Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IMIWAPPULTUBIS
|
6.9 | IC50 | 2 | — | |
JEWLNTYVEOVLDJ
|
6.9 | IC50 | 4 | — | |
JOAFMERUDZPPNN
|
6.9 | IC50 | 4 | — | |
JQZPHXVRUKBOIV
|
6.9 | IC50 | 3 | — | |
JROYVVPLLZICTQ
|
6.9 | IC50 | 4 | — | |
KNGYNRPKVJRSCS
|
6.9 | IC50 | 2 | — | |
KOCMBIKLUSRLCW
|
6.9 | IC50 | 4 | — | |
KOJOWJGCRTVIMZ
|
6.9 | IC50 | 3 | — | |
LRKVCZLAEJBOCR
|
6.9 | IC50 | 3 | — | |
LYBWHFGDCBIJOZ
|
6.9 | IC50 | 4 | — | |
MATNJDUYNSNQAP
|
6.9 | IC50 | 3 | — | |
MDUMQYWNCWDCFN
|
6.9 | IC50 | 2 | — | |
MVKPTHHFJXWIKQ
|
6.9 | IC50 | 4 | — | |
NVNVJMMINIYGSC
|
6.9 | IC50 | 3 | — | |
NZPNDEFTDKMRTD
|
6.9 | IC50 | 3 | — | |
OAACLZHMPVPUCR
|
6.9 | IC50 | 2 | — | |
PTYCAJJZCVUFAH
|
6.9 | IC50 | 2 | — | |
QXXAYAZKUCZZCU
|
6.9 | IC50 | 2 | — | |
UEPSEWZKBBSEIR
|
6.9 | IC50 | 3 | — | |
UGZJEEACQBQYAZ
|
6.9 | IC50 | 2 | — | |
ULMGILFSLBVEHM
|
6.9 | IC50 | 4 | — | |
UOIFLDNBEYDHRI
|
6.9 | IC50 | 4 | — | |
UZPQUBHBXBSNBP
|
6.9 | IC50 | 2 | — | |
VCLIPTAHOIBJCI
|
6.9 | IC50 | 2 | — | |
WNQUARCCIKLBAE
|
6.9 | IC50 | 4 | — | |
XFURXPJZSULRHJ
|
6.9 | IC50 | 2 | — | |
XUYMTPYPUQKVNL
|
6.9 | IC50 | 3 | — | |
YGXZSSISOXOCBF
|
6.9 | IC50 | 2 | — | |
ZDLKGMWZIWWDAC
|
6.9 | IC50 | 3 | — | |
ZQAOKGPEOCTXLO
|
6.9 | IC50 | 3 | — | |
ZVGCJEWDDCZXNH
|
6.9 | IC50 | 3 | — | |
ZVUOPVKBPNUNBU
|
6.9 | IC50 | 3 | — | |
CHYRHTDWXRVJMJ
|
6.9 | IC50 | 5 | — | |
FRKAOJSMULEWJT
|
6.9 | IC50 | 4 | — | |
FVOAPVPGTADZMK
|
6.9 | Kd | 5 | — | |
ZGKIVVODTURAMT
|
6.9 | IC50 | 3 | — | |
FQDRWRLLOXGGSS
|
6.9 | IC50 | 4 | — | |
GSTHTWGRLIWKTQ
|
6.9 | IC50 | 4 | — | |
HOGUOXLIWYGQAR
|
6.9 | Kd | 3 | — | |
KNPOOYXLOYFJMB
|
6.9 | IC50 | 4 | — | |
LPHGQGHRAUKWMN
|
6.9 | IC50 | 2 | — | |
BBNFZHSVWAORMK
|
6.9 | IC50 | 3 | — | |
HUTNEDYZVCYOIK
|
6.9 | IC50 | 4 | — | |
NQFKHCPZYMIACL
|
6.9 | IC50 | 2 | — | |
OPKYWWXALAAUOX
|
6.9 | IC50 | 5 | — | |
QTLMLSKDPMFIPH
|
6.9 | IC50 | 4 | — | |
XARWOHKDCBRPBQ
|
6.9 | IC50 | 6 | — | |
AJDPVRCTXQVCTL
|
6.9 | IC50 | 3 | — | |
BXEDCNVFSZUBPI
|
6.9 | IC50 | 6 | Yes | |
CWWGWUITOJWIQB
|
6.9 | IC50 | 5 | — |