Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KQAKIPZTLWPTMC
|
8.0 | IC50 | 3 | — | |
LYADGAGFYYXXIO
|
8.0 | IC50 | 82 | — | |
OSZVHJYNXBUVAH
|
8.0 | IC50 | 12 | — | |
QHBVJFHZCWJZPO
|
8.0 | IC50 | 3 | — | |
TUJGAAZZROOKNS
|
8.0 | IC50 | 3 | — | |
WOSKHXYHFSIKNG
|
8.0 | IC50 | 24 | — | |
XEZPJZVKUKRDDU
|
8.0 | IC50 | 3 | — | |
ZHJNDQAMSAUBBB
|
8.0 | IC50 | 3 | — | |
ZKQWBIBGYRHIPV
|
8.0 | IC50 | 3 | — | |
BDKJDXXVJPMWPB
|
8.0 | IC50 | 3 | — | |
DCPCRIARGMFUEP
|
8.0 | IC50 | 5 | — | |
IVRYMOBVZPFZQJ
|
8.0 | IC50 | 5 | — | |
YRNGUNZRBVYKCB
|
8.0 | IC50 | 3 | — | |
YXFWKMCVZXUIMK
|
8.0 | IC50 | 5 | — | |
IJENXCZIMOXLKN
|
7.9 | IC50 | 5 | — | |
IQQVSAGBFNJDMB
|
7.9 | IC50 | 5 | — | |
RFJKJMVXZQNREI
|
7.9 | IC50 | 5 | — | |
IHWSMDNQFDZGTJ
|
7.9 | IC50 | 5 | — | |
LFTXCKTUPGWQGQ
|
7.9 | IC50 | 3 | — | |
RYNCXRBJRSKWJE
|
7.9 | IC50 | 5 | — | |
WXCQNRFWIHJMLJ
|
7.9 | IC50 | 5 | — | |
AJQGJOSWZUAVFV
|
7.9 | IC50 | 3 | — | |
DCWCFKXCIYCNTA
|
7.9 | IC50 | 3 | — | |
DGLQLMVKZQVYDS
|
7.9 | IC50 | 3 | — | |
DPSDPDLIGHEHRB
|
7.9 | IC50 | 3 | — | |
HFFXKEYAEKHCQX
|
7.9 | IC50 | 3 | — | |
IGWDLODVRIEGNQ
|
7.9 | IC50 | 3 | — | |
KNPLSRBVKFTLQU
|
7.9 | IC50 | 3 | — | |
KTMMZCLUGNPLAT
|
7.9 | IC50 | 3 | — | |
LXTAEWHGOAKRPZ
|
7.9 | IC50 | 3 | — | |
MQYOWYIEYBIMAM
|
7.9 | IC50 | 3 | — | |
MUDOCUNTLILGNS
|
7.9 | IC50 | 5 | — | |
NCPSPEUSGOPVQV
|
7.9 | IC50 | 5 | — | |
TVBYDWWNVYOOIA
|
7.9 | IC50 | 3 | — | |
UCUKGOVQHPVFAN
|
7.9 | IC50 | 5 | — | |
XIGWDTLDLMHFCU
|
7.9 | IC50 | 3 | — | |
YDQIGYMEVQJYJF
|
7.9 | IC50 | 3 | — | |
DFRRHNQYSACYDX
|
7.9 | IC50 | 5 | — | |
GITYCPDVBYJBGY
|
7.9 | IC50 | 3 | — | |
OMNISBCHBVYMCT
|
7.9 | IC50 | 5 | — | |
ORUNGMOTBJGTPU
|
7.9 | IC50 | 5 | — | |
PPFQKJGJQXSDJS
|
7.9 | IC50 | 5 | — | |
SGPDKZMOPAHQPP
|
7.9 | IC50 | 5 | — | |
WJQLXQXBPJJDTC
|
7.9 | IC50 | 4 | — | |
XOAPPSGARFEIQW
|
7.9 | IC50 | 5 | — | |
YIDCCLXYFLNYHA
|
7.9 | IC50 | 5 | — | |
HXKRTTRYDVNOTH
|
7.9 | IC50 | 2 | — | |
LYCYMSYZZMMABC
|
7.9 | IC50 | 3 | — | |
MBVVTXSJBVWMFV
|
7.9 | IC50 | 5 | — | |
NKOUTELHRIQKFT
|
7.9 | IC50 | 4 | — |