Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JGAIVBOWNPLAHY
|
8.1 | IC50 | 3 | — | |
JJPFEPQJBUBRFW
|
8.1 | IC50 | 5 | — | |
LNZDHCYDEDDMTH
|
8.1 | IC50 | 5 | — | |
OACFIPDTGXZIQH
|
8.1 | IC50 | 2 | — | |
OQWGMALEKOUCHV
|
8.1 | IC50 | 5 | — | |
RWMCOWYHZFANLF
|
8.1 | IC50 | 5 | — | |
UTGWNSVMZBOYIX
|
8.1 | IC50 | 5 | — | |
VBMZPUMENVSUEK
|
8.1 | IC50 | 2 | — | |
YRIBONQFXXVSAU
|
8.1 | IC50 | 5 | — | |
ZWDPQCVFSJWCFD
|
8.1 | IC50 | 2 | — | |
AHWOGVXLWKIELS
|
8.1 | IC50 | 5 | — | |
KZMWAICISUWYLE
|
8.1 | IC50 | 7 | — | |
MNPLRCNUAOZMSC
|
8.1 | IC50 | 2 | — | |
MSSUJWPHHVXXFT
|
8.1 | IC50 | 5 | — | |
OOJCSNDQUFLDIN
|
8.1 | IC50 | 2 | — | |
RBVQYTAEUBJSEY
|
8.1 | IC50 | 5 | — | |
RGYNBLDJVUWGQS
|
8.1 | IC50 | 5 | — | |
YMXQQOATOHFDLF
|
8.1 | IC50 | 5 | — | |
ZQTRKQPFZQBOMV
|
8.1 | IC50 | 2 | — | |
AHWOGVXLWKIELS
|
8.1 | IC50 | 5 | — | |
AXWXBTUICOYCLL
|
8.1 | IC50 | 5 | — | |
BEMNJULZEQTDJY
|
8.1 | IC50 | 8 | — | |
FCTVEMBOSZJMAX
|
8.1 | IC50 | 3 | — | |
FRZMZARFJKOYRE
|
8.1 | IC50 | 3 | — | |
GYSNMOKUABWZLQ
|
8.1 | IC50 | 3 | — | |
IQAIXSLQDLQWKO
|
8.1 | IC50 | 5 | — | |
MVIXBPATNRRIAA
|
8.1 | IC50 | 5 | — | |
PFPXVMRFOYULPT
|
8.1 | IC50 | 7 | Yes | |
SLLCQDKQRQLXEO
|
8.1 | IC50 | 3 | — | |
SOYCCBHGJYSWNQ
|
8.1 | IC50 | 5 | — | |
SRQIALHPCHADMP
|
8.1 | IC50 | 5 | — | |
BLWLIINBFDOXAP
|
8.1 | IC50 | 3 | — | |
BSINISOJOVJBAT
|
8.1 | IC50 | 5 | — | |
CUMCBEDCPQGOTJ
|
8.1 | IC50 | 5 | — | |
HZIAJKJBTRYTIC
|
8.1 | IC50 | 2 | — | |
JXGGHGLZZYBWNG
|
8.1 | IC50 | 5 | — | |
LNQLFTIOPSWROW
|
8.1 | IC50 | 3 | — | |
QTLLHDXOVYFXTM
|
8.1 | IC50 | 5 | — | |
ULZYEHHPVPISAH
|
8.1 | IC50 | 3 | — | |
YPAFPGOEBJGULD
|
8.1 | IC50 | 5 | — | |
BUICZXSBPLFBKK
|
8.1 | IC50 | 5 | — | |
DJSACWHIHAUSKQ
|
8.1 | IC50 | 3 | — | |
FOJJNIMHMLFIAZ
|
8.1 | IC50 | 3 | — | |
HGZFXVSSFDAUID
|
8.1 | IC50 | 3 | — | |
KDFJDPRUNMUDND
|
8.1 | IC50 | 3 | — | |
MXBVFLPGICOUHO
|
8.1 | IC50 | 3 | — | |
NYIBFGMWXRONJG
|
8.1 | IC50 | 2 | — | |
RELFWZSPSNCGEI
|
8.1 | IC50 | 3 | — | |
UAHJXPBYRPDINJ
|
8.1 | IC50 | 2 | — | |
UKYJKXMPIDEQFF
|
8.1 | IC50 | 16 | — |