Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HWZVKJOWBAEUJL
|
7.7 | IC50 | 3 | — | |
HZVSBPHWYBQBIP
|
7.7 | IC50 | 4 | — | |
JCBRKJGZGWDDLQ
|
7.7 | IC50 | 5 | — | |
JPXAJSFXSDRHFJ
|
7.7 | IC50 | 4 | — | |
JQUMKNULUUVBGV
|
7.7 | IC50 | 3 | — | |
JXXRWZVJKWAYOB
|
7.7 | IC50 | 3 | — | |
KLGBMYOAWNNWOT
|
7.7 | IC50 | 4 | — | |
KLMBVSNFAXRHOP
|
7.7 | IC50 | 3 | — | |
LHXHOAYXHBJZAD
|
7.7 | IC50 | 4 | — | |
LMBRUMBIWBMCJS
|
7.7 | IC50 | 4 | — | |
LUXVAUPYQFFUGB
|
7.7 | IC50 | 3 | — | |
LVXNNQUBWPVTEK
|
7.7 | IC50 | 3 | — | |
LYFIGUDTINIDEL
|
7.7 | IC50 | 4 | — | |
MJCHRWOPCVDEGN
|
7.7 | IC50 | 5 | — | |
MLLBUBJPNHKUSB
|
7.7 | IC50 | 4 | — | |
MSYUMSMBBQJIFX
|
7.7 | IC50 | 3 | — | |
MWPSTUHFRRKLNR
|
7.7 | IC50 | 3 | — | |
NDVWJSMBBJDBMM
|
7.7 | IC50 | 3 | — | |
NGHGPCUSBNNBGU
|
7.7 | IC50 | 3 | — | |
NKISUTDCFOPYEO
|
7.7 | IC50 | 3 | — | |
NWWFNKZYJAMTLG
|
7.7 | IC50 | 4 | — | |
NXRULZCRNIWEKE
|
7.7 | IC50 | 2 | — | |
OIYARKAWWFGJEX
|
7.7 | IC50 | 4 | — | |
OXVKMWBTKLBCDB
|
7.7 | IC50 | 3 | — | |
PFHZVQFORDMOSD
|
7.7 | IC50 | 4 | — | |
QJDIPINGKWKAJC
|
7.7 | IC50 | 4 | — | |
QZFSPYWWTHEARH
|
7.7 | IC50 | 3 | — | |
RATYINXGNCNVKD
|
7.7 | IC50 | 4 | — | |
RBGTVSQOBHMSRC
|
7.7 | IC50 | 4 | — | |
SAFNWUDTZOUTKV
|
7.7 | IC50 | 4 | — | |
SBZQKMMAIUJFOD
|
7.7 | IC50 | 4 | — | |
SKBMHHQBJOLYKF
|
7.7 | IC50 | 4 | — | |
SNKUTBKFTWJKTQ
|
7.7 | IC50 | 3 | — | |
SQYPRMZFZUIUJP
|
7.7 | IC50 | 3 | — | |
SSVNQWRWSYYNPM
|
7.7 | IC50 | 2 | — | |
STGSCEBJQRFOSA
|
7.7 | IC50 | 3 | — | |
STUBABXJEIUVID
|
7.7 | IC50 | 4 | — | |
TXTOJSVFWCTYGO
|
7.7 | IC50 | 3 | — | |
UPABTRODRQBAOX
|
7.7 | IC50 | 4 | — | |
URQOCFMHKKPXJG
|
7.7 | IC50 | 5 | — | |
UWOYTCITBQAVIR
|
7.7 | IC50 | 4 | — | |
VDUMAKNUEKYNBY
|
7.7 | IC50 | 4 | — | |
VGWVBGUWLJPSFJ
|
7.7 | IC50 | 3 | — | |
VINKWWCGAXQASJ
|
7.7 | IC50 | 4 | — | |
VUBGMBQEMYBWIS
|
7.7 | IC50 | 4 | — | |
WUYZYWTYHPJTBS
|
7.7 | IC50 | 4 | — | |
XDYKQAGJBSKWDW
|
7.7 | IC50 | 4 | — | |
XHOBSPUMHKAEIP
|
7.7 | IC50 | 4 | — | |
XIYCZVPHJCBKLO
|
7.7 | IC50 | 3 | — | |
XKCXEVPJDHREIR
|
7.7 | IC50 | 3 | — |