Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MQTVDWCDNQKMHP
|
7.8 | Kd | 3 | — | |
MTSOIUXASMCNHX
|
7.8 | IC50 | 5 | — | |
NZCCKKOANLHWDZ
|
7.8 | IC50 | 4 | — | |
RALRANHRVZDLCX
|
7.8 | IC50 | 3 | — | |
RGTPQWZZUGUUOY
|
7.8 | IC50 | 3 | — | |
YRFNUGHTYVDUEW
|
7.8 | IC50 | 3 | — | |
IRABEPFZBWUTFB
|
7.8 | IC50 | 5 | — | |
LVRQYRWZIOHHHF
|
7.8 | IC50 | 3 | — | |
NWCCEQWWXCFVQU
|
7.8 | IC50 | 3 | — | |
RUUWTDVRBGAQCD
|
7.8 | IC50 | 3 | — | |
IEZSYOTXLDGZAI
|
7.8 | Kd | 3 | — | |
IMYLSIBTGYMGSC
|
7.8 | Kd | 3 | — | |
INORBDLBUYXJNI
|
7.8 | IC50 | 3 | — | |
JJICTDAMZUTTPX
|
7.8 | IC50 | 3 | — | |
LHHDRTUNEIVZGK
|
7.8 | IC50 | 3 | — | |
NDGUSFBZIMQWNQ
|
7.8 | IC50 | 3 | — | |
NZBLGNHPIFEHLU
|
7.8 | IC50 | 3 | — | |
QSTFLZOOJVWRBM
|
7.8 | IC50 | 3 | — | |
SDZYXIXRAQNGSA
|
7.8 | IC50 | 3 | — | |
SUIFLKARRVDMQC
|
7.8 | IC50 | 3 | — | |
UWOKNQXHVAKWCJ
|
7.8 | IC50 | 5 | — | |
WYPRMGVPTUGHFM
|
7.8 | IC50 | 3 | — | |
XWGYUZGILVRSRS
|
7.8 | IC50 | 5 | — | |
FONDQLCAYMUQPO
|
7.8 | IC50 | 2 | — | |
JXMYXVQTSAHUJU
|
7.8 | IC50 | 2 | — | |
KWCUYDDWUFSZAY
|
7.8 | IC50 | 4 | — | |
MYGXNPCIHRPOSI
|
7.8 | IC50 | 3 | — | |
NEFZONWDMQKLAF
|
7.8 | IC50 | 5 | — | |
WIQBEPAALNQBFG
|
7.8 | IC50 | 3 | — | |
XHSUXSHBEVITPC
|
7.8 | IC50 | 5 | — | |
YZNIJUGKAUSLDO
|
7.8 | IC50 | 2 | — | |
BXBWZDDZLDSYQH
|
7.8 | IC50 | 5 | — | |
CUHPDSMNUKDETF
|
7.8 | IC50 | 3 | — | |
DULFLBNKXBAPSF
|
7.8 | IC50 | 5 | — | |
HIMWRONMJKQVOO
|
7.8 | IC50 | 5 | — | |
KDESKKDZZGVVFB
|
7.8 | IC50 | 2 | — | |
KMTYDGYYZOIXRG
|
7.8 | IC50 | 3 | — | |
QCYDLOHINRAHID
|
7.8 | IC50 | 5 | — | |
SMUWQHVFXRNAMW
|
7.8 | IC50 | 3 | — | |
AREYWCZYVPSHGS
|
7.8 | IC50 | 5 | — | |
CMWXIQFNVQJMQA
|
7.8 | IC50 | 5 | — | |
CVTLXZHZCMNAPK
|
7.8 | Kd | 3 | — | |
DPUPBFOGQNPWHT
|
7.8 | IC50 | 3 | — | |
FIPQREIXXPPEPA
|
7.8 | IC50 | 3 | — | |
IQJPWAAWPFBLPZ
|
7.8 | IC50 | 2 | — | |
JXHPZSZEBLPQKW
|
7.8 | IC50 | 3 | — | |
PNXHAMDNXPTINS
|
7.8 | IC50 | 5 | — | |
QMHOAFNGBZAYPM
|
7.8 | IC50 | 5 | — | |
RVDIEUJUJGRHHU
|
7.8 | IC50 | 3 | — | |
SUHYDZOOTHNRAB
|
7.8 | IC50 | 5 | — |