Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YPOMZOAOKGGCTH
|
7.2 | Kd | 4 | — | |
YTLHHVOVPRVGEK
|
7.2 | Kd | 4 | — | |
ZADKHKCWESQLMD
|
7.2 | Kd | 4 | — | |
ZNFNEVKOJDAJRK
|
7.2 | Kd | 4 | — | |
ZOAODOQFJZVCLZ
|
7.2 | Kd | 4 | — | |
ZTPZFCISZOWQEC
|
7.2 | Kd | 4 | — | |
ZXCRAGLNYNWMPV
|
7.2 | Kd | 4 | — | |
ZYJXKCVDCJYPHV
|
7.2 | IC50 | 4 | — | |
AMKNQROTNAOJQE
|
7.2 | IC50 | 7 | — | |
DWSQRXVYJVMLAJ
|
7.2 | IC50 | 5 | — | |
JARSMEDYFYAQRJ
|
7.2 | IC50 | 3 | — | |
VFUNZAFJEZQGGZ
|
7.2 | IC50 | 4 | — | |
WOAAWLOTSPDCPE
|
7.2 | IC50 | 5 | — | |
DHADFGSEMYCYHN
|
7.2 | IC50 | 4 | — | |
NPIPSFYAGMCQMP
|
7.2 | Kd | 5 | — | |
VNOICNWZXXPXMD
|
7.2 | IC50 | 3 | — | |
FAJMNJHLDPNTLS
|
7.2 | IC50 | 3 | — | |
FIPKJBQQLVYHGW
|
7.2 | IC50 | 5 | — | |
FNTYYRMQLQQXEI
|
7.2 | IC50 | 4 | — | |
JBXLEBAVNPBBTP
|
7.2 | Kd | 3 | — | |
MRXALCNCKIEVIU
|
7.2 | IC50 | 3 | — | |
NCKYHNJFFJIAOQ
|
7.2 | IC50 | 3 | — | |
QRNIDLJCQJRXOX
|
7.2 | IC50 | 2 | — | |
GGOULWQHNSLDAO
|
7.2 | IC50 | 2 | — | |
NEZWQSDNUYDARK
|
7.2 | IC50 | 2 | — | |
OIXSXBWXHOOWSI
|
7.2 | Kd | 3 | — | |
YSIMHBIGEXRRJS
|
7.2 | IC50 | 3 | — | |
PODHQRDKTIXYRI
|
7.2 | IC50 | 4 | — | |
QNABDSWBQJKBHK
|
7.2 | IC50 | 45 | — | |
LDRPTUAJCNQUAA
|
7.2 | IC50 | 4 | — | |
MCJMDQAWLHQTAP
|
7.2 | IC50 | 5 | — | |
ANRDBTWHHHRDGH
|
7.1 | IC50 | 3 | — | |
CPLYQZKEYHJUJZ
|
7.1 | IC50 | 4 | — | |
FZTNGFWPULVQOX
|
7.1 | IC50 | 3 | — | |
KFVPABDXNXQFRD
|
7.1 | IC50 | 3 | — | |
NHHQJBCNYHBUSI
|
7.1 | Kd | 220 | — | |
WBETVCGZCGUZGH
|
7.1 | IC50 | 3 | — | |
JDCRLLMMJUHCOS
|
7.1 | IC50 | 4 | — | |
DELHAEOXMJXGFI
|
7.1 | IC50 | 3 | — | |
MHZIGJBWNNGGBZ
|
7.1 | IC50 | 3 | — | |
NESPYTXPLQBOGE
|
7.1 | IC50 | 3 | — | |
VVEWWOOATHIBFT
|
7.1 | IC50 | 2 | — | |
ZNTZUQOJVAETBB
|
7.1 | IC50 | 2 | — | |
DOUQJCMUZWYEEN
|
7.1 | IC50 | 3 | — | |
NTPRYKFNRGGZJM
|
7.1 | IC50 | 4 | — | |
QOQWOVMERAEQMV
|
7.1 | IC50 | 5 | — | |
VBCUYTZWMKPDOM
|
7.1 | IC50 | 5 | — | |
VQCDZFWRGXFUMS
|
7.1 | IC50 | 5 | — | |
YGSJOHAJXSRCHZ
|
7.1 | IC50 | 5 | — | |
JKXJLIXEEITPGY
|
7.1 | IC50 | 3 | — |