Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MKVMEJKNLUWFSQ
|
7.3 | IC50 | 7 | Yes | |
OALGSXHIRDEVKH
|
7.3 | IC50 | 3 | — | |
TXIHQMLNWLFVHM
|
7.3 | IC50 | 6 | Yes | |
GPGFFJPUFNKAFY
|
7.3 | IC50 | 2 | — | |
IHZFSYQVOKXLQL
|
7.3 | IC50 | 4 | — | |
CHCRNUSFDLTSCW
|
7.3 | IC50 | 3 | — | |
IBIHVAILDLNSJB
|
7.3 | IC50 | 3 | — | |
YXUKTQQYFNLKGS
|
7.3 | IC50 | 4 | — | |
ZZXYMFBCKNUTKB
|
7.3 | IC50 | 5 | — | |
AKQRMZOMYBNHFA
|
7.3 | IC50 | 3 | — | |
PAZDFSJAERQBCY
|
7.3 | IC50 | 7 | Yes | |
UARDLGBJPODKSU
|
7.3 | Kd | 3 | — | |
VYTBQANMHOWXBJ
|
7.3 | IC50 | 4 | — | |
MMHADELJVDMSNQ
|
7.3 | IC50 | 7 | Yes | |
BEGHDVFYWWPCOW
|
7.3 | IC50 | 5 | — | |
BRHSQONMORDAKC
|
7.3 | IC50 | 4 | — | |
BVBQWWHKISLHNA
|
7.3 | IC50 | 3 | — | |
DKZWIVQXLWEMHT
|
7.3 | IC50 | 3 | — | |
DPGQEPDCBUAILJ
|
7.3 | IC50 | 4 | — | |
FSSSZUYRWRKQTG
|
7.3 | IC50 | 3 | — | |
GEVYWRKXSBJQDH
|
7.3 | IC50 | 4 | — | |
HASQYLAYAPUXFY
|
7.3 | IC50 | 3 | — | |
HUXAYMWWNBTISC
|
7.3 | IC50 | 4 | — | |
KFOBBZNALUDUBF
|
7.3 | IC50 | 3 | — | |
KMYOBCBTZOLZSF
|
7.3 | IC50 | 4 | — | |
SVWVQLLEQHHYGA
|
7.3 | IC50 | 4 | — | |
UYRPXCKSWOLKSQ
|
7.3 | IC50 | 4 | — | |
WUBFAXNVDMCVIO
|
7.3 | IC50 | 12 | Yes | |
ZEPQGUOIUNEIAO
|
7.3 | IC50 | 4 | — | |
BQHKHXMCVZGNBQ
|
7.2 | IC50 | 3 | — | |
IGDRSPHKZGFFEO
|
7.2 | IC50 | 5 | — | |
LUJNIROONWQIJG
|
7.2 | IC50 | 6 | — | |
ZSWKLCBAZCPCCQ
|
7.2 | IC50 | 3 | — | |
AHFBSEIEBDJLKY
|
7.2 | IC50 | 4 | — | |
CCJCJTIJCYCVGD
|
7.2 | IC50 | 3 | — | |
HJZADWAESABHBK
|
7.2 | IC50 | 3 | — | |
IQJPWAAWPFBLPZ
|
7.2 | IC50 | 2 | — | |
UTNNTOYFWYQAJK
|
7.2 | IC50 | 3 | — | |
HHAMLGNIKIGSCW
|
7.2 | IC50 | 5 | — | |
MUFKFZHTITXUCK
|
7.2 | IC50 | 5 | — | |
AJYPVIIYKOYXJT
|
7.2 | Kd | 4 | — | |
ATOKRZYNWKJUKU
|
7.2 | Kd | 4 | — | |
AUEAFLHHJOYOPQ
|
7.2 | Kd | 4 | — | |
AVKQAQABIOQCSE
|
7.2 | Kd | 4 | — | |
AWBYPEWMPJFEMQ
|
7.2 | Kd | 4 | — | |
BHTRYYDGKAPOGI
|
7.2 | Kd | 4 | — | |
BNHJJRHVPDWPJM
|
7.2 | Kd | 4 | — | |
BOVDQPIZOYYEFP
|
7.2 | Kd | 4 | — | |
BSQJCKAAVPVMPI
|
7.2 | Kd | 4 | — | |
CAPUTJVVKZMNLX
|
7.2 | Kd | 4 | — |