Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JXGGHGLZZYBWNG
|
8.2 | IC50 | 5 | — | |
YXAFWGPKAAKJHB
|
8.2 | IC50 | 5 | — | |
CUCIPRWCHXEPLX
|
8.2 | IC50 | 3 | — | |
DEEQWPIMFASFIP
|
8.2 | IC50 | 7 | Yes | |
FORDNJPIBXTMHT
|
8.2 | IC50 | 3 | — | |
JAYZLGOACZERIJ
|
8.2 | IC50 | 7 | Yes | |
JJICTDAMZUTTPX
|
8.2 | IC50 | 3 | — | |
NDGPXJXKLJJMFA
|
8.2 | IC50 | 3 | — | |
NEHXATHNSBBFDN
|
8.2 | IC50 | 5 | — | |
OSQLADYCJATFGA
|
8.2 | IC50 | 5 | — | |
OTMSABHPICNCIU
|
8.2 | IC50 | 3 | — | |
OTMSABHPICNCIU
|
8.2 | IC50 | 3 | — | |
QFUNEGRJTMMWQQ
|
8.2 | IC50 | 3 | — | |
QTMASMKMHNYBIC
|
8.2 | IC50 | 8 | Yes | |
QYDBJBJRCCHDBO
|
8.2 | IC50 | 3 | — | |
RJQYZMQDDGYSNW
|
8.2 | IC50 | 3 | — | |
STIFXGYUQWOWOQ
|
8.2 | IC50 | 3 | — | |
UVZKMOOZAKKRIJ
|
8.2 | IC50 | 3 | — | |
VEXULJTWOHELIA
|
8.2 | IC50 | 3 | — | |
XPJRQSVFOCSTQP
|
8.2 | IC50 | 3 | — | |
YBKOSRJNQSSJLC
|
8.2 | IC50 | 3 | — | |
YIDCCLXYFLNYHA
|
8.2 | IC50 | 5 | — | |
YRZKWAVVXPFIAT
|
8.2 | IC50 | 3 | — | |
AVUXLVYBASDKOX
|
8.2 | IC50 | 3 | — | |
IRVNUYFGIYEUAJ
|
8.2 | IC50 | 3 | — | |
NGFDOSWCXMLIIZ
|
8.2 | IC50 | 3 | — | |
OIAKQMVWXQYUFN
|
8.2 | IC50 | 2 | — | |
SOYCCBHGJYSWNQ
|
8.2 | IC50 | 5 | — | |
SSKBZCVOJJPLPP
|
8.2 | IC50 | 4 | — | |
UEOZGCZDSDHALE
|
8.2 | IC50 | 5 | — | |
ULLHSHIOCWGUPY
|
8.2 | IC50 | 3 | — | |
VPPBOEWOJRAJQM
|
8.2 | IC50 | 3 | — | |
VUDMYIHKNCGYRY
|
8.2 | IC50 | 3 | — | |
VUZFQBIKLRQDMD
|
8.2 | IC50 | 5 | — | |
ZMWVHMVSBKMRAW
|
8.2 | IC50 | 5 | — | |
AERNXUFRWJPKGR
|
8.2 | IC50 | 2 | — | |
GZRXWBJYUJUZNW
|
8.2 | IC50 | 3 | — | |
JXIJAMJJVILNQM
|
8.2 | IC50 | 3 | — | |
QWHOKJPXXTWASQ
|
8.2 | IC50 | 3 | — | |
UHPWIGXTFQRPCG
|
8.2 | IC50 | 5 | — | |
XNZSWBJDMRZZJL
|
8.2 | IC50 | 5 | — | |
XXMPSIKGMRIEIG
|
8.2 | IC50 | 5 | — | |
BPRHSQUDWOTSSU
|
8.2 | IC50 | 5 | — | |
BZKQOMNNFFOFRA
|
8.2 | IC50 | 5 | — | |
CMZLRIQSLLGABB
|
8.2 | IC50 | 3 | — | |
DDNOUEXAVDQPMR
|
8.2 | IC50 | 5 | — | |
DSBPVMDUESDKNK
|
8.2 | IC50 | 9 | Yes | |
GWOHWBYOVFLZGM
|
8.2 | IC50 | 2 | — | |
IMRAJPPXPOXARE
|
8.2 | IC50 | 5 | — | |
NCKMZTUTGFIFTA
|
8.2 | IC50 | 5 | — |