Target Details
| UniProt AC | P21817 |
|---|---|
| Gene Symbol | RYR1 |
| Protein Name | Ryanodine receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08709 (Ins145_P3_rec) PF00520 (Ion_trans) PF02815 (MIR) PF08454 (RIH_assoc) PF06459 (RR_TM4-6) PF01365 (RYDR_ITPR) PF21119 (RYDR_Jsol) PF02026 (RyR) PF00622 (SPRY) |
Summary
- Multi-target molecules 35
- Clinical molecules 0
- Avg pChEMBL 8.97
KEGG Pathways (8)
Associated Diseases (4)
Active Molecules (35)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MXSRCGHETGMNGI
|
9.4 | IC50 | 3 | — | |
AXONTVKFBHBALT
|
9.3 | IC50 | 3 | — | |
HWENSJQGPPXSPG
|
9.3 | IC50 | 3 | — | |
JXSXWPCGHMFVGR
|
9.2 | IC50 | 3 | — | |
QWHJEDGXVYDZGR
|
9.2 | IC50 | 3 | — | |
XGVWHMVZYCTASP
|
9.2 | IC50 | 3 | — | |
MACWQTHSUCWPOE
|
9.2 | IC50 | 3 | — | |
RJHWXUSDSADOOD
|
9.2 | IC50 | 3 | — | |
NNEGEHDJOHHIGP
|
9.1 | IC50 | 3 | — | |
HVOCYKRGXDBAPR
|
9.1 | IC50 | 3 | — | |
LKEPUSYXXXTDQI
|
9.1 | IC50 | 2 | — | |
MTAFDCDGNPHAKS
|
9.1 | IC50 | 3 | — | |
POWFJUCHFPYCRU
|
9.1 | IC50 | 2 | — | |
XJSPSRRPVKOQCW
|
9.1 | IC50 | 3 | — | |
GZBVSECJBWKOFI
|
9.0 | IC50 | 2 | — | |
XMJMYXPPWSLYBN
|
9.0 | IC50 | 3 | — | |
AIZHXUUSVDWSRD
|
9.0 | IC50 | 3 | — | |
BGXAKEYZRXIHGZ
|
9.0 | IC50 | 2 | — | |
ZASQNOFKMXADOA
|
9.0 | IC50 | 3 | — | |
BWGRHTJKFKCSGW
|
8.9 | IC50 | 3 | — | |
BWNZRZRECKJDGL
|
8.9 | IC50 | 3 | — | |
FNPBMTZGHSTSCD
|
8.8 | IC50 | 3 | — | |
JOMGWMSWUXJNHR
|
8.8 | IC50 | 3 | — | |
RJCVQFMGMSMVAX
|
8.8 | IC50 | 3 | — | |
SENHYTFMMJPFHA
|
8.8 | IC50 | 3 | — | |
ZEFSHHCIZUSSQS
|
8.8 | IC50 | 2 | — | |
ZZMROTDWVPXWJA
|
8.8 | IC50 | 2 | — | |
ZMXMTLXHUISIRF
|
8.8 | IC50 | 3 | — | |
BZKRFBALBPSKAK
|
8.8 | IC50 | 2 | — | |
CJROUFPGIGKBGZ
|
8.8 | IC50 | 3 | — | |
PAOJZRPLNNXONF
|
8.8 | IC50 | 3 | — | |
PILSAMURLMDHHO
|
8.8 | IC50 | 2 | — | |
NBCDCMYRULBOTN
|
8.7 | IC50 | 3 | — | |
PCZMIWZARLASMT
|
8.7 | IC50 | 2 | — | |
UQROQVVPXLGCTI
|
8.7 | IC50 | 2 | — |