Target Details
| UniProt AC | P21980 |
|---|---|
| Gene Symbol | TGM2 |
| Protein Name | Protein-glutamine gamma-glutamyltransferase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00927 (Transglut_C) PF01841 (Transglut_core) PF00868 (Transglut_N) |
Summary
- Multi-target molecules 109
- Clinical molecules 0
- Avg pChEMBL 6.91
KEGG Pathways (1)
Active Molecules (109)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
USDHUZPYPQHFDF
|
7.0 | IC50 | 2 | — | |
YJPRKLMOVDRCAS
|
7.0 | IC50 | 2 | — | |
KVXYMLDQLRULQZ
|
6.9 | IC50 | 2 | — | |
AYRUOQVKLKAZSR
|
6.9 | IC50 | 2 | — | |
GKYUMQAHUKCTFF
|
6.9 | IC50 | 2 | — | |
ACWATKJJUKSZQP
|
6.9 | IC50 | 2 | — | |
VNQPCKMVGJKTJH
|
6.9 | IC50 | 2 | — | |
HSJFIKQFCGIASR
|
6.8 | IC50 | 2 | — | |
MYULBZNAQWBTNR
|
6.8 | IC50 | 2 | — | |
FTAUSXYITUEDBR
|
6.8 | IC50 | 2 | — | |
QETQXZZDUYKSLT
|
6.8 | IC50 | 2 | — | |
LXGRQANYXIETIX
|
6.8 | IC50 | 2 | — | |
QLXWMPCZCUDTNR
|
6.8 | IC50 | 2 | — | |
YNCLTMDYTQONDJ
|
6.8 | IC50 | 2 | — | |
LWAMOXQCZPZLPQ
|
6.8 | IC50 | 2 | — | |
VLNFXQAOBBSNKE
|
6.8 | IC50 | 2 | — | |
NPPFXOSTKHCNFF
|
6.8 | IC50 | 4 | — | |
ADEYZLJKYDETQM
|
6.8 | IC50 | 2 | — | |
KDSOLMQUXOVVMH
|
6.7 | IC50 | 2 | — | |
VIBBHXNFIOPNNL
|
6.7 | IC50 | 2 | — | |
XMNBZHULQOIYJP
|
6.7 | IC50 | 2 | — | |
ANNVTFXGUOTPFJ
|
6.7 | IC50 | 2 | — | |
CDNYKJWMFPLSCF
|
6.7 | IC50 | 2 | — | |
HUSXJSWBEDZQOM
|
6.7 | IC50 | 2 | — | |
YRNGWIRXJKRYIH
|
6.7 | IC50 | 2 | — | |
COYVFVIKFYVYSP
|
6.7 | IC50 | 2 | — | |
MWZBNEMHQOAPBA
|
6.7 | IC50 | 2 | — | |
OFESJBNCGCTWMR
|
6.7 | IC50 | 2 | — | |
ZZMBUQMIXHHHHO
|
6.7 | IC50 | 2 | — | |
KFYIBLRUWLRNDO
|
6.6 | IC50 | 2 | — | |
WIBAZTHQTQWZHI
|
6.6 | IC50 | 2 | — | |
NHCXGUDVOIMHSD
|
6.6 | IC50 | 2 | — | |
FYDGIPZGOAHZLU
|
6.6 | IC50 | 2 | — | |
WZTJFZPMDNYCQU
|
6.5 | IC50 | 2 | — | |
BJMDBTYPZXELHV
|
6.5 | IC50 | 2 | — | |
GTJWEIZJYGZHRC
|
6.5 | IC50 | 2 | — | |
WOFVKXAEDONAOH
|
6.5 | IC50 | 2 | — | |
RDOUMSQWXZDIAX
|
6.5 | IC50 | 2 | — | |
TWFOJSGRBGECRZ
|
6.5 | IC50 | 2 | — | |
IHBGOWJVCCERSM
|
6.5 | IC50 | 2 | — | |
HHRHIFUFVSETDV
|
6.5 | IC50 | 2 | — | |
HBSBXYQAOQSDOH
|
6.4 | IC50 | 2 | — | |
WYEOUUFRUVATIG
|
6.4 | IC50 | 2 | — | |
UTOANJDVDDTCAE
|
6.3 | IC50 | 2 | — | |
LRPVZBYNRPUWGT
|
6.3 | IC50 | 2 | — | |
BCXLWTAPIXVTHU
|
6.3 | IC50 | 2 | — | |
DJMTYLNAGSTKIS
|
6.3 | IC50 | 2 | — | |
WYMLIRAIPXONOR
|
6.3 | IC50 | 2 | — | |
DJMTYLNAGSTKIS
|
6.3 | IC50 | 2 | — | |
PAVNCPWGPWLGKA
|
6.2 | IC50 | 2 | — |