Target Details
| UniProt AC | P21918 |
|---|---|
| Gene Symbol | DRD5 |
| Protein Name | D(1B) dopamine receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 220
- Clinical molecules 8
- Avg pChEMBL 7.26
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (220)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LLBLNMUONVVVPG
|
6.2 | Ki | 17 | — | |
OIDVIVFTQMTONJ
|
6.2 | Ki | 4 | — | |
OVKBSFKFSBQCLW
|
6.2 | Ki | 5 | — | |
VUCKSZWMRCSPME
|
6.2 | Ki | 7 | — | |
CVRMQFHSOSVJET
|
6.1 | Ki | 6 | — | |
RAPZEAPATHNIPO
|
6.1 | Ki | 28 | Yes | |
GVNRTSAPTNNIPL
|
6.1 | Ki | 6 | — | |
OPXIAQIQFMLKDK
|
6.1 | Ki | 6 | — | |
CILDROBPHGWMGB
|
6.0 | Ki | 6 | — | |
HXCJZIBJTFITNI
|
6.0 | Ki | 3 | — | |
PLZGEHCHVFNRGK
|
6.0 | Ki | 5 | — | |
MNZXCYDDVWTITD
|
6.0 | Ki | 3 | — | |
WKWADEWWLCVVLF
|
6.0 | Ki | 14 | — | |
DUKNIHFTDAXJON
|
6.0 | Ki | 13 | — | |
GXGVWEMSSIKHOZ
|
6.0 | Ki | 8 | — | |
HMXDWDSNPRNUKI
|
6.0 | Ki | 72 | — | |
HUXFXXWYIRBVJR
|
6.0 | Ki | 9 | — | |
JJKPSOUEWPDPFS
|
6.0 | IC50 | 9 | Yes | |
UDYXSPVICNNUPJ
|
6.0 | Ki | 9 | — | |
UQKLFSKKULYASF
|
6.0 | Ki | 5 | — |