Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HNMFYNZSWBGHHO
|
8.5 | IC50 | 3 | — | |
IATQVFKHNZFWTF
|
8.5 | IC50 | 3 | — | |
IGXJTXDPMDXZJZ
|
8.5 | IC50 | 3 | — | |
IIGRWRUGUUITMA
|
8.5 | IC50 | 5 | — | |
JWBKKCJZIDXHLG
|
8.5 | IC50 | 3 | — | |
JWOIPGHVEJHTRG
|
8.5 | IC50 | 3 | — | |
KSQSKRYGIKNQHZ
|
8.5 | IC50 | 2 | — | |
LFIHPORZEBZZHY
|
8.5 | IC50 | 3 | — | |
MDOANUHLWYXBTL
|
8.5 | IC50 | 3 | — | |
MNGPWOAYMBPUSQ
|
8.5 | IC50 | 5 | — | |
MNUGHQYUMFMXIC
|
8.5 | IC50 | 5 | — | |
NVWPJAMSFZHMRS
|
8.5 | IC50 | 3 | — | |
OMHJAMXRVWTRAY
|
8.5 | IC50 | 3 | — | |
PFFKWQNVRNBIGB
|
8.5 | IC50 | 5 | — | |
QQXJQMPWTRDVIY
|
8.5 | IC50 | 3 | — | |
RNLTTXGJGQZWAF
|
8.5 | IC50 | 3 | — | |
SRFTVRWDQRUZRY
|
8.5 | IC50 | 3 | — | |
SRLZJSAQKFBYKX
|
8.5 | IC50 | 2 | — | |
SRNXPZGAZRUEQV
|
8.5 | IC50 | 3 | — | |
VJGVQTRRTNVNTM
|
8.5 | IC50 | 3 | — | |
VKGKMAJKOZBZQC
|
8.5 | IC50 | 3 | — | |
VSNIYTDVOFCOEC
|
8.5 | IC50 | 3 | — | |
XFGMNTTVFYLJIS
|
8.5 | IC50 | 2 | — | |
XOQVZSSDIQQUGO
|
8.5 | IC50 | 3 | — | |
XSDFUOBWKCWNGD
|
8.5 | IC50 | 3 | — | |
ZMEWJQRHELGMRY
|
8.5 | IC50 | 5 | — | |
GUHZQOUGERIFMY
|
8.5 | IC50 | 5 | — | |
IGZKSXILFWECCS
|
8.5 | IC50 | 3 | — | |
IXKVURLQMWDRPS
|
8.5 | IC50 | 5 | — | |
LFFMUTDOMVUDHX
|
8.5 | IC50 | 2 | — | |
MCCRDQXDXGETPQ
|
8.5 | IC50 | 5 | — | |
MDGGVKPYDJLWOU
|
8.5 | IC50 | 5 | — | |
OXFRISWNUYFISN
|
8.5 | IC50 | 5 | — | |
PYQPSJDRRIQAPP
|
8.5 | IC50 | 5 | — | |
RDIKEQDHARQJCT
|
8.5 | IC50 | 5 | — | |
RJOWKASSFBQDER
|
8.5 | IC50 | 4 | — | |
AUFUDTOCLCOVHF
|
8.5 | IC50 | 5 | — | |
GSJCRSBKLFGBOV
|
8.5 | IC50 | 5 | — | |
GXQZPCUWRYWOJV
|
8.5 | IC50 | 5 | — | |
LDZIHQWKUDOFTP
|
8.5 | IC50 | 5 | — | |
LOLPPWBBNUVNQZ
|
8.5 | IC50 | 97 | Yes | |
OLAHOMJCDNXHFI
|
8.5 | IC50 | 5 | — | |
OYHDEFFNZNIKPS
|
8.5 | IC50 | 5 | — | |
SYQCXJZLWMRWKD
|
8.5 | IC50 | 5 | — | |
XMVITVIKEQWXPB
|
8.5 | IC50 | 5 | — | |
XYUUXJDAJMUQMZ
|
8.5 | IC50 | 5 | — | |
YASHODHUWYIHDK
|
8.5 | IC50 | 5 | — | |
YWWFVNOOHJHQOP
|
8.5 | IC50 | 5 | — | |
CZKFBZFMVHZPQK
|
8.5 | IC50 | 5 | — | |
HTMVIKSMELCDMN
|
8.5 | IC50 | 2 | — |