Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XZXJKJYGIPJZNE
|
7.7 | IC50 | 2 | — | |
YVMFSTFAXMETML
|
7.7 | IC50 | 3 | — | |
ZJMNOPJGTBPAJZ
|
7.7 | IC50 | 2 | — | |
ZPKKCQCKJWTLIA
|
7.7 | IC50 | 4 | — | |
HWWQXUZGAMVNAJ
|
7.7 | IC50 | 5 | — | |
KDMGWBBETGCJDN
|
7.7 | IC50 | 5 | — | |
KYUCAVCNFWUMDG
|
7.7 | IC50 | 5 | — | |
XZSXONRVTYXHDG
|
7.7 | IC50 | 5 | — | |
YFVSIFXYGYSXNP
|
7.7 | IC50 | 5 | — | |
BPXQYAXTDCQZHB
|
7.7 | IC50 | 7 | Yes | |
BWALYWIIRRRSEU
|
7.7 | IC50 | 3 | — | |
CLVWKDUSLOCSHG
|
7.7 | IC50 | 3 | — | |
HSDFQCXZKQOGKH
|
7.7 | IC50 | 5 | — | |
LFPRKVXYLRYTJA
|
7.7 | IC50 | 3 | — | |
QJELWMWTMJODCA
|
7.7 | IC50 | 5 | — | |
SGDXIVFGEXXEAO
|
7.7 | IC50 | 3 | — | |
SSCBEDGUPGJMQZ
|
7.7 | IC50 | 3 | — | |
ZHSQXZZMKDUQLK
|
7.7 | IC50 | 7 | — | |
CPIJKYWNBZHZKX
|
7.7 | IC50 | 3 | — | |
GHWXUQIYJKZOLT
|
7.7 | IC50 | 5 | — | |
HVOAVCKNIPEVHJ
|
7.7 | IC50 | 5 | — | |
PQLSSHDPNXYVAQ
|
7.7 | IC50 | 5 | — | |
YHMCTXHAEKLNNV
|
7.7 | IC50 | 5 | — | |
BPLVEFPXYUJTQJ
|
7.7 | IC50 | 4 | — | |
GLJPBDSLDMSNAD
|
7.7 | IC50 | 5 | — | |
IVGKGVVDKSMSSX
|
7.7 | IC50 | 3 | — | |
PKVOTNHPZNFTAB
|
7.7 | IC50 | 3 | — | |
SJDCIGRTECLEPF
|
7.7 | IC50 | 3 | — | |
VYUVGFPNMUTKOT
|
7.7 | IC50 | 3 | — | |
XMAIAGUHQHUOKQ
|
7.7 | IC50 | 3 | — | |
ZIWGJOKZVXLDJP
|
7.7 | IC50 | 3 | — | |
ZJFCBQXPTQSTCZ
|
7.7 | IC50 | 8 | — | |
QUDARNVMIVVBFA
|
7.7 | IC50 | 3 | — | |
SJZFQNLVTDWVLK
|
7.7 | IC50 | 2 | — | |
UMBIRSZUCJNBHB
|
7.7 | IC50 | 18 | — | |
ACJUWCBUAIPYFB
|
7.6 | IC50 | 3 | — | |
CVGMBUVWKDQMIA
|
7.6 | IC50 | 5 | — | |
HKLFXGIFTLYVQG
|
7.6 | IC50 | 3 | — | |
JTZDABVPKBSXNS
|
7.6 | IC50 | 3 | — | |
LUPSYDSJDYGOGY
|
7.6 | IC50 | 6 | Yes | |
NKOQGUAOVGXWMB
|
7.6 | IC50 | 3 | — | |
RBNKCLPELCJMAS
|
7.6 | IC50 | 2 | — | |
TVFMZRKDNNYDFP
|
7.6 | IC50 | 3 | — | |
ZDPPQYBGIHHFAW
|
7.6 | IC50 | 3 | — | |
AFXWEQMFHKVCOA
|
7.6 | IC50 | 3 | — | |
JBMDPQHNWRVKTP
|
7.6 | IC50 | 4 | — | |
OGIVRWCGCBWJHX
|
7.6 | IC50 | 5 | — | |
GRSDVXUJKVFBBM
|
7.6 | IC50 | 3 | — | |
KJZWLNUAUHEQCJ
|
7.6 | IC50 | 5 | — | |
VIRKYOQOEOUNGV
|
7.6 | IC50 | 3 | — |