Target Details
| UniProt AC | P21860 |
|---|---|
| Gene Symbol | ERBB3 |
| Protein Name | Receptor tyrosine-protein kinase erbB-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF14843 (GF_recep_IV) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) |
Summary
- Multi-target molecules 109
- Clinical molecules 23
- Avg pChEMBL 7.39
KEGG Pathways (7)
Associated Diseases (2)
Active Molecules (109)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SKBWQUPLWQUWPH
|
7.4 | IC50 | 6 | Yes | |
MCEJMTKEBSFUJK
|
7.4 | IC50 | 4 | — | |
YROLHQZDEFQCCR
|
7.4 | IC50 | 4 | — | |
QZMGOBDHHJBODW
|
7.4 | IC50 | 4 | — | |
HUFOZJXAKZVRNJ
|
7.3 | IC50 | 10 | — | |
ZYVUNNQGVXTJSW
|
7.3 | IC50 | 4 | — | |
QFMCOTDYFYKZNH
|
7.3 | IC50 | 4 | — | |
RKUBYGFDHATQAZ
|
7.3 | IC50 | 4 | — | |
PAFOOYBINUNMGT
|
7.3 | IC50 | 6 | Yes | |
GPHGJEXSAYLLDB
|
7.2 | IC50 | 2 | — | |
XWHJPZMQYNMSOJ
|
7.2 | IC50 | 4 | — | |
RRXVMGHOCPACNG
|
7.2 | IC50 | 6 | Yes | |
IEZFFFOOLULQBR
|
7.2 | IC50 | 4 | — | |
FAFWJMNGAWQHOH
|
7.2 | IC50 | 5 | — | |
WFWGCFGIGNLAGO
|
7.2 | IC50 | 4 | — | |
YSULEGHESGUMPH
|
7.2 | IC50 | 2 | — | |
QMOJTBYMFQXLLU
|
7.1 | IC50 | 6 | Yes | |
TXVGFVZTROUDRA
|
7.0 | IC50 | 2 | — | |
HKJUUPKKOAGVDB
|
7.0 | IC50 | 6 | Yes | |
LDLBFITVAGVRNV
|
7.0 | IC50 | 6 | Yes | |
SGQJPPQXKVUHGS
|
7.0 | IC50 | 6 | Yes | |
ALLOGFWHFYNGAI
|
7.0 | IC50 | 4 | — | |
ZXNLHZGFHDHRCO
|
7.0 | IC50 | 4 | — | |
YSROCLXNQLJIKL
|
7.0 | IC50 | 5 | — | |
MFAQYJIYDMLAIM
|
6.9 | Kd | 130 | Yes | |
VAARYSWULJUGST
|
6.8 | Kd | 119 | Yes | |
JEQABWAFHZXXLZ
|
6.8 | IC50 | 4 | — | |
LJQVSABKPVFCTG
|
6.8 | IC50 | 4 | — | |
LVNYQEFSHJDOCT
|
6.8 | IC50 | 4 | — | |
HYCYVMNKZFALHN
|
6.8 | IC50 | 5 | — | |
UHTHHESEBZOYNR
|
6.8 | Kd | 66 | Yes | |
KZHGNEQISTYYRV
|
6.8 | IC50 | 2 | — | |
ACTXRPZBCPTJSQ
|
6.7 | IC50 | 2 | — | |
XXJWYDDUDKYVKI
|
6.7 | Kd | 52 | — | |
UDVRGRBOAMOTGS
|
6.7 | IC50 | 4 | — | |
HCONVOOBXMEDII
|
6.7 | IC50 | 4 | — | |
OMZCMEYTWSXEPZ
|
6.7 | Kd | 43 | Yes | |
PEGQWGLLBPWDAS
|
6.7 | IC50 | 4 | — | |
LFSVOMOBKPCKHF
|
6.6 | IC50 | 2 | — | |
WTCWMZHEAXFWPJ
|
6.6 | IC50 | 4 | — | |
AUFNWHLGERWYHJ
|
6.6 | IC50 | 2 | — | |
MDTJFOFYNXHTKV
|
6.6 | IC50 | 5 | — | |
AQAMLFJHLGJOCZ
|
6.6 | IC50 | 5 | — | |
JCKPXXCMARLTQI
|
6.6 | IC50 | 6 | Yes | |
NKUFCHJXONJOLU
|
6.5 | IC50 | 4 | — | |
PAFOOYBINUNMGT
|
6.5 | IC50 | 6 | Yes | |
UVWRRZRGHPHHLL
|
6.4 | Kd | 4 | — | |
DLQXAWIVHRHOQT
|
6.4 | IC50 | 6 | Yes | |
XPUIECRALWERTL
|
6.4 | IC50 | 4 | — | |
DJCDHWXQLRMRTB
|
6.3 | IC50 | 5 | — |