 | 2 | — | |
QYICUUHLNRBIMS
|
7.0 | IC50 | 2 | — | |
AWQSFBWLDFPCKC
|
6.9 | IC50 | 3 | — | |
BJRMDIIIWVVQSZ
|
6.8 | IC50 | 2 | — | |
MMCFFZBMJHBWGM
|
6.8 | IC50 | 2 | — | |
YSNROTHUHBZNDE
|
6.8 | IC50 | 2 | — | |
GVOVTRIALVWKIK
|
6.7 | IC50 | 2 | — | |
HVZWHAHDNKMEHJ
|
6.7 | IC50 | 2 | — | |
OTSKYWVPYJRLJF
|
6.7 | IC50 | 2 | — | |
DUVMSDROOBQDDF
|
6.6 | IC50 | 2 | — | |
GAKQXDXJHZRVJC
|
6.6 | IC50 | 2 | — | |
USFGZWPSRSTMGP
|
6.5 | IC50 | 2 | — | |
KSZRMQOUHDNLBY
|
6.5 | IC50 | 2 | — | |
NUGSUIAMNWUMFA
|
6.5 | IC50 | 2 | — | |
DRZGUYAHIWXYDK
|
6.5 | IC50 | 2 | — | |
GIZJXCZQTLNBNJ
|
6.5 | IC50 | 2 | — | |
XSVYDPIWGWYQKU
|
6.5 | IC50 | 2 | — | |
KMDJBICPSGCNQO
|
6.4 | IC50 | 2 | — | |
SIVCFZOBMAVEST
|
6.4 | IC50 | 2 | — | |
WBEQJJJAOUDSDB
|
6.3 | IC50 | 2 | — | |
INIUOCWMNJACSH
|
6.3 | IC50 | 2 | — |