Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AOYJOQPVLIISJS
|
8.9 | IC50 | 4 | — | |
LKMLECIRYJPQOC
|
8.9 | IC50 | 5 | — | |
USBWBRLHRGYCPG
|
8.9 | IC50 | 4 | — | |
YJPRCVWTWRDRGM
|
8.9 | IC50 | 5 | — | |
AWNATJMQNZMYAX
|
8.8 | IC50 | 5 | — | |
JVIIZPUVKMLGDE
|
8.8 | IC50 | 3 | — | |
QIXCNXNXARCJIU
|
8.8 | IC50 | 3 | — | |
RFPTZQDUVNZXTN
|
8.8 | IC50 | 3 | — | |
UBGBIWLWSXCNJS
|
8.8 | IC50 | 3 | — | |
UQZPQFKVJWOQTM
|
8.8 | IC50 | 4 | — | |
WITKAEIQNFPTFS
|
8.8 | IC50 | 5 | — | |
YLUAUDRMSFJFJJ
|
8.8 | IC50 | 4 | — | |
AHAHQLJJHZPGFT
|
8.8 | IC50 | 5 | — | |
QPILVXXWABVBBV
|
8.8 | IC50 | 5 | — | |
SQEZUHWWJYSRDG
|
8.8 | IC50 | 5 | — | |
XTLRUHNSWCKNBK
|
8.8 | IC50 | 5 | — | |
PHTNPGCZALDYLD
|
8.8 | IC50 | 4 | — | |
DBAMREJIAGZICQ
|
8.8 | IC50 | 3 | — | |
HFMVSRPUPXYHGG
|
8.8 | IC50 | 2 | — | |
HKMTYQNMRIBAHX
|
8.8 | IC50 | 4 | — | |
NHSCTFBEZPHZRZ
|
8.8 | IC50 | 5 | — | |
PHOLJWMEQMFEMO
|
8.8 | IC50 | 5 | — | |
SFYNOFFYMQHBAL
|
8.8 | IC50 | 4 | — | |
SUXYGJZMCWKJJI
|
8.8 | IC50 | 26 | Yes | |
XSCIHVCSBPPQDG
|
8.8 | IC50 | 3 | — | |
XVQAACIPBICWNT
|
8.8 | IC50 | 2 | — | |
DPRCWKSNIPIOOK
|
8.8 | IC50 | 5 | — | |
KTQNUSVVKAQAIV
|
8.8 | IC50 | 5 | — | |
QZUYKKDZNXWNPD
|
8.8 | IC50 | 5 | — | |
CYWDLLRCEFUKME
|
8.8 | IC50 | 3 | — | |
LABBTNAJUXRSJY
|
8.8 | IC50 | 3 | — | |
MKEGPZIMUWZUKO
|
8.8 | IC50 | 4 | — | |
NMFMLTFZEUDACF
|
8.8 | IC50 | 4 | — | |
OWFCRBSDJKZKBD
|
8.8 | IC50 | 5 | — | |
PMWJNWXMNAKMHW
|
8.8 | IC50 | 5 | — | |
ROOGKKMRYAUSLO
|
8.8 | IC50 | 3 | — | |
MXMLJQCILGAGCP
|
8.8 | IC50 | 5 | — | |
UHBAVEAIOQERCE
|
8.8 | IC50 | 4 | — | |
AVHLETMOCLYGNK
|
8.8 | IC50 | 5 | — | |
SBKRUFBQSKWUSE
|
8.8 | IC50 | 5 | — | |
SXANNSUWWUIUKO
|
8.8 | IC50 | 2 | — | |
BNZAPGUSNOSNGF
|
8.8 | IC50 | 2 | — | |
FCCSDYKLOXTQPP
|
8.8 | IC50 | 4 | — | |
KONCHEYJKNSRJF
|
8.8 | IC50 | 5 | — | |
UWGPKLQEDALKIM
|
8.8 | IC50 | 2 | — | |
GWBUXINOYBCSHF
|
8.8 | IC50 | 2 | — | |
IVQXFJNVCKJIHX
|
8.8 | IC50 | 5 | — | |
NHVRJDXWYOYVDB
|
8.8 | IC50 | 3 | — | |
OLAHOMJCDNXHFI
|
8.8 | IC50 | 5 | — | |
AHSYHYFTUKZLCI
|
8.8 | IC50 | 5 | — |