Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ROHJEIACUNTGFP
|
7.4 | IC50 | 16 | — | |
SLJDNVLLZVPBBP
|
7.4 | IC50 | 3 | — | |
ZDHGZDSUPWLHQJ
|
7.4 | IC50 | 3 | — | |
BOOGXXSASXAIRQ
|
7.4 | IC50 | 3 | — | |
JGEBLDKNWBUGRZ
|
7.4 | IC50 | 20 | Yes | |
POBFQGSWQFFYGS
|
7.4 | IC50 | 3 | — | |
UBHNHZFEBHPHCU
|
7.4 | IC50 | 3 | — | |
XKYKMEFXVHYFRM
|
7.4 | IC50 | 5 | — | |
YXARVHZXTQVAOP
|
7.4 | IC50 | 11 | — | |
AJYHQOVGZKVPCX
|
7.4 | IC50 | 3 | — | |
BPUWFUZFMBQQHH
|
7.4 | IC50 | 3 | — | |
CLVSAAPONJRSGJ
|
7.4 | IC50 | 7 | — | |
FFRZNGZQCMXHFG
|
7.4 | IC50 | 5 | — | |
IOFKHMOBIMMQEZ
|
7.4 | IC50 | 3 | — | |
WWCNDWUCWUTCSJ
|
7.4 | IC50 | 3 | — | |
XMEUXGVNDCEFRR
|
7.4 | IC50 | 3 | — | |
YHVHYWYQEFELOW
|
7.4 | IC50 | 44 | — | |
AYQXERSJLFQLST
|
7.4 | IC50 | 4 | — | |
RMDBTAYWYWJRIC
|
7.4 | IC50 | 3 | — | |
XLQWGSJRCYXEBO
|
7.4 | IC50 | 3 | — | |
AKWPNUYFJIBLPT
|
7.4 | IC50 | 3 | — | |
APHFSWUAUANWQN
|
7.4 | IC50 | 3 | — | |
CKXQGKOTLUERBE
|
7.4 | IC50 | 5 | — | |
DWOSRPACOIQSTD
|
7.4 | IC50 | 3 | — | |
GNUPRONFIQLGBG
|
7.4 | IC50 | 3 | — | |
ODJYOEFFPIQYEF
|
7.4 | IC50 | 3 | — | |
RMSUYVFJOYLGSV
|
7.4 | IC50 | 3 | — | |
VGRUOSBHWZUWNW
|
7.4 | IC50 | 3 | — | |
ZHKJWOIKWGAMMG
|
7.4 | IC50 | 3 | — | |
PDRZSJXTKWJVHW
|
7.4 | IC50 | 5 | — | |
YYCRQWMDRNTZLT
|
7.4 | IC50 | 4 | — | |
HQQABXMYFDMKIT
|
7.4 | IC50 | 5 | — | |
IFPPYSWJNWHOLQ
|
7.4 | IC50 | 52 | Yes | |
KNCMFVBGBJGBGI
|
7.4 | IC50 | 7 | Yes | |
LAQISKDGTLGFIK
|
7.4 | IC50 | 5 | — | |
OGQXSEPTYDNHKF
|
7.4 | IC50 | 3 | — | |
SRWBBPJNBPSOFD
|
7.4 | IC50 | 5 | — | |
LJEJQSGDKVPZTB
|
7.3 | Kd | 4 | — | |
WCHAWRNEALMUFZ
|
7.3 | IC50 | 5 | — | |
WRXMILDAPMMJQN
|
7.3 | IC50 | 3 | — | |
HOSLGTLYFRADJZ
|
7.3 | IC50 | 2 | — | |
KPPYNHRMNFKBRA
|
7.3 | IC50 | 7 | — | |
QRRIRGBKZLRRLS
|
7.3 | IC50 | 3 | — | |
WEZLWZYLJAMPNY
|
7.3 | IC50 | 2 | — | |
AMHUBFWCCMLLCJ
|
7.3 | IC50 | 15 | — | |
CRMQCPICYHHFIL
|
7.3 | IC50 | 5 | — | |
FFRZNGZQCMXHFG
|
7.3 | IC50 | 4 | — | |
HRMKTZOBLPIBBW
|
7.3 | IC50 | 4 | — | |
WTIZTZHDEUCFJA
|
7.3 | IC50 | 5 | — | |
BFLRXUQCNYUNBN
|
7.3 | IC50 | 5 | — |