Target Details
UniProt ACP21731
Gene SymbolTBXA2R
Protein NameThromboxane A2 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 286
  • Clinical molecules 6
  • Avg pChEMBL 7.02
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (286)
InChIKey pChEMBL Type Targets Clinical
PHEUETCAYVRPIK 7.3 IC50 2
QTOGSJCFEGPTJN 7.3 IC50 2
QTOGSJCFEGPTJN 7.3 IC50 2
OCLFNCNUYRWKPS 7.2 IC50 2
VDSYMHSEFRKHET 7.2 Kd 2
ZJZSLRMNGAAIAC 7.2 IC50 2
CDEOOMRKYGZADT 7.2 IC50 2
MMDSGIVIWHELNX 7.2 IC50 2
SBJWASMXBSBHSJ 7.2 Ki 3
SAKWDHBZKHMQPN 7.2 Kd 2
LACPPBQCKQXQIH 7.2 Kd 2
LNPWCFLOKKYSBZ 7.2 Ki 2
LOPWWKRHBBYKSR 7.2 IC50 2
HQAGYVZFEKMBFE 7.1 IC50 2
SXIFZKGCEZUKRA 7.1 Kd 2
DSIPHKLHGKYYCB 7.1 IC50 2
DSIPHKLHGKYYCB 7.1 IC50 2
RFHFLABUEIMYLC 7.1 Ki 2
GLEGXNCPSWSVAL 7.1 Ki 2
KWCSGHGCXOSYQY 7.1 Ki 3
CPFQQGFWCIINTC 7.1 IC50 2
PVQYCYOIOKLQMP 7.1 IC50 2
PVQYCYOIOKLQMP 7.1 IC50 2
DOIVAJMCRLNJKI 7.1 Kd 2
OXTRWYUMANEPHR 7.1 IC50 2
RMDNILWXZXFTSB 7.1 IC50 2
JTCXJAJLGOTNRH 7.1 Kd 2
LSPSJQUSSWRPTE 7.1 Ki 2
NMJYFIAGWNELHF 7.1 IC50 2
PXFUYKMANFDTAA 7.1 Ki 2
NEJDMJAJYOXVJF 7.0 IC50 2
UZGOIKLVDRHFFW 7.0 Ki 2
WRMLVALLVQNILX 7.0 Ki 2
ZXBHFWFKSIYJEK 7.0 IC50 3
BRGRVTXBZSDTQZ 7.0 Ki 2
FVCQVNNARRQDCP 7.0 IC50 2
KGFDNQQQBPWRCG 7.0 Ki 2
RRDVGFBNUNMAKI 7.0 Ki 2
ZHBPUNZHLIFKIH 7.0 Kd 2
IBCFVGVAMLZBIX 7.0 Ki 2
FMGMZPGNRHRJQC 7.0 Kd 2
SRGNPNSJCLBDOM 7.0 IC50 2
SRGNPNSJCLBDOM 7.0 IC50 2
RISLJJMLXCMMAD 7.0 Ki 2
XJKMOZFCIYEDDT 7.0 Kd 2
CPHBHPJSMLOFHV 6.9 IC50 2
MRBWBFJXHIUJNQ 6.9 Ki 2
STXGLNVWWYTFOV 6.9 Kd 2
UASKRIFPIWYGAQ 6.9 Kd 2
UEBOELMCZQDCEI 6.9 IC50 2
2D structure