Target Details
| UniProt AC | P21802 |
|---|---|
| Gene Symbol | FGFR2 |
| Protein Name | Fibroblast growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,130
- Clinical molecules 64
- Avg pChEMBL 7.82
KEGG Pathways (13)
- Calcium signaling pathway
- Central carbon metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Gastric cancer
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Associated Diseases (12)
- Antley-Bixler syndrome
- Apert syndrome
- Beare-Stevenson syndrome
- Bent bone dysplasia syndrome
- Crouzon syndrome
- Gastric cancer
- Jackson-Weiss syndrome
- Lacrimo-auriculo-dento-digital syndrome
- Pfeiffer syndrome
- Saethre-Chotzen syndrome
- Scaphocephaly, maxillary retrusion, and impaired intellectual development
- Syndromic craniosynostoses
Active Molecules (2,130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QQZSRHQZWOITQR
|
10.0 | IC50 | 4 | — | |
MXSDIGYURCYKOV
|
9.9 | IC50 | 5 | — | |
LHWABYLWRJNIIY
|
9.8 | IC50 | 7 | — | |
HRSOTZFHFDXFAE
|
9.7 | IC50 | 5 | — | |
XGJBIMKIGAOMPJ
|
9.7 | IC50 | 3 | — | |
YYMGAHUGGLEVAR
|
9.7 | IC50 | 4 | — | |
DDHPDOGCZLIDPA
|
9.6 | IC50 | 4 | — | |
FHYRHQXTHUGBJV
|
9.6 | IC50 | 4 | — | |
QUDUPSBANJZEIW
|
9.5 | IC50 | 4 | — | |
FVBNNGBLKUMCEF
|
9.5 | IC50 | 3 | — | |
MPYUMMWCLQVMLG
|
9.5 | IC50 | 11 | — | |
UXYDXGKJWBUZOQ
|
9.5 | IC50 | 4 | — | |
ZKKBDZUWZDKUIQ
|
9.5 | IC50 | 2 | — | |
WFLAIALBWODQSL
|
9.4 | IC50 | 2 | — | |
OCMFTUJIRAAZFF
|
9.4 | IC50 | 5 | — | |
CGXQXIOHFLFFRH
|
9.4 | IC50 | 4 | — | |
LCEOGRIPTKTUOV
|
9.4 | IC50 | 4 | — | |
TWFUXWGJXASISK
|
9.3 | IC50 | 2 | — | |
HCDMJFOHIXMBOV
|
9.3 | IC50 | 4 | — | |
LPQUYUMWALKVKH
|
9.3 | IC50 | 2 | — | |
QHCGPJPIPKDWAT
|
9.3 | IC50 | 8 | — | |
XSFHSBDHUMMKQC
|
9.3 | IC50 | 4 | — | |
CEYCXVCSPGUEPS
|
9.3 | IC50 | 2 | — | |
SBMIDSNPTHVUMU
|
9.3 | IC50 | 2 | — | |
ZKKMRDODNGIIGF
|
9.3 | IC50 | 2 | — | |
QEOFKIKDUSYLPY
|
9.3 | IC50 | 2 | — | |
YRBAKPVAQIOONM
|
9.3 | IC50 | 2 | — | |
GJPKPBGGTZOMIL
|
9.2 | IC50 | 2 | — | |
FFMFQCPBWNBRTM
|
9.2 | IC50 | 2 | — | |
JTFVQKRKLOURMQ
|
9.2 | IC50 | 2 | — | |
FMGRQWRWTCYNKA
|
9.2 | IC50 | 5 | — | |
PTNPCFXETPRXSF
|
9.2 | IC50 | 3 | — | |
VDZZYOJYLLNBTD
|
9.2 | IC50 | 4 | — | |
HUVVCRLMPWOMJX
|
9.2 | IC50 | 4 | — | |
CGGIZDLKLSTLFH
|
9.2 | IC50 | 2 | — | |
PTTBIZQLFMRTIQ
|
9.2 | IC50 | 2 | — | |
CTUHAAWNNBQIDY
|
9.2 | IC50 | 4 | — | |
LGWVEHCWSZKUPK
|
9.2 | IC50 | 4 | — | |
OCIIUHMXXRNNNL
|
9.2 | IC50 | 2 | — | |
UDMCHVHNRKDUMF
|
9.2 | IC50 | 3 | — | |
YISJWEXLNFHRNW
|
9.2 | IC50 | 4 | — | |
MRSOJHDLCLHTOL
|
9.1 | IC50 | 5 | — | |
DFYOEDRVJUNFKB
|
9.1 | IC50 | 2 | — | |
CYSLQXJWRTXVKS
|
9.1 | IC50 | 2 | — | |
LGDDCZVVBAYDDI
|
9.1 | IC50 | 2 | — | |
YXTHFMOUCQZVJH
|
9.1 | IC50 | 3 | — | |
ZMYXCQOKPQVAIY
|
9.1 | IC50 | 4 | — | |
AYMIOSAGFUFSMC
|
9.1 | IC50 | 4 | — | |
TUFWCZFZSQLLMZ
|
9.1 | IC50 | 4 | — | |
YHIGPAIFBVOPKV
|
9.1 | IC50 | 4 | — |