Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RXSORSCKDDIFPE
|
7.1 | IC50 | 4 | — | |
HYUAHSHYXCUQFA
|
7.1 | IC50 | 5 | — | |
QKNXNIJTPNITNW
|
7.1 | IC50 | 4 | — | |
ULIJLYCJYRQKBG
|
7.1 | IC50 | 7 | Yes | |
CUDVHEFYRIWYQD
|
7.1 | IC50 | 11 | — | |
HLPZBUCKWKGYBH
|
7.1 | IC50 | 4 | — | |
ANBUERYCJLDFHA
|
7.1 | IC50 | 3 | — | |
GJSGCDJNBXKAGX
|
7.1 | IC50 | 3 | — | |
UIVVZQXKDIOKDR
|
7.1 | IC50 | 3 | — | |
SACIBDXGXFJPQN
|
7.0 | IC50 | 5 | — | |
SDIZOFZVSQJIHJ
|
7.0 | IC50 | 4 | — | |
JQDCEZKFIOQSIK
|
7.0 | IC50 | 2 | — | |
KXEMINRANVTICS
|
7.0 | IC50 | 9 | — | |
NWFHDWLGIMCVRK
|
7.0 | Kd | 3 | — | |
MCUVUHFGOBRXMR
|
7.0 | IC50 | 5 | — | |
JYRCWIALULHJNT
|
7.0 | IC50 | 3 | — | |
IJQYMGBALOJSDL
|
7.0 | IC50 | 4 | — | |
RWCAQQLPZYSTLH
|
7.0 | IC50 | 3 | — | |
YBYROMOZHMOYRQ
|
7.0 | IC50 | 5 | — | |
CNUXPGAXDUDMDQ
|
7.0 | IC50 | 4 | — | |
HKSZLNNOFSGOKW
|
7.0 | Kd | 213 | — | |
SAZIXFAROZCPDO
|
7.0 | IC50 | 7 | Yes | |
TXGHNTNBBSGNGF
|
7.0 | Kd | 3 | — | |
BMTRLYMQWMETEI
|
7.0 | IC50 | 5 | — | |
GIBYRJLRSLPQGP
|
7.0 | IC50 | 6 | — | |
HYIAWTNBECBRDG
|
7.0 | IC50 | 5 | — | |
LTGQGTOGUOJONG
|
7.0 | IC50 | 3 | — | |
ZRDNUCXRIXLMNC
|
7.0 | IC50 | 5 | — | |
VNQNDAAGNJESBU
|
7.0 | IC50 | 3 | — | |
NGMHHQOCOVUJGA
|
7.0 | IC50 | 3 | — | |
AZRYWRIZWVORFG
|
7.0 | IC50 | 2 | — | |
JILYVQBGAUYZHM
|
7.0 | IC50 | 2 | — | |
MHVVNNKZAOUIQX
|
7.0 | IC50 | 3 | — | |
QKMYJNCUYMFPMF
|
7.0 | IC50 | 3 | — | |
RITAVMQDGBJQJZ
|
7.0 | Kd | 43 | — | |
VKZBLNHYOGTBFX
|
7.0 | Kd | 3 | — | |
WCWUXEGQKLTGDX
|
7.0 | Kd | 22 | Yes | |
WMYLESPXATZBNH
|
7.0 | IC50 | 4 | — | |
ATLWKYGJPAIBQP
|
6.9 | IC50 | 2 | — | |
BNWOJWBIDQYRGE
|
6.9 | IC50 | 3 | — | |
CHNIXQFJUWPQIE
|
6.9 | IC50 | 3 | — | |
DKHFDFCYFZTWRU
|
6.9 | IC50 | 2 | — | |
DKRMLOOSLSMXGR
|
6.9 | IC50 | 3 | — | |
DQQVACSMEANERY
|
6.9 | IC50 | 4 | — | |
DZFWCZZWYHIBQD
|
6.9 | IC50 | 3 | — | |
FIRSCNNHKKRUPO
|
6.9 | IC50 | 2 | — | |
FJAZRHLEJFERMY
|
6.9 | IC50 | 3 | — | |
FSGGEVVZGGOLIG
|
6.9 | IC50 | 2 | — | |
FVVOTLOJZNGNRW
|
6.9 | IC50 | 2 | — | |
GVSFWLZASUTWRB
|
6.9 | IC50 | 4 | — |