Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YIZQBOQRVQNOOF
|
9.1 | IC50 | 2 | — | |
FDYYKFWGYGBXLY
|
9.1 | IC50 | 4 | — | |
JCHUZEULHHBDND
|
9.1 | IC50 | 4 | — | |
UIUUIHADIPAKSK
|
9.1 | IC50 | 5 | — | |
XNRZJGZKJIEPIW
|
9.1 | IC50 | 3 | — | |
CBHANRIYVOOCIB
|
9.0 | IC50 | 2 | — | |
NYJMVCWYBMPHTD
|
9.0 | IC50 | 4 | — | |
BAUFTYOWRVUSNA
|
9.0 | IC50 | 2 | — | |
POMPWDXYMSRSAW
|
9.0 | IC50 | 4 | — | |
QKQUURVQHYEPRX
|
9.0 | IC50 | 2 | — | |
OYJDTEBZSGLLNC
|
9.0 | IC50 | 2 | — | |
CCUVJTVUUVQKFK
|
9.0 | IC50 | 3 | — | |
CYHGHBQCTXVJCN
|
9.0 | IC50 | 3 | — | |
NFYDPTASEPAEMT
|
9.0 | IC50 | 4 | — | |
NKNHEZFIUHHBJX
|
9.0 | IC50 | 3 | — | |
PQBDYJCATQLIFW
|
9.0 | IC50 | 2 | — | |
SJEVLHTYUBABDJ
|
9.0 | IC50 | 4 | — | |
URIOWDLDOGYPLK
|
9.0 | IC50 | 2 | — | |
VLXIXYDIKYYMAQ
|
9.0 | IC50 | 7 | — | |
XKKGIGFZDVPVNO
|
9.0 | IC50 | 4 | — | |
XKKGIGFZDVPVNO
|
9.0 | IC50 | 4 | — | |
YTDWYXQAKOWNAV
|
9.0 | IC50 | 4 | — | |
HCDBDJBZIKAUDL
|
9.0 | IC50 | 2 | — | |
USCLDZNWLVHDPF
|
9.0 | IC50 | 5 | — | |
WRLCMSJRWBXEIO
|
9.0 | IC50 | 4 | — | |
ACXLCIADWYPDHD
|
9.0 | IC50 | 2 | — | |
AMXKOAUPVJWSGA
|
9.0 | IC50 | 3 | — | |
GYXODBZTJVUDOH
|
9.0 | IC50 | 4 | — | |
SENVOZNIDWYYED
|
9.0 | IC50 | 4 | — | |
ZYBQELLBNQSEEB
|
9.0 | IC50 | 2 | — | |
QLCFILNKJFBLGJ
|
8.9 | IC50 | 2 | — | |
SPQDHLUXHUIWBR
|
8.9 | IC50 | 2 | — | |
MAMVVNACJMPVQQ
|
8.9 | IC50 | 5 | — | |
FHDKNSAADPLWFU
|
8.9 | IC50 | 2 | — | |
PZMMTZOZIZQHCK
|
8.9 | IC50 | 2 | — | |
USRVMHONXWVKPD
|
8.9 | IC50 | 4 | — | |
VDTUZTRVIPIQEC
|
8.9 | Kd | 3 | — | |
WWGLOQFMJUZFTJ
|
8.9 | IC50 | 8 | — | |
ZQTUTQJCMVRZQW
|
8.9 | IC50 | 2 | — | |
BZFULTDZKYXUOC
|
8.9 | IC50 | 5 | — | |
QLONORAXWCHYSN
|
8.9 | IC50 | 4 | — | |
RNLCEYKRDCFQPX
|
8.9 | IC50 | 2 | — | |
KEIPNCCJPRMIAX
|
8.9 | IC50 | 5 | — | |
KPBLASRJMVBLEW
|
8.9 | IC50 | 3 | — | |
LJJPNXWNMVOUCI
|
8.9 | IC50 | 2 | — | |
LTWBXHYYWOPFGA
|
8.9 | IC50 | 2 | — | |
PUIXMSRTTHLNKI
|
8.9 | IC50 | 12 | — | |
QNXOYMFBIACDSL
|
8.9 | IC50 | 5 | — | |
YWDKSGWRKAMORO
|
8.9 | IC50 | 5 | — | |
ZMSXGEYSNDHGJO
|
8.9 | IC50 | 3 | — |