Target Details
| UniProt AC | P21860 |
|---|---|
| Gene Symbol | ERBB3 |
| Protein Name | Receptor tyrosine-protein kinase erbB-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF14843 (GF_recep_IV) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) |
Summary
- Multi-target molecules 109
- Clinical molecules 23
- Avg pChEMBL 7.39
KEGG Pathways (7)
Associated Diseases (2)
Active Molecules (109)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FYSLYZBOZFMTDD
|
6.3 | IC50 | 6 | Yes | |
IZUCNCXKMINXNV
|
6.2 | IC50 | 4 | — | |
VCBUVKNXUBPBBX
|
6.2 | IC50 | 2 | — | |
OKYKKFLCZPGQHI
|
6.2 | IC50 | 5 | — | |
CJAOTOWETHYRND
|
6.1 | IC50 | 5 | — | |
XGALLCVXEZPNRQ
|
6.1 | Kd | 39 | Yes | |
FAQVIRHBDLOKHC
|
6.1 | IC50 | 2 | — | |
SKBWQUPLWQUWPH
|
6.1 | IC50 | 6 | Yes | |
SGQJPPQXKVUHGS
|
6.1 | IC50 | 6 | Yes |