Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UQWHJXRXUPVHMN
|
7.8 | IC50 | 3 | — | |
UWABVCHLZLOQNQ
|
7.8 | IC50 | 3 | — | |
VDTUZTRVIPIQEC
|
7.8 | Kd | 3 | — | |
GUEZCEZQFMVREH
|
7.8 | IC50 | 3 | — | |
YXVDEILMUVTDMK
|
7.8 | IC50 | 3 | — | |
KGJGNTKVAMGHGP
|
7.8 | IC50 | 5 | — | |
NSKMAMKHOOUMNN
|
7.8 | IC50 | 3 | — | |
RDDXIDPAWAFIMB
|
7.8 | IC50 | 3 | — | |
WBZQNSDDLQRNJI
|
7.8 | IC50 | 5 | — | |
BUWHPVVMBQAYBT
|
7.7 | IC50 | 3 | — | |
BWVBBQUABJTTLI
|
7.7 | IC50 | 5 | — | |
CUAQIKLHHIWLCQ
|
7.7 | IC50 | 3 | — | |
FIJPTPVDGFMHFC
|
7.7 | IC50 | 3 | — | |
JHNXJFLNZAUFGJ
|
7.7 | IC50 | 3 | — | |
MAXGMZGUSCSCRT
|
7.7 | IC50 | 2 | — | |
QUDARNVMIVVBFA
|
7.7 | IC50 | 3 | — | |
SMAHSHLEAZMURC
|
7.7 | IC50 | 3 | — | |
WYIHKBXXYYTYDX
|
7.7 | IC50 | 3 | — | |
ZSFKGAXZQCZBTJ
|
7.7 | IC50 | 3 | — | |
DXVWDCOHXAEMCI
|
7.7 | IC50 | 3 | — | |
RZRVTNNQCLYNOB
|
7.7 | IC50 | 5 | — | |
SDFCBOWBJRMBSN
|
7.7 | IC50 | 2 | — | |
VOZIDBQIYRSKJX
|
7.7 | IC50 | 3 | — | |
BACJIHHGMXVPAT
|
7.7 | IC50 | 3 | — | |
CMQYMJDTQIBHDE
|
7.7 | IC50 | 3 | — | |
DYRPBDPBCUBZEZ
|
7.7 | IC50 | 3 | — | |
GJZVBYXLNIFOGB
|
7.7 | IC50 | 2 | — | |
OQIOOVKROVOWAL
|
7.7 | IC50 | 3 | — | |
ALDCMWFWAWYYBZ
|
7.7 | IC50 | 2 | — | |
DTNHNJVOHCLYPS
|
7.7 | IC50 | 5 | — | |
FPQZQEVKWJHGCS
|
7.7 | IC50 | 5 | — | |
WRSADQAXUUZHPM
|
7.7 | IC50 | 5 | — | |
XJOQXSSQHKPXSP
|
7.7 | IC50 | 5 | — | |
AMILFCGKIUEALD
|
7.7 | IC50 | 4 | — | |
AYIHTAQUCBAXSB
|
7.7 | IC50 | 3 | — | |
BPJHGOMDDBBUSG
|
7.7 | IC50 | 3 | — | |
BUESLRRHEILKRP
|
7.7 | IC50 | 3 | — | |
CPCQWWLXCICUER
|
7.7 | IC50 | 4 | — | |
CXALXWSKLQJHRX
|
7.7 | IC50 | 3 | — | |
DEMWYUOYYYJCQV
|
7.7 | IC50 | 4 | — | |
DNOZUCALPBNKAF
|
7.7 | IC50 | 3 | — | |
FHMRFTIIYIIJFV
|
7.7 | IC50 | 4 | — | |
FRFMTYIUSMUYBO
|
7.7 | IC50 | 3 | — | |
GIUMENLXKRSSEI
|
7.7 | IC50 | 4 | — | |
GMYCPVQQFIVFGR
|
7.7 | IC50 | 3 | — | |
HFPTTWKUDKQJKO
|
7.7 | IC50 | 4 | — | |
HJBUVPWQDSLNIU
|
7.7 | IC50 | 3 | — | |
HPBZDCWPSLVFFJ
|
7.7 | IC50 | 4 | — | |
HWMZNVOKUYTQOU
|
7.7 | IC50 | 4 | — | |
HWTHFHISUFVKHI
|
7.7 | IC50 | 3 | — |