Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UGEHMFOAQXSJDX
|
8.4 | IC50 | 5 | — | |
XALXWJVCZUHIBS
|
8.4 | IC50 | 3 | — | |
YZFIDVOGSPMNRW
|
8.4 | IC50 | 5 | — | |
BQXBOPDGBZRCFL
|
8.4 | IC50 | 5 | — | |
BXMUZNHPFQUNSZ
|
8.4 | IC50 | 5 | — | |
DKJBIJZRZMXJAG
|
8.4 | IC50 | 5 | — | |
DSBGPNZCYAOULK
|
8.4 | IC50 | 2 | — | |
GVEQLTBABUNRMS
|
8.4 | IC50 | 2 | — | |
IVVNCQGZOKJKEC
|
8.4 | IC50 | 5 | — | |
JPJVHSSGRZKSDJ
|
8.4 | IC50 | 5 | — | |
LNJMXIZSFNEQQF
|
8.4 | IC50 | 4 | — | |
MIAPCUPTSBUFIH
|
8.4 | IC50 | 5 | — | |
MJZLZOOCTKZOHS
|
8.4 | IC50 | 5 | — | |
NCJIBESSDGQBKH
|
8.4 | IC50 | 5 | — | |
SARNRLIVUZSXNG
|
8.4 | IC50 | 5 | — | |
SIHZJQZSPAIYMX
|
8.4 | IC50 | 4 | — | |
UZZUQDLJRHRISA
|
8.4 | Kd | 3 | — | |
YEIRROBVFZDCIW
|
8.4 | IC50 | 7 | — | |
YKAWIHSYTZKAKA
|
8.4 | IC50 | 5 | — | |
YXFOOAQCZMCCOW
|
8.4 | IC50 | 5 | — | |
ITALYUWJRXCJRQ
|
8.3 | IC50 | 5 | — | |
JIDWYSMCSIWSQL
|
8.3 | IC50 | 5 | — | |
JKEDZMIFSJMZHH
|
8.3 | IC50 | 2 | — | |
MPXSKHFKEUVGAU
|
8.3 | IC50 | 5 | — | |
NSRRVSVPEXCSGE
|
8.3 | IC50 | 5 | — | |
NYBWRPLFCRQSSV
|
8.3 | IC50 | 5 | — | |
OIYSNFGRVNTTAT
|
8.3 | IC50 | 3 | — | |
OWLHHVGNWXMBFF
|
8.3 | IC50 | 2 | — | |
XIQQPHOWVZOQQP
|
8.3 | IC50 | 4 | — | |
JVHRYVZNKJPNLU
|
8.3 | IC50 | 5 | — | |
NDXXZPUMKRBNQB
|
8.3 | IC50 | 3 | — | |
NXQWBKIKMLKVOS
|
8.3 | IC50 | 5 | — | |
OJURKTZIXKTKOA
|
8.3 | IC50 | 5 | — | |
PLKAJXMYXBXIGX
|
8.3 | IC50 | 7 | Yes | |
RVNHZXXYNAWXJQ
|
8.3 | IC50 | 5 | — | |
SHMLFYDRRWCODZ
|
8.3 | IC50 | 5 | — | |
SIXYJXHMORMEHB
|
8.3 | IC50 | 5 | — | |
DXQAUQWASZIRTJ
|
8.3 | IC50 | 2 | — | |
FVUYKZNGSHSNBI
|
8.3 | IC50 | 5 | — | |
ICBLVWSVBHFPJP
|
8.3 | IC50 | 5 | — | |
LTKSJPZMTYBCRM
|
8.3 | IC50 | 2 | — | |
NOCCEPOVUSRFDS
|
8.3 | IC50 | 5 | — | |
PRHQXNORMNLDST
|
8.3 | IC50 | 5 | — | |
SQPOQDJDYNYPIZ
|
8.3 | IC50 | 5 | — | |
WAKJUGXHBUNUIT
|
8.3 | IC50 | 5 | — | |
WJZSUSVUKVZGLF
|
8.3 | IC50 | 7 | Yes | |
WOGGKLMGFJJKGY
|
8.3 | IC50 | 5 | — | |
ARDLUUQELBPNNT
|
8.3 | IC50 | 5 | — | |
PJULDAZFBKZYLU
|
8.3 | IC50 | 5 | — | |
SRAFQIWHQBJFJJ
|
8.3 | IC50 | 2 | — |