Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WWBXYIDLWINHSB
|
8.6 | IC50 | 2 | — | |
AHSYHYFTUKZLCI
|
8.6 | IC50 | 5 | — | |
FXTIMSGNOBJVAE
|
8.6 | IC50 | 4 | — | |
HWWONGHTSRGZJQ
|
8.6 | IC50 | 2 | — | |
KFKYFVCBOAGDTP
|
8.6 | IC50 | 3 | — | |
SBXJWOVGQTVLAE
|
8.6 | IC50 | 3 | — | |
TUNDEPCHRSSRHC
|
8.6 | IC50 | 4 | — | |
VEGCSHHXEINKOV
|
8.6 | IC50 | 4 | — | |
VGCISMLLKUTUAO
|
8.6 | IC50 | 5 | — | |
ZRJOWLUBZFAUCV
|
8.6 | IC50 | 5 | — | |
IIGOWKTZNCRSCJ
|
8.6 | IC50 | 5 | — | |
MJBNLVZGJYYOOP
|
8.6 | IC50 | 5 | — | |
QECODAPTOHJSRN
|
8.6 | IC50 | 5 | — | |
RTFQRZUYRSOSBU
|
8.6 | IC50 | 5 | — | |
RYRVRXVRRSZALT
|
8.6 | IC50 | 5 | — | |
WAHZMINPROSVEH
|
8.6 | IC50 | 5 | — | |
AZOXWOCICFEBCQ
|
8.6 | IC50 | 11 | — | |
DOUKVHHXGYUDNB
|
8.6 | IC50 | 2 | — | |
HTLBPVHYAPCHEP
|
8.6 | IC50 | 2 | — | |
IGQPIMXAOKZGSL
|
8.6 | IC50 | 5 | — | |
MBQTZWPSYBLXMC
|
8.6 | IC50 | 5 | — | |
MMGNRRUXETXMDE
|
8.6 | IC50 | 5 | — | |
NYEZHXSUIICMSA
|
8.6 | IC50 | 5 | — | |
OLAHOMJCDNXHFI
|
8.6 | IC50 | 6 | — | |
SKIAWPBWOAQQEZ
|
8.6 | IC50 | 5 | — | |
VRQMAABPASPXMW
|
8.6 | IC50 | 8 | — | |
WRSYRDYMLSQTFT
|
8.6 | IC50 | 5 | — | |
YIKYPGSFLXUTQT
|
8.6 | IC50 | 5 | — | |
AYJLMQKFNIMDMS
|
8.6 | IC50 | 5 | — | |
CVTLXZHZCMNAPK
|
8.6 | Kd | 3 | — | |
GKJCVYLDJWTWQU
|
8.6 | IC50 | 6 | — | |
JCQODDIJVHORMY
|
8.6 | IC50 | 5 | — | |
KRHJVQBHCYJAPS
|
8.6 | IC50 | 2 | — | |
NKVDPZYKPGKBTK
|
8.6 | IC50 | 5 | — | |
PAGYYFBXLGVGOO
|
8.6 | IC50 | 3 | — | |
QBOPLHQHJDUIPC
|
8.6 | IC50 | 4 | — | |
WZWCHRIODAFYKY
|
8.6 | IC50 | 5 | — | |
KYDPEBSICGOHJT
|
8.6 | IC50 | 5 | — | |
NIHYIKXINLALJA
|
8.6 | IC50 | 5 | — | |
GHEIOFQIMGYHML
|
8.6 | IC50 | 5 | — | |
HCFBZSOLPIWAPX
|
8.6 | IC50 | 5 | — | |
JNTRATZGRSGDTJ
|
8.6 | IC50 | 2 | — | |
OBQHIGGTXIFTRF
|
8.6 | IC50 | 4 | — | |
RAMCMRRBGWIDLK
|
8.6 | IC50 | 8 | Yes | |
UCWGZZUXJLIYIK
|
8.6 | IC50 | 4 | — | |
YHGCMZIYHWHQKR
|
8.6 | IC50 | 5 | — | |
YMKCMNJQFGEWCA
|
8.6 | IC50 | 8 | Yes | |
ZFMBRQRHSFCSAB
|
8.6 | IC50 | 2 | — | |
DDNOUEXAVDQPMR
|
8.6 | IC50 | 5 | — | |
DDUJNWDXTYPSCS
|
8.6 | IC50 | 5 | — |