Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
INWHLZUNIJSPHA
|
8.5 | IC50 | 5 | — | |
IZIDHKRDFQGCMR
|
8.5 | IC50 | 2 | — | |
JMGHVRJQMLUCCL
|
8.5 | IC50 | 3 | — | |
KBATXXSVGCJBDV
|
8.5 | IC50 | 2 | — | |
MEKRRNGBDAULRT
|
8.5 | IC50 | 3 | — | |
MLUFVERLBQGOEV
|
8.5 | IC50 | 5 | — | |
ODVWBADYBXDOHC
|
8.5 | IC50 | 3 | — | |
OVZKBAUSZIANJA
|
8.5 | IC50 | 5 | — | |
UHBZJNMSQJZNCB
|
8.5 | IC50 | 5 | — | |
VUKUZGSFRAYWPM
|
8.5 | IC50 | 2 | — | |
WGEUPMAJTYQVEP
|
8.5 | IC50 | 3 | — | |
ARMOWUIZJHLBIQ
|
8.5 | IC50 | 5 | — | |
CFSRQGNLLQKRJE
|
8.5 | IC50 | 5 | — | |
FWUSQYKXFMDVPH
|
8.5 | IC50 | 5 | — | |
IOJGQJINDPXDDW
|
8.5 | IC50 | 5 | — | |
NWFHDWLGIMCVRK
|
8.5 | Kd | 3 | — | |
WHXUXVVTKNDEIG
|
8.5 | IC50 | 2 | — | |
YURYMGHZHGYXAW
|
8.5 | IC50 | 5 | — | |
AYLDOIMOFYNYQP
|
8.5 | IC50 | 5 | — | |
AYLGNVUDASUDAB
|
8.5 | IC50 | 5 | — | |
FJKSLOFTCKXLSC
|
8.5 | IC50 | 2 | — | |
IEMVLSQUPRKUEE
|
8.5 | IC50 | 6 | — | |
JDDJMJIAWGNUGT
|
8.5 | IC50 | 5 | — | |
JYQPFNMDHXKRKL
|
8.5 | IC50 | 5 | — | |
LCIPUHSYYUXUFV
|
8.5 | IC50 | 5 | — | |
LUQCVGYRUMKEMD
|
8.5 | IC50 | 5 | — | |
MLUFVERLBQGOEV
|
8.5 | IC50 | 5 | — | |
NIKYJDORPJPERE
|
8.5 | IC50 | 5 | — | |
PFTPAJNMFJOUIG
|
8.5 | IC50 | 5 | — | |
SXYFYNVZTYNDKV
|
8.5 | IC50 | 5 | — | |
TVWOUPGUUIDZET
|
8.5 | IC50 | 6 | — | |
UWJYHBHRJHNCHQ
|
8.5 | IC50 | 5 | — | |
WPAMXPNNWJGKNP
|
8.5 | IC50 | 5 | — | |
YHYVUGXKQJNEDM
|
8.5 | IC50 | 3 | — | |
ZATQHWAWTFBUEN
|
8.5 | IC50 | 4 | — | |
ZAWBYXATEBIOBQ
|
8.5 | IC50 | 5 | — | |
ZDPMRTCLIVGQSN
|
8.5 | IC50 | 5 | — | |
ZVFYULVCRUAESA
|
8.5 | IC50 | 2 | — | |
BAPFBTJYCKDGNL
|
8.5 | IC50 | 5 | — | |
DIVGFMHEBBBJGH
|
8.5 | IC50 | 2 | — | |
HGOIJUTXACYYTH
|
8.5 | IC50 | 5 | — | |
JZADASHLALTDDI
|
8.5 | IC50 | 2 | — | |
MWLGIUCUYKLSHV
|
8.5 | IC50 | 5 | — | |
RFPQZVZQZKKHQS
|
8.5 | IC50 | 5 | — | |
SAHTUCUOJHIHGN
|
8.5 | IC50 | 5 | — | |
UJGBKUMKLLDSQI
|
8.5 | IC50 | 5 | — | |
WOMBJJKPVIDFFI
|
8.5 | IC50 | 5 | — | |
XBRAGXSHNWCDEC
|
8.5 | IC50 | 5 | — | |
XMLPCBKZIXENAI
|
8.5 | IC50 | 4 | — | |
FFFJXBUHHHYLPP
|
8.4 | IC50 | 5 | — |