Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JTIMRSSBBONYGV
|
8.4 | IC50 | 5 | — | |
KPQQBBDCGUBBFQ
|
8.4 | IC50 | 5 | — | |
OPRRDMNWSFSACR
|
8.4 | IC50 | 5 | — | |
QJZANLWCNGSFGW
|
8.4 | IC50 | 5 | — | |
UOWDVWIHJKFQPY
|
8.4 | IC50 | 5 | — | |
UXRRRYIVIGHOBW
|
8.4 | IC50 | 5 | — | |
WSEXAZBKZQGSDN
|
8.4 | IC50 | 5 | — | |
ZNKBNXVWLPQHKJ
|
8.4 | IC50 | 5 | — | |
ZXCGLXZIDVIUJE
|
8.4 | IC50 | 5 | — | |
BCOJIDFRCFXQSL
|
8.4 | IC50 | 3 | — | |
BYCZXBZXUBUKGX
|
8.4 | IC50 | 2 | — | |
JPCRGCMZCOBSNE
|
8.4 | IC50 | 3 | — | |
MHHLXYGRKUMXPW
|
8.4 | IC50 | 2 | — | |
MJHFGTHWKHPARC
|
8.4 | IC50 | 5 | — | |
OQWGMALEKOUCHV
|
8.4 | IC50 | 5 | — | |
QTZWCECBLKRZBR
|
8.4 | IC50 | 4 | — | |
SYVJHJOWIMUQMA
|
8.4 | IC50 | 5 | — | |
BPADCCSYOOULLP
|
8.4 | IC50 | 5 | — | |
CMMUVKONDKDCCZ
|
8.4 | IC50 | 5 | — | |
COMXNOYVEFLSSH
|
8.4 | IC50 | 3 | — | |
CUSVCRYSGDMLAF
|
8.4 | IC50 | 3 | — | |
DLLAXFDTFVKUAV
|
8.4 | IC50 | 2 | — | |
DWXMGHZIWRZUMA
|
8.4 | IC50 | 3 | — | |
FXWYSUDYIQPVOJ
|
8.4 | IC50 | 5 | — | |
JWSLDBSDJDFRSK
|
8.4 | IC50 | 5 | — | |
LLWAEGOAXVEIMG
|
8.4 | IC50 | 5 | — | |
LYDRTKDNCXYTQA
|
8.4 | IC50 | 5 | — | |
MDPWQSCOLLDWIY
|
8.4 | IC50 | 5 | — | |
MLUFVERLBQGOEV
|
8.4 | IC50 | 5 | — | |
NIKYJDORPJPERE
|
8.4 | IC50 | 5 | — | |
OCKLCHHQTFDHGO
|
8.4 | IC50 | 2 | — | |
QCVYUGLDSRBVIC
|
8.4 | IC50 | 3 | — | |
QTGVMULYBGRVHT
|
8.4 | IC50 | 5 | — | |
RHIYIXKVGFLFDX
|
8.4 | IC50 | 2 | — | |
UGADWCXPZTYDIJ
|
8.4 | IC50 | 2 | — | |
AWNNYXYBCDYFFX
|
8.4 | IC50 | 5 | — | |
DDNOUEXAVDQPMR
|
8.4 | IC50 | 5 | — | |
MLWCCXUMKLCBTL
|
8.4 | IC50 | 5 | — | |
NYYKCMGNIZNHAN
|
8.4 | IC50 | 5 | — | |
OEIJEWDFQMITII
|
8.4 | IC50 | 5 | — | |
RMVONVMXMXKGPN
|
8.4 | IC50 | 5 | — | |
ZEONLOUAYWYGAS
|
8.4 | IC50 | 5 | — | |
COLZQIUHTLJTII
|
8.4 | IC50 | 3 | — | |
GRJFVVYLSWWNRI
|
8.4 | IC50 | 2 | — | |
HHRGGSVSAUUCLO
|
8.4 | IC50 | 5 | — | |
HPCVPAAIFAFKQL
|
8.4 | IC50 | 5 | — | |
IOKLYXDNQOPONA
|
8.4 | IC50 | 3 | — | |
MVUTVOTUBKSFAZ
|
8.4 | IC50 | 5 | — | |
OOWSKBMTGLHFAR
|
8.4 | IC50 | 5 | — | |
SDEGOUSDMNTQQS
|
8.4 | IC50 | 5 | — |