Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UPGIHICOGVAEBN
|
8.1 | IC50 | 2 | — | |
XFGMNTTVFYLJIS
|
8.1 | IC50 | 2 | — | |
XHCHGZHSYDYRKE
|
8.1 | IC50 | 3 | — | |
YCKCPZLJEACLLQ
|
8.1 | IC50 | 5 | — | |
FIFDRXCJFUTRRL
|
8.1 | IC50 | 5 | — | |
FMWDLYTVSRVYQS
|
8.1 | IC50 | 5 | — | |
GEEWFYSWIUQFGV
|
8.1 | IC50 | 5 | — | |
GFZIDFHTIFIOOM
|
8.1 | IC50 | 5 | — | |
HDUMTFLTRMYGKD
|
8.1 | IC50 | 3 | — | |
LIHHZURFBCGBNP
|
8.1 | IC50 | 3 | — | |
MWMHYAXGYUGPBU
|
8.1 | IC50 | 5 | — | |
SVPYHIXSUHWOCA
|
8.1 | IC50 | 5 | — | |
FXUDALBVHPNJCZ
|
8.1 | IC50 | 2 | — | |
HEVVAJIKBWBWSD
|
8.1 | IC50 | 3 | — | |
JBJLDYOTZAKYCV
|
8.1 | IC50 | 5 | — | |
JHRJOTWCULWCKL
|
8.1 | IC50 | 2 | — | |
NGLRSTVZLVHSJO
|
8.1 | IC50 | 5 | — | |
NOOKOYPSNNYWOH
|
8.1 | IC50 | 5 | — | |
RBZPOZTUZQJYKH
|
8.1 | IC50 | 3 | — | |
AGBXUKHUCRHKSZ
|
8.1 | IC50 | 6 | — | |
FACLICQSXLCKBZ
|
8.1 | IC50 | 3 | — | |
GTZRCWSMTBJVNU
|
8.1 | IC50 | 3 | — | |
GWOHWBYOVFLZGM
|
8.1 | IC50 | 2 | — | |
JOAFWIHZEBKYQK
|
8.1 | IC50 | 10 | — | |
KHTGGYNVCUTUEK
|
8.1 | IC50 | 3 | — | |
SPXNVPJERGMJSD
|
8.1 | IC50 | 3 | — | |
SWKVBTAXZKMYFH
|
8.1 | IC50 | 5 | — | |
XNCPXNXXBVMOTI
|
8.1 | IC50 | 5 | — | |
XPKLWQVCOXZZKV
|
8.1 | IC50 | 5 | — | |
XRLFKHYILNWINJ
|
8.1 | IC50 | 3 | — | |
XVPPCNTYUSCWJA
|
8.1 | IC50 | 3 | — | |
CHRFXWRFOHSHLD
|
8.1 | IC50 | 5 | — | |
KEJHKWDFKQXLMG
|
8.1 | IC50 | 2 | — | |
NTPSXOIFCGNPHC
|
8.1 | IC50 | 3 | — | |
PRMCZXTVLDRKKA
|
8.1 | IC50 | 5 | — | |
UZVFQJWFEJNXPR
|
8.1 | IC50 | 5 | — | |
AMMKZXLXQZTHBG
|
8.1 | IC50 | 5 | — | |
JFKAABZHYCNZIU
|
8.1 | IC50 | 3 | — | |
JQLWGEZBIJYETF
|
8.1 | IC50 | 3 | — | |
MLQQTOJZLDQPMV
|
8.1 | IC50 | 5 | — | |
PPFXHUHUMARHQF
|
8.1 | IC50 | 3 | — | |
RFPCUHZRLMHSTG
|
8.1 | IC50 | 5 | — | |
SGHUCPHHNVDAPN
|
8.1 | IC50 | 5 | — | |
SRNXPZGAZRUEQV
|
8.1 | IC50 | 3 | — | |
ULTCGGKUGQUOMR
|
8.1 | IC50 | 5 | — | |
UQWOQACFVFKPQK
|
8.1 | IC50 | 3 | — | |
BRKGRQVBHFZISR
|
8.0 | IC50 | 7 | Yes | |
JQUMBFRGCVDDBS
|
8.0 | IC50 | 5 | — | |
POHLKOAYIRHFFP
|
8.0 | IC50 | 5 | — | |
QNIMLRHYPMIYSE
|
8.0 | IC50 | 7 | Yes |