Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LCWWFMHHNQAPDZ
|
8.8 | IC50 | 5 | — | |
LCWWFMHHNQAPDZ
|
8.8 | IC50 | 5 | — | |
LWJVODKOEBQHPO
|
8.8 | IC50 | 5 | — | |
PDCHXVOBVIQUEZ
|
8.8 | IC50 | 5 | — | |
VLOPFGZLJSYVCD
|
8.8 | IC50 | 4 | — | |
WEASQIMFKRBYLI
|
8.8 | IC50 | 5 | — | |
AKINNIMWOKBQKR
|
8.7 | IC50 | 2 | — | |
BINZKUIUUZZJSK
|
8.7 | IC50 | 3 | — | |
FXIBXFGZSDZFSP
|
8.7 | IC50 | 5 | — | |
INWHLZUNIJSPHA
|
8.7 | IC50 | 5 | — | |
MSLILZFULYZLIC
|
8.7 | IC50 | 3 | — | |
OARJPSVHVHBFTL
|
8.7 | IC50 | 2 | — | |
QMXGFRWKHLJTJA
|
8.7 | IC50 | 2 | — | |
SISPBNWXCLKBKE
|
8.7 | IC50 | 5 | — | |
WNLHGAXRRIMFGV
|
8.7 | IC50 | 5 | — | |
ZAPUSNWRFJVSGX
|
8.7 | IC50 | 5 | — | |
DIYIEVQNIORQDL
|
8.7 | IC50 | 5 | — | |
LPAVQJHVSDAOKU
|
8.7 | IC50 | 5 | — | |
MCCRDQXDXGETPQ
|
8.7 | IC50 | 5 | — | |
ABQSJCCISLWTEW
|
8.7 | IC50 | 8 | Yes | |
AISWQGLURAAAKE
|
8.7 | IC50 | 7 | — | |
BYEGVFRRTLAAQA
|
8.7 | IC50 | 2 | — | |
BYJMQCNNDWXBRA
|
8.7 | IC50 | 5 | — | |
GITNDHUJOBXSCE
|
8.7 | IC50 | 4 | — | |
GMNMMGZZBZYAMO
|
8.7 | IC50 | 2 | — | |
GWCJUEKQORIUTJ
|
8.7 | IC50 | 5 | — | |
MLGJITMGHIKNFO
|
8.7 | IC50 | 3 | — | |
PRXXXHCKGRNFLJ
|
8.7 | IC50 | 8 | — | |
QECODAPTOHJSRN
|
8.7 | IC50 | 5 | — | |
QULAUQOGDDJGPW
|
8.7 | IC50 | 5 | — | |
XGKDTJAGVPINNR
|
8.7 | IC50 | 4 | — | |
CMQBIUKGSMOTTQ
|
8.7 | IC50 | 5 | — | |
DIDLAUMNKKUFSF
|
8.7 | IC50 | 5 | — | |
HQCPXLHKIKERQR
|
8.7 | IC50 | 2 | — | |
HQKHKYBURJLEMV
|
8.7 | IC50 | 5 | — | |
JMBVTEKOAZJGIC
|
8.7 | IC50 | 5 | — | |
WXAXVITWIABKBN
|
8.7 | IC50 | 5 | — | |
BAWZESLJEVSFRN
|
8.7 | IC50 | 6 | — | |
BBZNFKRCGVBNLL
|
8.7 | IC50 | 3 | — | |
BIZAIIWAPNOYPN
|
8.7 | IC50 | 5 | — | |
CYOSEXIUDLKBBP
|
8.7 | IC50 | 3 | — | |
DXIOQMYZLOTSFT
|
8.7 | IC50 | 2 | — | |
GEATXDJAPAHPTP
|
8.7 | IC50 | 10 | — | |
KEKXLNDHFOMLPS
|
8.7 | IC50 | 3 | — | |
MEEJXBYUJRNZGM
|
8.7 | IC50 | 3 | — | |
NEDQSDMNOSMYHF
|
8.7 | IC50 | 5 | — | |
NZYVQKUNDWKOTA
|
8.7 | IC50 | 4 | — | |
OLFIHCSTOANEMN
|
8.7 | IC50 | 5 | — | |
PGLZJHICUYCCJE
|
8.7 | IC50 | 7 | — | |
PHXJVRSECIGDHY
|
8.7 | IC50 | 59 | — |