Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RCKYRBVOWKAURY
|
8.2 | IC50 | 5 | — | |
RZKSYYNMHKFROG
|
8.2 | IC50 | 5 | — | |
UHXFZAJAHLALQP
|
8.2 | IC50 | 5 | — | |
UYKJFPOYPRLHCO
|
8.2 | IC50 | 3 | — | |
WEYMBVBPABXYAP
|
8.2 | IC50 | 3 | — | |
WTEYUYQDYILCNS
|
8.2 | IC50 | 5 | — | |
YVNMVJWJGAAQLE
|
8.2 | IC50 | 5 | — | |
DXQBCGUEDOHNHP
|
8.2 | IC50 | 12 | — | |
GKINEURMFPNAJS
|
8.2 | IC50 | 2 | — | |
GXIHBWCRCZNSHX
|
8.2 | IC50 | 3 | — | |
IWPIUSKMWHWQQF
|
8.2 | IC50 | 5 | — | |
LMNYJDMVSCGLHG
|
8.2 | IC50 | 5 | — | |
MJMIZDWOYMOFDX
|
8.2 | IC50 | 3 | — | |
OCAAZMTTXWHARF
|
8.2 | IC50 | 3 | — | |
OSPKANQURMXUIE
|
8.2 | IC50 | 7 | Yes | |
OXJWXQVCCWDQJS
|
8.2 | IC50 | 6 | — | |
RELGFRXCVJYWMA
|
8.2 | IC50 | 5 | — | |
TWEPCUUZZJESFX
|
8.2 | IC50 | 3 | — | |
UOCJRPUXXNKLHL
|
8.2 | IC50 | 3 | — | |
FZFKBDZAXOFANZ
|
8.2 | IC50 | 2 | — | |
NTPSXOIFCGNPHC
|
8.2 | IC50 | 3 | — | |
USWTXIMYBIOVHO
|
8.2 | IC50 | 5 | — | |
DDSWQEAKOABACX
|
8.2 | IC50 | 3 | — | |
KMUSZSJDHZHXQA
|
8.2 | IC50 | 4 | — | |
NTSVKEPNLGDQBL
|
8.2 | IC50 | 5 | — | |
RBVQYTAEUBJSEY
|
8.2 | IC50 | 5 | — | |
XZWWCRJOEPEAFT
|
8.2 | IC50 | 3 | — | |
YYBZWPUIOONRPU
|
8.2 | IC50 | 2 | — | |
AHEDUFSEDRFCTH
|
8.2 | IC50 | 4 | — | |
AJGWZFROWJUKON
|
8.2 | IC50 | 5 | — | |
CAMOGMXHVRSGKE
|
8.2 | IC50 | 5 | — | |
DNIRANACJWUPII
|
8.2 | IC50 | 5 | — | |
DXCUKNQANPLTEJ
|
8.2 | IC50 | 7 | — | |
GXMSDNOAHZYMEL
|
8.2 | IC50 | 3 | — | |
GYNREAFZDKMQML
|
8.2 | IC50 | 3 | — | |
GZNXUSKIWXUYJZ
|
8.2 | IC50 | 3 | — | |
HNVRKBGXTRVLEI
|
8.2 | IC50 | 5 | — | |
MBGSKLWXWZBIRH
|
8.2 | IC50 | 3 | — | |
MYFRXSIWRAGTKV
|
8.2 | IC50 | 5 | — | |
OTMSABHPICNCIU
|
8.2 | IC50 | 3 | — | |
SEHOCSFHPAZLLH
|
8.2 | IC50 | 2 | — | |
TUKVBIHBLUMARN
|
8.2 | IC50 | 3 | — | |
UVKSSOACQPJGBB
|
8.2 | IC50 | 2 | — | |
XEZPJZVKUKRDDU
|
8.2 | IC50 | 3 | — | |
XHCHGZHSYDYRKE
|
8.2 | IC50 | 3 | — | |
ZZTNIXAOUAZNRE
|
8.2 | IC50 | 3 | — | |
BIEQCIXMEKROFP
|
8.1 | IC50 | 5 | — | |
GUOKMFDFLUGBPS
|
8.1 | IC50 | 7 | Yes | |
HRMKTZOBLPIBBW
|
8.1 | IC50 | 5 | — | |
IJOGTDNCYKJLOQ
|
8.1 | IC50 | 2 | — |