Target Details
| UniProt AC | P21860 |
|---|---|
| Gene Symbol | ERBB3 |
| Protein Name | Receptor tyrosine-protein kinase erbB-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF14843 (GF_recep_IV) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) |
Summary
- Multi-target molecules 109
- Clinical molecules 23
- Avg pChEMBL 7.39
KEGG Pathways (7)
Associated Diseases (2)
Active Molecules (109)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GYFAPMADUQCILZ
|
9.2 | IC50 | 5 | — | |
UBPYILGKFZZVDX
|
9.1 | Kd | 130 | Yes | |
FOOPCYOJMREECW
|
9.1 | IC50 | 5 | — | |
TUYDDIWQXWTNSW
|
9.0 | IC50 | 2 | — | |
YVXVVBRYZHAWFN
|
8.9 | IC50 | 2 | — | |
ZAWWCTXYZTURLN
|
8.9 | IC50 | 4 | — | |
IMLBZWHQWRDARS
|
8.8 | IC50 | 4 | — | |
VSZMJABKDRJXRI
|
8.8 | IC50 | 2 | — | |
IRMHXRHXLFRZFM
|
8.7 | IC50 | 2 | — | |
LJKPCPFZGRKCSR
|
8.7 | IC50 | 2 | — | |
OONFNUWBHFSNBT
|
8.7 | IC50 | 11 | — | |
DUYJMQONPNNFPI
|
8.7 | IC50 | 11 | — | |
AZSRSNUQCUDCGG
|
8.5 | IC50 | 4 | — | |
DFJSJLGUIXFDJP
|
8.4 | IC50 | 9 | — | |
JYIUNVOCEFIUIU
|
8.4 | IC50 | 2 | — | |
JZSLVCXMHPNGNA
|
8.3 | IC50 | 5 | — | |
BFSRTTWIPACGMI
|
8.3 | IC50 | 4 | — | |
GNIFAULXFNJRKN
|
8.3 | IC50 | 4 | — | |
HNFWPMOZPVUYBB
|
8.2 | IC50 | 4 | — | |
NSIQZZLWJHBVJS
|
8.2 | IC50 | 2 | — | |
VEQYCEHJTJSHLO
|
8.1 | IC50 | 4 | — | |
JWNPDZNEKVCWMY
|
8.1 | Kd | 57 | Yes | |
QWAHCSOEUYGXDS
|
8.1 | IC50 | 4 | — | |
HLSFKKBVOPHVAO
|
8.1 | IC50 | 2 | — | |
FXRLTQRMUHOCQN
|
8.0 | IC50 | 4 | — | |
YYNUBPUXFJKWOK
|
8.0 | IC50 | 4 | — | |
AAKJLRGGTJKAMG
|
8.0 | IC50 | 50 | Yes | |
VHGQJLWYOGRRAE
|
8.0 | IC50 | 4 | — | |
CMMUJJHJYMYOJR
|
7.8 | IC50 | 4 | — | |
LOFBARGGJCBDJT
|
7.8 | IC50 | 4 | — | |
SJMHQTPAHZSCGB
|
7.8 | IC50 | 4 | — | |
QIAHWAXXEKSCCE
|
7.7 | IC50 | 2 | — | |
ZBNZXTGUTAYRHI
|
7.7 | Kd | 102 | Yes | |
HHAXMCRVXIYOJR
|
7.7 | IC50 | 4 | — | |
VVIRSVARIBXZHS
|
7.7 | IC50 | 4 | — | |
DIQMCPYEEIZMCH
|
7.7 | IC50 | 2 | — | |
ODMXWZROLKITMS
|
7.7 | IC50 | 3 | — | |
ABLXXKUDDSMAHU
|
7.7 | IC50 | 4 | — | |
ZYQXEVJIFYIBHZ
|
7.6 | IC50 | 5 | — | |
AYIGALYNJFDMRN
|
7.6 | IC50 | 4 | — | |
FDPQKRUPPHXZMQ
|
7.6 | IC50 | 2 | — | |
RWQIOAPAHWFTMQ
|
7.6 | IC50 | 4 | — | |
JFEKMLAOHVYFGS
|
7.5 | IC50 | 4 | — | |
XGCIQQCBKZDMPK
|
7.5 | IC50 | 2 | — | |
DLQXAWIVHRHOQT
|
7.5 | IC50 | 6 | Yes | |
MHJBSGVISQZKDI
|
7.5 | IC50 | 4 | — | |
FLFHZVYTVPANLR
|
7.5 | IC50 | 4 | — | |
BWWLZGAQCJRAGF
|
7.5 | IC50 | 4 | — | |
OXAZPVDJCIJPFP
|
7.5 | IC50 | 4 | — | |
BVNDWJSTWPXVCD
|
7.4 | IC50 | 2 | — |