Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZLAPDNQBMPUQNA
|
8.3 | IC50 | 3 | — | |
BMRGVWYMLHCENU
|
8.3 | IC50 | 5 | — | |
IBHOLSBDZMIPPT
|
8.3 | IC50 | 5 | — | |
KXSVTQYXRGDXLW
|
8.3 | IC50 | 4 | — | |
MRSBZNMRJKJWIX
|
8.3 | IC50 | 5 | — | |
MZLXXVIDRYUZIM
|
8.3 | IC50 | 5 | — | |
ONSIKNVJAKVKOG
|
8.3 | IC50 | 5 | — | |
RUEUJHIYTXZELK
|
8.3 | IC50 | 5 | — | |
RZQBKZYEBJUPTF
|
8.3 | IC50 | 5 | — | |
CBBWGFHEXFNSKG
|
8.3 | IC50 | 5 | — | |
FINBKAHPSHPPIO
|
8.3 | IC50 | 5 | — | |
GNLBGLKGCLZAOZ
|
8.3 | IC50 | 2 | — | |
HHILMGVBNVWONY
|
8.3 | IC50 | 3 | — | |
HXHAJRMTJXHJJZ
|
8.3 | IC50 | 52 | Yes | |
KVOZGEJRFWGHFZ
|
8.3 | IC50 | 4 | — | |
NRBSFHSUWBAYCI
|
8.3 | IC50 | 5 | — | |
NTCROAMSHNBTJA
|
8.3 | IC50 | 5 | — | |
NYYKCMGNIZNHAN
|
8.3 | IC50 | 5 | — | |
QAGLJDWYCCJEHH
|
8.3 | IC50 | 7 | Yes | |
VITKBUDPMVQPFZ
|
8.3 | IC50 | 5 | — | |
WRABCNDMFRHWIR
|
8.3 | IC50 | 6 | — | |
XUDRPPZFODNIIN
|
8.3 | IC50 | 5 | — | |
ZXPUNZSPQJIHJB
|
8.3 | IC50 | 5 | — | |
WOMBJJKPVIDFFI
|
8.3 | IC50 | 4 | — | |
XPJZNFSHCZZAQF
|
8.3 | IC50 | 3 | — | |
ALBDTYWVJPCHKL
|
8.3 | IC50 | 5 | — | |
DBFMFHYDGXJVLJ
|
8.3 | IC50 | 5 | — | |
IJNFMKJSNQLEOT
|
8.3 | IC50 | 5 | — | |
KHSGFGUZFDJBCR
|
8.3 | IC50 | 3 | — | |
KUVWKWBBXWESBE
|
8.3 | IC50 | 3 | — | |
NCHRMJWKKXNHAK
|
8.3 | IC50 | 3 | — | |
QAXXFBBSSGFFAE
|
8.3 | IC50 | 3 | — | |
WHKAUZLLCXOVEV
|
8.3 | IC50 | 5 | — | |
WVXNSAVVKYZVOE
|
8.3 | IC50 | 92 | — | |
CCWQRQKDZAKBBS
|
8.2 | IC50 | 6 | — | |
HEIWGGHLGABSLB
|
8.2 | Kd | 10 | — | |
JXPPMHWXIOAVMA
|
8.2 | IC50 | 5 | — | |
KKOOCJNBZXZVFR
|
8.2 | IC50 | 5 | — | |
MBFNJGNWXZAXKI
|
8.2 | IC50 | 2 | — | |
OOWSKBMTGLHFAR
|
8.2 | IC50 | 5 | — | |
SWJBPGCYSKADTC
|
8.2 | IC50 | 3 | — | |
YAQMWABNMQSFJS
|
8.2 | IC50 | 3 | — | |
CLOKTLNQBBIROQ
|
8.2 | IC50 | 5 | — | |
DBHJLUJUJXVKKB
|
8.2 | IC50 | 5 | — | |
HKSZLNNOFSGOKW
|
8.2 | IC50 | 408 | — | |
HLRBIOMHENPNQT
|
8.2 | IC50 | 3 | — | |
PLBQTNASSCLIRL
|
8.2 | IC50 | 5 | — | |
SBJBNKSOBUWICX
|
8.2 | IC50 | 5 | — | |
VSHIWUXLTDVVEO
|
8.2 | IC50 | 3 | — | |
BJRANMBFDCJTTQ
|
8.2 | IC50 | 5 | — |