Target Details
| UniProt AC | P21980 |
|---|---|
| Gene Symbol | TGM2 |
| Protein Name | Protein-glutamine gamma-glutamyltransferase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00927 (Transglut_C) PF01841 (Transglut_core) PF00868 (Transglut_N) |
Summary
- Multi-target molecules 109
- Clinical molecules 0
- Avg pChEMBL 6.91
KEGG Pathways (1)
Active Molecules (109)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FQJALHVQVRBZAV
|
8.0 | IC50 | 2 | — | |
NWFPBQYIKXKLNF
|
8.0 | IC50 | 3 | — | |
PPWTZJSWZPBNAR
|
7.9 | IC50 | 2 | — | |
XCTOMICEQKFIHG
|
7.8 | IC50 | 2 | — | |
NHUHIZWFCRMBPE
|
7.8 | IC50 | 2 | — | |
NVPKGMMRESDDIZ
|
7.8 | IC50 | 2 | — | |
UHLAXZLHHGCTPG
|
7.7 | IC50 | 2 | — | |
OYEOXFZRVNDRKZ
|
7.6 | IC50 | 5 | — | |
WAZOFYYWAQHTQZ
|
7.5 | IC50 | 2 | — | |
VKBTYOLWPAQPQN
|
7.5 | IC50 | 2 | — | |
VKBTYOLWPAQPQN
|
7.5 | IC50 | 2 | — | |
KFEJNIOLFTZKGK
|
7.5 | IC50 | 2 | — | |
LRALVUHFEBURCW
|
7.5 | IC50 | 2 | — | |
ADEYZLJKYDETQM
|
7.4 | IC50 | 2 | — | |
ILXQHEXDPPFFMG
|
7.4 | IC50 | 2 | — | |
HGHMBXSRMHYTTI
|
7.4 | IC50 | 2 | — | |
PXHUPSZLKUMVDF
|
7.4 | IC50 | 2 | — | |
CDKQBMPFADMQPE
|
7.3 | IC50 | 2 | — | |
VYZAWJGFABJTFI
|
7.3 | IC50 | 2 | — | |
MBWCZMOHXUQUNT
|
7.3 | IC50 | 2 | — | |
YJAMSUUVGADKPC
|
7.3 | IC50 | 2 | — | |
XHSXBLKEPKFAKN
|
7.3 | IC50 | 2 | — | |
YLFFVZRZVCYQKV
|
7.3 | IC50 | 2 | — | |
FHKFISJKLJDQGA
|
7.3 | IC50 | 2 | — | |
IJUIDQWNEGTWHT
|
7.3 | IC50 | 2 | — | |
IJUIDQWNEGTWHT
|
7.3 | IC50 | 2 | — | |
VRDFMCKVXUFVQZ
|
7.3 | IC50 | 2 | — | |
YDQPDMPSNNWJLX
|
7.3 | IC50 | 2 | — | |
GVOGSWMECLVCGB
|
7.2 | IC50 | 2 | — | |
IXGYYBUDUYQAKL
|
7.2 | IC50 | 2 | — | |
QXPGBZSOGVCSDE
|
7.2 | IC50 | 2 | — | |
NQBKYYQCMVCECJ
|
7.2 | IC50 | 2 | — | |
YQGFARSMJDYNKQ
|
7.2 | IC50 | 2 | — | |
IAPBEGPEZRDIQR
|
7.2 | IC50 | 2 | — | |
FDPHLPHLATXLCE
|
7.2 | IC50 | 2 | — | |
IDVFAXVNLAAPBC
|
7.2 | IC50 | 2 | — | |
VCYXFCBTBKTENL
|
7.2 | IC50 | 2 | — | |
LSDONZLKFHWCQG
|
7.1 | IC50 | 2 | — | |
GFUHZWGGEHHBLH
|
7.1 | IC50 | 2 | — | |
PIFOKPGDWWGCKA
|
7.1 | IC50 | 2 | — | |
WMJKIMAXEPLJFO
|
7.1 | IC50 | 2 | — | |
DGMDMBJEUDSTCY
|
7.1 | IC50 | 2 | — | |
DILRPFMIKQIFPZ
|
7.0 | IC50 | 2 | — | |
PAVNCPWGPWLGKA
|
7.0 | IC50 | 2 | — | |
HSROVNPCCIYQKL
|
7.0 | IC50 | 2 | — | |
MWZBNEMHQOAPBA
|
7.0 | IC50 | 2 | — | |
VTNSZKSWGBRJSL
|
7.0 | IC50 | 2 | — | |
AUAPVOQGBUKHMB
|
7.0 | IC50 | 3 | — | |
NSUSTSLQHFZJBZ
|
7.0 | IC50 | 2 | — | |
PSZSXLJBEDTGAZ
|
7.0 | IC50 | 2 | — |