Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TTXZUQMGQAGEFO
|
8.4 | IC50 | 5 | — | |
XIRSUXKSURTZHN
|
8.4 | IC50 | 5 | — | |
ANMVTYAYYHHSTF
|
8.4 | IC50 | 2 | — | |
CLPZHWNOBVVCEB
|
8.4 | IC50 | 5 | — | |
CWYNPLCFBQOJSH
|
8.4 | IC50 | 3 | — | |
DOWDUUHTYDZTMS
|
8.4 | IC50 | 3 | — | |
GLYUIGNYFSCICA
|
8.4 | IC50 | 2 | — | |
GXMSDNOAHZYMEL
|
8.4 | IC50 | 3 | — | |
HAMQGTWNMUEACH
|
8.4 | IC50 | 5 | — | |
HEAOOEBHFBBENP
|
8.4 | IC50 | 3 | — | |
HYTKNUZBKDBMMN
|
8.4 | IC50 | 5 | — | |
INORBDLBUYXJNI
|
8.4 | IC50 | 3 | — | |
INWHLZUNIJSPHA
|
8.4 | IC50 | 5 | — | |
JQYPWJCACYTKIC
|
8.4 | IC50 | 5 | — | |
KFKMPCWDJDVUQL
|
8.4 | IC50 | 5 | — | |
KVNSXBAQSWMTDX
|
8.4 | IC50 | 2 | — | |
LCAJAFNIVVFNGM
|
8.4 | IC50 | 3 | — | |
MDOANUHLWYXBTL
|
8.4 | IC50 | 3 | — | |
MPJFEYNSRDQXTR
|
8.4 | IC50 | 5 | — | |
MRHRUXQFKYBZBW
|
8.4 | IC50 | 3 | — | |
NVWPJAMSFZHMRS
|
8.4 | IC50 | 3 | — | |
ONINVXNOMWDCJH
|
8.4 | IC50 | 3 | — | |
PYUIBNGQBBAKFO
|
8.4 | IC50 | 7 | Yes | |
QTQBJRCBSLLTBA
|
8.4 | IC50 | 3 | — | |
QTQBJRCBSLLTBA
|
8.4 | IC50 | 3 | — | |
RDFNGKQMOZKREL
|
8.4 | IC50 | 3 | — | |
RHLRQFRHMLTKDY
|
8.4 | IC50 | 2 | — | |
STINDBVFOPRZHE
|
8.4 | IC50 | 8 | Yes | |
UAFNMQXZNBBJQS
|
8.4 | IC50 | 3 | — | |
WCIAPCXKGZRGFQ
|
8.4 | IC50 | 5 | — | |
WFESDNSPSXROQT
|
8.4 | IC50 | 3 | — | |
XWRLHVWTHQFHSY
|
8.4 | IC50 | 5 | — | |
YPSGPGKTXWJQKA
|
8.4 | IC50 | 5 | — | |
YQSKZEBWBPKMIQ
|
8.4 | IC50 | 3 | — | |
YZRLWPBYTMKRQR
|
8.4 | IC50 | 11 | — | |
KXTGQCBCZZJSHS
|
8.4 | IC50 | 5 | — | |
NYYKCMGNIZNHAN
|
8.4 | IC50 | 5 | — | |
UHSDGQHRNMRTLI
|
8.4 | IC50 | 5 | — | |
AVEPOXATJSYYGP
|
8.4 | IC50 | 5 | — | |
IWBVZILESKBVJL
|
8.4 | IC50 | 6 | — | |
JBXLEBAVNPBBTP
|
8.4 | Kd | 3 | — | |
MXHREEFYRGHUCY
|
8.4 | IC50 | 5 | — | |
SXKYHAHPQBODAA
|
8.4 | IC50 | 5 | — | |
ZELUDNIRCNOVHB
|
8.4 | IC50 | 2 | — | |
FBKIPMHVNJQANW
|
8.4 | IC50 | 3 | — | |
KIDZNCKPIJZGHH
|
8.4 | IC50 | 5 | — | |
OOWSKBMTGLHFAR
|
8.4 | IC50 | 5 | — | |
PKDVKKBPKSYAPH
|
8.4 | IC50 | 3 | — | |
PRQYUAHLKCIUTM
|
8.4 | IC50 | 5 | — | |
QGWHVBBKJAQYRM
|
8.4 | IC50 | 4 | — |