Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CXZJXVJPISUKMR
|
6.5 | IC50 | 6 | — | |
FVAUWSNXHKYZKA
|
6.5 | IC50 | 4 | — | |
HEJWDMSZDBYDME
|
6.5 | IC50 | 3 | — | |
HYWSNPJICYRJJW
|
6.5 | IC50 | 2 | — | |
IAXXRGACLVIRBH
|
6.5 | IC50 | 3 | — | |
IDRGFNPZDVBSSE
|
6.5 | IC50 | 3 | — | |
JUEXCQYUGREKRI
|
6.5 | IC50 | 2 | — | |
LOHGOSYFXUKKCF
|
6.5 | IC50 | 3 | — | |
LTMRAJBNXMUMGW
|
6.5 | IC50 | 2 | — | |
MFBGSEULLCUEGY
|
6.5 | IC50 | 2 | — | |
MQHRWBGHHGJHTA
|
6.5 | IC50 | 2 | — | |
MXDCACLUETVZNL
|
6.5 | IC50 | 8 | — | |
NFBJDTDBPBKXCM
|
6.5 | IC50 | 2 | — | |
NUUDCMWMURFYJL
|
6.5 | IC50 | 2 | — | |
OKNNCKJQXLUIJK
|
6.5 | IC50 | 3 | — | |
OZCYACNGDDKBEX
|
6.5 | IC50 | 3 | — | |
PGRJFPIBHFUXKF
|
6.5 | IC50 | 3 | — | |
RCZXWPDZUWTFFT
|
6.5 | IC50 | 2 | — | |
SCHRCCHASZMVAB
|
6.5 | IC50 | 7 | — | |
SDVGDLIRSAANJQ
|
6.5 | IC50 | 2 | — | |
SNJGLLPXSZFEJC
|
6.5 | IC50 | 2 | — | |
WOAXRKYXUKTLEM
|
6.5 | IC50 | 7 | — | |
XTEQFWKBNUKCEQ
|
6.5 | IC50 | 2 | — | |
GQXHZLUUXHPIAG
|
6.5 | IC50 | 3 | — | |
RUNFHROXJGUGHE
|
6.5 | IC50 | 3 | — | |
IQJPWAAWPFBLPZ
|
6.5 | IC50 | 2 | — | |
SHMHUSCNIYPOFW
|
6.5 | IC50 | 3 | — | |
ZHMXXVNQAFCXKK
|
6.5 | IC50 | 15 | — | |
GDELGHCKNKINFD
|
6.5 | Kd | 3 | — | |
SNOZVZWRCAEAQT
|
6.5 | IC50 | 4 | — | |
YHWHYCTUDCULTF
|
6.5 | IC50 | 4 | — | |
GOOHQQKXWCOUPK
|
6.5 | IC50 | 3 | — | |
IRPMVZSWQAOIAN
|
6.5 | Kd | 4 | — | |
QYEHCYDRHZCGMU
|
6.5 | IC50 | 3 | — | |
VDVZOCBAFGDAKS
|
6.5 | IC50 | 5 | — | |
HHEGTWYVXJJAQX
|
6.5 | IC50 | 3 | — | |
NMNCNSNYQUWXHG
|
6.5 | IC50 | 3 | — | |
NZUXTCRYWPXTJA
|
6.5 | IC50 | 6 | Yes | |
VJOXMKASEXHOQP
|
6.5 | IC50 | 5 | — | |
LLGFEJJPLZCCQL
|
6.4 | IC50 | 10 | Yes | |
OSVUGUHRKMMBSE
|
6.4 | Kd | 170 | — | |
SMHHULBWHKVYLT
|
6.4 | IC50 | 3 | — | |
UNDMKZSXJIATGJ
|
6.4 | IC50 | 3 | — | |
UXBPLRFFIZKKDS
|
6.4 | IC50 | 3 | — | |
IPUQQXBHNNBVBU
|
6.4 | IC50 | 2 | — | |
YBAINXIJZYKTME
|
6.4 | IC50 | 4 | — | |
YOQKLHUPUONSAT
|
6.4 | IC50 | 4 | — | |
UGWVKPNXNPMUKR
|
6.4 | IC50 | 3 | — | |
AALXHEPRLHLNCZ
|
6.4 | IC50 | 3 | — | |
DGDQLZKKOIZBKE
|
6.4 | IC50 | 4 | — |