Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SXVONVWXEBCQAQ
|
7.9 | IC50 | 3 | — | |
GWHKGQOWAXERHA
|
7.9 | IC50 | 3 | — | |
IQAIXSLQDLQWKO
|
7.9 | IC50 | 5 | — | |
JRDGKLCLEFCXSH
|
7.9 | IC50 | 5 | — | |
JVJWECTXCJCFPU
|
7.9 | IC50 | 3 | — | |
KCIGGSIEQASIPY
|
7.9 | IC50 | 2 | — | |
QKZIVVJZESETFG
|
7.9 | IC50 | 3 | — | |
RYLYPXANRHKWKH
|
7.9 | IC50 | 5 | — | |
SMOUPPZEQRHDDS
|
7.9 | IC50 | 5 | — | |
SRQWEDJUTCYYPZ
|
7.9 | IC50 | 5 | — | |
TTZHPWRERCHHAK
|
7.9 | IC50 | 3 | — | |
WLMOBZCQXJLKAR
|
7.9 | IC50 | 5 | — | |
AJGWZFROWJUKON
|
7.9 | IC50 | 5 | — | |
GBXSGEIAMQTWMD
|
7.9 | IC50 | 5 | — | |
NMUMTMSFCTWPOO
|
7.9 | IC50 | 3 | — | |
SSORSGHXGDTLFJ
|
7.9 | IC50 | 5 | — | |
SZRFDSHUSQGOKS
|
7.9 | IC50 | 3 | — | |
VYWXBPWMVHMUQW
|
7.9 | IC50 | 7 | — | |
CBQNTAOEEUWZPV
|
7.9 | IC50 | 3 | — | |
JLVYDBJMHNJJKE
|
7.9 | IC50 | 5 | — | |
GPLOXTXOSLIAOO
|
7.9 | IC50 | 4 | — | |
HVIMAXORBAESDU
|
7.9 | IC50 | 2 | — | |
KSSPOJIRAMTGMO
|
7.9 | IC50 | 5 | — | |
CVOXIJBPYJDKHX
|
7.8 | IC50 | 3 | — | |
KQUZULPXQBSMSS
|
7.8 | IC50 | 5 | — | |
ONDLQNORJPRVQM
|
7.8 | IC50 | 3 | — | |
QNVUTZQLKFYKPS
|
7.8 | IC50 | 5 | — | |
SGDJFAPTKOZVKU
|
7.8 | IC50 | 2 | — | |
SHTARXDORUZIAD
|
7.8 | IC50 | 3 | — | |
YXTPQQRBJPBXQQ
|
7.8 | IC50 | 3 | — | |
ZKJBUNLEWIFNIX
|
7.8 | IC50 | 3 | — | |
BAZVFUXBEXJILA
|
7.8 | IC50 | 5 | — | |
GCDSDVNITVBCDW
|
7.8 | IC50 | 17 | — | |
IBRJKAVHCWQUPP
|
7.8 | IC50 | 3 | — | |
KEAWMUNHKYSQEN
|
7.8 | IC50 | 3 | — | |
SEVOZKSFLJRZMK
|
7.8 | IC50 | 5 | — | |
FUUUVMVISCOTOP
|
7.8 | IC50 | 5 | — | |
IOBVOHPLKSGFCC
|
7.8 | IC50 | 5 | — | |
VIMGDHNUHDOJNR
|
7.8 | IC50 | 5 | — | |
BTHCJMVMWFFHPR
|
7.8 | IC50 | 4 | — | |
CCDNYIWGTYFDSI
|
7.8 | IC50 | 5 | — | |
CDOLGQDRZSLRFK
|
7.8 | IC50 | 3 | — | |
CJVVXRNKGDZSSX
|
7.8 | IC50 | 3 | — | |
CQDXYQFRLSRPQH
|
7.8 | IC50 | 5 | — | |
CTTRKDHLWWJCCI
|
7.8 | IC50 | 3 | — | |
GEIITDFWTJJONU
|
7.8 | IC50 | 5 | — | |
GHHZJQUAHVVLOV
|
7.8 | IC50 | 4 | — | |
JYZXTSDUMOPSSZ
|
7.8 | Kd | 3 | — | |
KJGQZAPNEIXLDS
|
7.8 | IC50 | 3 | — | |
LZUCMYASLOBNKP
|
7.8 | IC50 | 3 | — |