Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XLHXAKNUXURIJF
|
7.6 | IC50 | 4 | — | |
XVHQBHLEUMQQIV
|
7.6 | IC50 | 5 | — | |
FYSWRJTZQOHOOU
|
7.6 | Kd | 4 | — | |
GFYSRXDFPQGTBC
|
7.6 | IC50 | 3 | — | |
AQIPZTFTBQQQFZ
|
7.6 | IC50 | 2 | — | |
DGOJHYZMDAOBKI
|
7.6 | IC50 | 6 | — | |
IANQNWVOZRBDPD
|
7.6 | IC50 | 6 | — | |
IJGJTVDBFPOSRT
|
7.6 | IC50 | 3 | — | |
NVVJIKMAQUOOHJ
|
7.6 | IC50 | 5 | — | |
QXIOZIFTPMAING
|
7.6 | IC50 | 17 | — | |
RCYHCFDDBFAHNT
|
7.6 | IC50 | 3 | — | |
RUROKZDZIPBDNX
|
7.6 | IC50 | 5 | — | |
SCXUCUKEHHIEDN
|
7.6 | IC50 | 5 | — | |
BFLRXUQCNYUNBN
|
7.6 | IC50 | 5 | — | |
WWAYYWJGGVLUAS
|
7.6 | IC50 | 5 | — | |
AQWDWTGCVNYFBN
|
7.6 | IC50 | 4 | — | |
DKIQJCCUKVKITR
|
7.6 | IC50 | 3 | — | |
FMYCPNBASOLHNV
|
7.6 | IC50 | 2 | — | |
FWUPGRCAIARXDF
|
7.6 | IC50 | 3 | — | |
KESJSLSZDNGMAM
|
7.6 | IC50 | 3 | — | |
KTZAXOPOMIBTDN
|
7.6 | IC50 | 2 | — | |
NYNQETWJMMSWJX
|
7.6 | IC50 | 3 | — | |
VQXBFPOCHKNAOT
|
7.6 | IC50 | 5 | — | |
HAKZRRLEELHDIL
|
7.6 | IC50 | 4 | — | |
JIBBGYSUSKAPDY
|
7.6 | IC50 | 19 | — | |
ROPXRZFMHWDEMR
|
7.6 | IC50 | 3 | — | |
SFHBVSAUUQEUEZ
|
7.6 | IC50 | 5 | — | |
YMWNLONTKXQMAJ
|
7.6 | IC50 | 3 | — | |
GXQRKBRJAOUSGL
|
7.6 | IC50 | 3 | — | |
HICVGIIDYAHAGN
|
7.6 | IC50 | 2 | — | |
PQMJXZUWJZKZJJ
|
7.6 | IC50 | 3 | — | |
PRQXFOSXTOETEQ
|
7.6 | IC50 | 3 | — | |
QOTKZBTTZSPMNH
|
7.6 | IC50 | 5 | Yes | |
VVMFTDMSORZANW
|
7.6 | IC50 | 3 | — | |
CDHUCXPNWMRKCW
|
7.5 | IC50 | 5 | — | |
CLPXGKIBPZOTAS
|
7.5 | IC50 | 3 | — | |
CPKWWDUXGFBILN
|
7.5 | IC50 | 5 | — | |
USVYMZOVWBQPDX
|
7.5 | IC50 | 3 | — | |
YUQWQAFXEWVXRJ
|
7.5 | IC50 | 3 | — | |
ADTITEYDHLKQCU
|
7.5 | IC50 | 3 | — | |
CARUXIIPTLTRNX
|
7.5 | IC50 | 3 | — | |
CNKVGRHQVUWEFQ
|
7.5 | IC50 | 3 | — | |
KEIPNCCJPRMIAX
|
7.5 | IC50 | 3 | — | |
MOPGLVUDBLCPTB
|
7.5 | IC50 | 4 | — | |
QIRFTSVGPCWENL
|
7.5 | IC50 | 3 | — | |
SCUJGFBGOVGZGU
|
7.5 | IC50 | 3 | — | |
PEJTUNMIBFQQFF
|
7.5 | IC50 | 4 | — | |
ANWHQLGKGDJLJO
|
7.5 | IC50 | 6 | — | |
HLNPWTJAVUGIEO
|
7.5 | IC50 | 5 | — | |
JEMQSZABKSZHQU
|
7.5 | IC50 | 3 | — |