Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MJBNLVZGJYYOOP
|
8.6 | IC50 | 5 | — | |
NKJIZRCNNJXSHH
|
8.6 | IC50 | 5 | — | |
PXRZIWUUBMUSOA
|
8.6 | IC50 | 5 | — | |
UXFVYTDPWIHCQK
|
8.6 | IC50 | 5 | — | |
BKZXMPAAWRKKRN
|
8.6 | IC50 | 5 | — | |
BTGLYCHFNHKNDV
|
8.6 | IC50 | 3 | — | |
GAYZGPGTYYBZNE
|
8.6 | IC50 | 4 | — | |
IHIQKRYMXUFAGS
|
8.6 | IC50 | 5 | — | |
JXGGHGLZZYBWNG
|
8.6 | IC50 | 5 | — | |
KRYZCYZIWKIKGN
|
8.6 | IC50 | 5 | — | |
LCWWFMHHNQAPDZ
|
8.6 | IC50 | 5 | — | |
LUQCVGYRUMKEMD
|
8.6 | IC50 | 5 | — | |
QECODAPTOHJSRN
|
8.6 | IC50 | 5 | — | |
VFFSRBOFGPSKTB
|
8.6 | IC50 | 5 | — | |
WZRAHVCKWICVFZ
|
8.6 | IC50 | 3 | — | |
YLMMYYCOZCUKKA
|
8.6 | IC50 | 5 | — | |
BQCQOBOXMZWHQL
|
8.5 | IC50 | 5 | — | |
FTBKZEPCWTYABP
|
8.5 | IC50 | 5 | — | |
GAMHYLRQXHJKEU
|
8.5 | IC50 | 3 | — | |
HQKHKYBURJLEMV
|
8.5 | IC50 | 5 | — | |
KFDQGFBOAAQCJQ
|
8.5 | IC50 | 3 | — | |
NVJBAXNECMDGLO
|
8.5 | IC50 | 5 | — | |
POKUGRIXYDIRKM
|
8.5 | IC50 | 3 | — | |
QVLVKBIGNUAHQR
|
8.5 | IC50 | 5 | — | |
QZTONRVOLAYTPJ
|
8.5 | IC50 | 5 | — | |
RLLJBVQJFQMSFQ
|
8.5 | IC50 | 3 | — | |
SLEJFRIKJJZQKL
|
8.5 | IC50 | 5 | — | |
UMBCDTSTLGNZAT
|
8.5 | IC50 | 3 | — | |
URZRQIDVBBEEHP
|
8.5 | IC50 | 2 | — | |
VZUAVFLTRIZLOD
|
8.5 | IC50 | 5 | — | |
WHUMKUVVBUUDAQ
|
8.5 | IC50 | 5 | — | |
YEGXHZZEFKJQGY
|
8.5 | IC50 | 5 | — | |
FBJRJSLJQISKRR
|
8.5 | IC50 | 5 | — | |
FRFIDSQIINSGEA
|
8.5 | IC50 | 5 | — | |
FWIRJQMGGXJLNW
|
8.5 | IC50 | 5 | — | |
GHNNOOKRRJQEEH
|
8.5 | IC50 | 5 | — | |
GLLVJFAKHOOPKT
|
8.5 | IC50 | 5 | — | |
IHCZEJLZOMIBDV
|
8.5 | IC50 | 5 | — | |
LLLHXFXUIWPWMH
|
8.5 | IC50 | 5 | — | |
MOJFGNLMKZRCMV
|
8.5 | IC50 | 5 | — | |
PILVYDBBHFTMOU
|
8.5 | IC50 | 5 | — | |
QLWRWFVHNSZTSI
|
8.5 | IC50 | 5 | — | |
WRSYRDYMLSQTFT
|
8.5 | IC50 | 5 | — | |
AQMXONPVPCMPJM
|
8.5 | IC50 | 3 | — | |
BFQGJTMYIGHGLT
|
8.5 | IC50 | 5 | — | |
CQDRTFWUDOIACC
|
8.5 | IC50 | 5 | — | |
FHSRSKPIXRNREU
|
8.5 | IC50 | 3 | — | |
GIGLTKPRJFVONN
|
8.5 | IC50 | 3 | — | |
GIWGPTOTMRZIBE
|
8.5 | IC50 | 5 | — | |
HGZFXVSSFDAUID
|
8.5 | IC50 | 3 | — |